BR0109885A - Moléculas duais, processo de preparação das mesmas, composições farmacêuticas, e, utilização das moléculas duais - Google Patents
Moléculas duais, processo de preparação das mesmas, composições farmacêuticas, e, utilização das moléculas duaisInfo
- Publication number
- BR0109885A BR0109885A BR0109885-3A BR0109885A BR0109885A BR 0109885 A BR0109885 A BR 0109885A BR 0109885 A BR0109885 A BR 0109885A BR 0109885 A BR0109885 A BR 0109885A
- Authority
- BR
- Brazil
- Prior art keywords
- dual molecules
- dual
- pharmaceutical compositions
- molecules
- preparing same
- Prior art date
Links
- 230000009977 dual effect Effects 0.000 title abstract 5
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 abstract 2
- 230000000078 anti-malarial effect Effects 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 150000007513 acids Chemical class 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 150000001408 amides Chemical class 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 230000027326 copulation Effects 0.000 abstract 1
- -1 cyclic peroxide Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 125000003367 polycyclic group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229940124530 sulfonamide Drugs 0.000 abstract 1
- 150000003456 sulfonamides Chemical class 0.000 abstract 1
- 150000003568 thioethers Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D323/00—Heterocyclic compounds containing more than two oxygen atoms as the only ring hetero atoms
- C07D323/04—Six-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
"MOLéCULAS DUAIS, PROCESSO DE PREPARAçãO DAS MESMAS, COMPOSIçõES FARMACêUTICAS, E, UTILIZAçãO DAS MOLéCULAS DUAIS". A invenção visa moléculas duais formadas de produtos de copulação com um resíduo de molécula com atividade anti-palúdica, 1 ou 2 cadeias alquileno em C1 a C5, compreendendo uma função amina, amida, sulfonamida, carboxila, éter ou tioéter, assegurando a ligação entre as 2 cadeias, uma estrutura policíclica ligada a um peróxido cíclico de 4 a 8 membros, e seus sais de adição com os ácidos farmacologicamente aceitáveis. Aplicação como medicamento com atividade anti-palúdica.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0004422A FR2807433B1 (fr) | 2000-04-06 | 2000-04-06 | Molecules duales contenant un derives peroxydique, leur synthese et leurs applications therapeutiques |
| PCT/FR2001/001013 WO2001077105A1 (fr) | 2000-04-06 | 2001-04-04 | Molecules duales contenant un derive peroxydique, leur synthese et leurs applications therapeutiques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0109885A true BR0109885A (pt) | 2003-06-03 |
Family
ID=8848956
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0109885-3A BR0109885A (pt) | 2000-04-06 | 2001-04-04 | Moléculas duais, processo de preparação das mesmas, composições farmacêuticas, e, utilização das moléculas duais |
Country Status (27)
| Country | Link |
|---|---|
| US (2) | US6949569B2 (pt) |
| EP (1) | EP1268470B1 (pt) |
| JP (1) | JP2004521855A (pt) |
| KR (1) | KR100832047B1 (pt) |
| CN (1) | CN1193028C (pt) |
| AP (1) | AP1399A (pt) |
| AR (1) | AR041773A1 (pt) |
| AT (1) | ATE387441T1 (pt) |
| AU (2) | AU4846301A (pt) |
| BR (1) | BR0109885A (pt) |
| CA (1) | CA2405076C (pt) |
| CY (1) | CY1108071T1 (pt) |
| DE (1) | DE60132981T2 (pt) |
| DK (1) | DK1268470T3 (pt) |
| ES (1) | ES2302727T3 (pt) |
| FR (1) | FR2807433B1 (pt) |
| HU (1) | HUP0300428A2 (pt) |
| IL (2) | IL151918A0 (pt) |
| IS (1) | IS6579A (pt) |
| MX (1) | MXPA02009856A (pt) |
| MY (1) | MY128443A (pt) |
| NO (1) | NO329526B1 (pt) |
| NZ (1) | NZ521774A (pt) |
| OA (1) | OA13294A (pt) |
| PT (1) | PT1268470E (pt) |
