BR0203501A - Formulações de multipartìculas biomoduladas - Google Patents
Formulações de multipartìculas biomoduladasInfo
- Publication number
- BR0203501A BR0203501A BR0203501-4A BR0203501A BR0203501A BR 0203501 A BR0203501 A BR 0203501A BR 0203501 A BR0203501 A BR 0203501A BR 0203501 A BR0203501 A BR 0203501A
- Authority
- BR
- Brazil
- Prior art keywords
- formulations
- biomodulated
- multiparticle
- multiparticle formulations
- release rate
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 4
- 238000009472 formulation Methods 0.000 title abstract 3
- OJRHUICOVVSGSY-RXMQYKEDSA-N (2s)-2-chloro-3-methylbutan-1-ol Chemical compound CC(C)[C@H](Cl)CO OJRHUICOVVSGSY-RXMQYKEDSA-N 0.000 abstract 1
- 229960001770 atorvastatin calcium Drugs 0.000 abstract 1
- 239000002775 capsule Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/485—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1611—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Obesity (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
Abstract
"FORMULAçõES DE MULTIPARTìCULAS BIOMODULADAS". A presente invenção refere-se com os meios para ajuste da biodisponibilidade da atorvastatina de cálcio por modulação da sua taxa de liberação de formulações de multipartículas e com formulações de multipartículas, especialmente comprimidos e cápsulas, tendo a referida taxa de liberação modulada.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0121436.0A GB0121436D0 (en) | 2001-09-04 | 2001-09-04 | Biomodulated multiparticulate formulations |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0203501A true BR0203501A (pt) | 2003-05-20 |
Family
ID=9921522
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0203501-4A BR0203501A (pt) | 2001-09-04 | 2002-08-30 | Formulações de multipartìculas biomoduladas |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP1287821A1 (pt) |
| JP (1) | JP2003128544A (pt) |
| BR (1) | BR0203501A (pt) |
| CA (1) | CA2400565A1 (pt) |
| GB (1) | GB0121436D0 (pt) |
| MX (1) | MXPA02008059A (pt) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030190343A1 (en) * | 2002-03-05 | 2003-10-09 | Pfizer Inc. | Palatable pharmaceutical compositions for companion animals |
| CA2465693A1 (en) * | 2003-06-12 | 2004-12-12 | Warner-Lambert Company Llc | Pharmaceutical compositions of atorvastatin |
| JP3821139B2 (ja) * | 2004-05-14 | 2006-09-13 | コニカミノルタビジネステクノロジーズ株式会社 | データ出力システム、およびデータ出力装置 |
| EP1825848A3 (de) * | 2006-02-10 | 2010-03-03 | Stada Arzneimittel Ag | Stabile pharmazeutische Zusammensetzungen umfassend einen HMG-CoA-Reduktase Inhibitor |
| EP1818050A1 (de) * | 2006-02-10 | 2007-08-15 | Stada Arzneimittel Ag | Stabile pharmazeutische Zusammensetzungen umfassend einen HMG-CoA-Reduktase Inhibitor |
| BRPI0920170A2 (pt) | 2008-10-17 | 2016-06-21 | Metabolex Inc | métodos para diminuir a quantidade de partículas ldl pequenas e densas e de níveis de triglicerídeos e ldl no sangue em um humano, e para identificar um indivíduo candidato para tratamento com um composto ou um sal, prodroga ou isômero do mesmo, composto ou um sal, prodroga ou isômero do mesmo, e método. |
| WO2010093285A1 (en) * | 2009-02-12 | 2010-08-19 | Aduro Material Ab | Composition comprising biodegradable carrier for controlled drug delivery |
| WO2012042951A1 (ja) * | 2010-09-30 | 2012-04-05 | アステラス製薬株式会社 | アトルバスタチン含有医薬錠剤 |
| JP2013231011A (ja) * | 2012-05-01 | 2013-11-14 | Sawai Pharmaceutical Co Ltd | アトルバスタチン含有医薬組成物およびそれを用いた口腔内崩壊錠 |
| CN108421045B (zh) * | 2018-04-02 | 2021-09-24 | 北京海晶生物医药科技有限公司 | 一种阿托伐他汀钙组合物、制剂及其制备方法 |
| CN110151721B (zh) * | 2019-06-10 | 2021-11-12 | 乐普制药科技有限公司 | 一种含有阿托伐他汀钙的片剂及其制备方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI94339C (fi) * | 1989-07-21 | 1995-08-25 | Warner Lambert Co | Menetelmä farmaseuttisesti käyttökelpoisen /R-(R*,R*)/-2-(4-fluorifenyyli)- , -dihydroksi-5-(1-metyylietyyli)-3-fenyyli-4-/(fenyyliamino)karbonyyli/-1H-pyrroli-1-heptaanihapon ja sen farmaseuttisesti hyväksyttävien suolojen valmistamiseksi |
| JP3254219B2 (ja) * | 1993-01-19 | 2002-02-04 | ワーナー−ランバート・コンパニー | 安定な経口用のci−981製剤およびその製法 |
| US6248363B1 (en) * | 1999-11-23 | 2001-06-19 | Lipocine, Inc. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
| EP1272181A2 (en) * | 2000-04-13 | 2003-01-08 | Synthon B.V. | Modified release formulations containing a hypnotic agent |
-
2001
- 2001-09-04 GB GBGB0121436.0A patent/GB0121436D0/en not_active Ceased
-
2002
- 2002-08-19 MX MXPA02008059A patent/MXPA02008059A/es active IP Right Grant
- 2002-08-21 EP EP02255847A patent/EP1287821A1/en not_active Withdrawn
- 2002-08-30 BR BR0203501-4A patent/BR0203501A/pt not_active IP Right Cessation
- 2002-08-30 CA CA002400565A patent/CA2400565A1/en not_active Abandoned
- 2002-09-04 JP JP2002258464A patent/JP2003128544A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EP1287821A1 (en) | 2003-03-05 |
| CA2400565A1 (en) | 2003-03-04 |
| JP2003128544A (ja) | 2003-05-08 |
| MXPA02008059A (es) | 2003-04-09 |
| GB0121436D0 (en) | 2001-10-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE 7A. E 8A. ANUIDADE(S). |
|
| B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: REFERENTE AO DESPACHO PUBLICADO NA RPI 2103 DE 26/04/2011. |