| WO (1) | WO2001077105A1 (pt) |
| ZA (1) | ZA200207851B (pt) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2862304A1 (fr) * | 2003-11-14 | 2005-05-20 | Centre Nat Rech Scient | Molecules duales racemiques ou achirales contenant un derive peroxydique, leur synthese et leurs applications therapeutiques |
| TW200728315A (en) * | 2005-12-06 | 2007-08-01 | Nippon Chemical Ind | Phosphorus transition-metal complex, method of producing the same, and anticancer agent forming the same |
| FR2902100A1 (fr) * | 2006-06-13 | 2007-12-14 | Sanofi Aventis Sa | Molecules duales contenant un derive peroxydique, leur synthese et leurs applications en therapeutique |
| FR2924343A1 (fr) * | 2007-12-04 | 2009-06-05 | Palumed Sa | Nouvelles utilisations therapeutiques de molecules duales contenant un derive peroxydique. |
| US9018409B2 (en) * | 2010-10-27 | 2015-04-28 | Meurice R&D Asbl | Process for functionalization of unsaturated compounds |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT876346E (pt) * | 1995-11-16 | 2002-01-30 | Hoffmann La Roche | Derivados de quinolina com actividade anti-malaria |
-
2000
- 2000-04-06 FR FR0004422A patent/FR2807433B1/fr not_active Expired - Fee Related
-
2001
- 2001-04-04 JP JP2001575578A patent/JP2004521855A/ja active Pending
- 2001-04-04 AU AU4846301A patent/AU4846301A/xx active Pending
- 2001-04-04 IL IL15191801A patent/IL151918A0/xx unknown
- 2001-04-04 AP APAP/P/2002/002646A patent/AP1399A/en active
- 2001-04-04 ES ES01921476T patent/ES2302727T3/es not_active Expired - Lifetime
- 2001-04-04 CA CA2405076A patent/CA2405076C/fr not_active Expired - Fee Related
- 2001-04-04 OA OA1200200308A patent/OA13294A/fr unknown
- 2001-04-04 MX MXPA02009856A patent/MXPA02009856A/es active IP Right Grant
- 2001-04-04 CN CNB018088066A patent/CN1193028C/zh not_active Expired - Fee Related
- 2001-04-04 PT PT01921476T patent/PT1268470E/pt unknown
- 2001-04-04 AU AU2001248463A patent/AU2001248463B2/en not_active Ceased
- 2001-04-04 HU HU0300428A patent/HUP0300428A2/hu unknown
- 2001-04-04 AT AT01921476T patent/ATE387441T1/de active
- 2001-04-04 US US10/240,929 patent/US6949569B2/en not_active Expired - Fee Related
- 2001-04-04 DK DK01921476T patent/DK1268470T3/da active
- 2001-04-04 BR BR0109885-3A patent/BR0109885A/pt not_active IP Right Cessation
- 2001-04-04 WO PCT/FR2001/001013 patent/WO2001077105A1/fr not_active Ceased
- 2001-04-04 EP EP01921476A patent/EP1268470B1/fr not_active Expired - Lifetime
- 2001-04-04 NZ NZ521774A patent/NZ521774A/en not_active IP Right Cessation
- 2001-04-04 KR KR1020027013363A patent/KR100832047B1/ko not_active Expired - Fee Related
- 2001-04-04 DE DE60132981T patent/DE60132981T2/de not_active Expired - Lifetime
- 2001-04-06 AR ARP010101655A patent/AR041773A1/es not_active Application Discontinuation
- 2001-04-06 MY MYPI20011659A patent/MY128443A/en unknown
-
2002
- 2002-09-25 IL IL151918A patent/IL151918A/en not_active IP Right Cessation
- 2002-09-30 ZA ZA200207851A patent/ZA200207851B/en unknown
- 2002-10-03 IS IS6579A patent/IS6579A/is unknown
- 2002-10-04 NO NO20024795A patent/NO329526B1/no not_active IP Right Cessation
-
2005
- 2005-08-04 US US11/196,979 patent/US7566710B2/en not_active Expired - Fee Related
-
2008
- 2008-05-26 CY CY20081100544T patent/CY1108071T1/el unknown
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
| B07F | Notification of approval that there is no relation to art. 229 of lpi (pipeline patents) [chapter 7.6 patent gazette] |
Free format text: NOTIFICACAO DE NAO ANUENCIA RELACIONADA COM O ART. 229 DA LPI |
|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 13A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2258 DE 15/04/2014. |