BR112012014683A2 - processo para a produção de derivados de ácido 1-alquil/1-aril-5-pirazolcarboxílico - Google Patents

processo para a produção de derivados de ácido 1-alquil/1-aril-5-pirazolcarboxílico

Info

Publication number
BR112012014683A2
BR112012014683A2 BR112012014683A BR112012014683A BR112012014683A2 BR 112012014683 A2 BR112012014683 A2 BR 112012014683A2 BR 112012014683 A BR112012014683 A BR 112012014683A BR 112012014683 A BR112012014683 A BR 112012014683A BR 112012014683 A2 BR112012014683 A2 BR 112012014683A2
Authority
BR
Brazil
Prior art keywords
aryl
alkyl
production
acid derivatives
substituted
Prior art date
Application number
BR112012014683A
Other languages
English (en)
Other versions
BR112012014683B1 (pt
Inventor
Igor Gerus
Norbert Lui
Sergii Pazenok
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR112012014683A2 publication Critical patent/BR112012014683A2/pt
Publication of BR112012014683B1 publication Critical patent/BR112012014683B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/30—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

patente de invenção. processo para a produção de derivados de ácido 1-alquil-/1 arik-5-pirazilcarboxílico. a presente invenção se refere a um processo para a produção de derivados de ácido 5-pirazolcarboxílico 1-alquil ou 1-aril- substituídos, compreendendo a reação de 1,3-dioxolanos e 1,4-dioxanos substituídos com aquil- ou aril-hridrozinas para dihidro-1h-pirazóis 1-alquil- ou 1-aril+ substituídos, bem como a sua ulterior reação para derivados de ácido 5-pirazolcarboxílico 1-alquil ou 1-aril- substituídos, os quais podem encontrar uso como valiosos produtos intermediários para a produção de amidas de ácido antranílico de ação inseticida.
BR112012014683-1A 2009-12-15 2010-12-10 Process for the production of 5-pyrazolcarboxylic acid derivatives 1-alkyl- / 1-aryl-substituted and compound acid BR112012014683B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09179299.4 2009-12-15
EP09179299 2009-12-15
PCT/EP2010/069385 WO2011073101A1 (de) 2009-12-15 2010-12-10 Verfahren zur herstellung von 1-alkyl-/1-aryl-5-pyrazolcarbonsäurederivaten

Publications (2)

Publication Number Publication Date
BR112012014683A2 true BR112012014683A2 (pt) 2015-09-15
BR112012014683B1 BR112012014683B1 (pt) 2017-11-07

Family

ID=41569911

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012014683-1A BR112012014683B1 (pt) 2009-12-15 2010-12-10 Process for the production of 5-pyrazolcarboxylic acid derivatives 1-alkyl- / 1-aryl-substituted and compound acid

Country Status (12)

Country Link
US (1) US8586753B2 (pt)
EP (1) EP2513063B1 (pt)
JP (1) JP5753856B2 (pt)
KR (1) KR101758201B1 (pt)
CN (1) CN102753531B (pt)
BR (1) BR112012014683B1 (pt)
DK (1) DK2513063T3 (pt)
ES (1) ES2437923T3 (pt)
IL (1) IL220211A (pt)
MX (1) MX2012006723A (pt)
TW (1) TWI504590B (pt)
WO (1) WO2011073101A1 (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5753855B2 (ja) * 2009-12-15 2015-07-22 バイエル・クロップサイエンス・アーゲーＢａｙｅｒ Ｃｒｏｐｓｃｉｅｎｃｅ Ａｇ 新規ジオキソラン及びジオキサン誘導体並びにそれらを製造する方法
MX2014000318A (es) 2011-07-08 2014-02-19 Bayer Ip Gmbh Procedimiento de preparacion de derivados de diamida del acido antranilico sustituidos con tetrazol mediante la reaccion de acidos de pirazol con esteres antranilicos.
MX349771B (es) 2011-08-26 2017-08-10 Bayer Ip Gmbh Procedimiento para preparar derivados de diamida de acido antranilico sustituida con tetrazol haciendo reaccionar benzoxazinonas con aminas.
CN109689629B (zh) * 2016-09-21 2022-11-29 拜耳作物科学股份公司 制备3-氟烷基-5-吡唑羧酸酯和3-氟烷基-5-吡唑羧酸的方法
WO2019224678A1 (en) 2018-05-21 2019-11-28 Pi Industries Ltd. A novel process for the preparation of anthranilic diamides
MX2021000226A (es) 2018-07-20 2021-03-31 Pi Industries Ltd Nuevo proceso para la preparacion de diamidas antranilicas.
CN116134023A (zh) * 2020-07-23 2023-05-16 拜耳公司 制备氨基呋喃的方法
US20240010626A1 (en) * 2020-10-06 2024-01-11 Bayer Aktiengesellschaft Method for producing carbonylaminofurans
EP4376616A1 (en) 2021-07-27 2024-06-05 Syngenta Crop Protection AG Method for controlling diamide resistant pests & compounds therefor
US20240308988A1 (en) 2021-08-05 2024-09-19 Syngenta Crop Protection Ag Method For Controlling Diamide Resistant Pests and Compounds Therefor
WO2023110710A1 (en) 2021-12-13 2023-06-22 Syngenta Crop Protection Ag Method for controlling diamide resistant pests & compounds therefor
EP4197333A1 (en) 2021-12-15 2023-06-21 Syngenta Crop Protection AG Method for controlling diamide resistant pests & compounds therefor
WO2024133426A1 (en) 2022-12-21 2024-06-27 Syngenta Crop Protection Ag Method for controlling diamide resistant pests and compounds therefor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW438796B (en) * 1996-05-15 2001-06-07 Hoffmann La Roche 2,4-diaminopyrimidine derivatives, the manufacture process thereof, and the antibiotically-active pharmaceutical composition containing the same
KR20010013977A (ko) 1997-06-19 2001-02-26 블레어 큐. 퍼거슨 중성 ｐ1 특이성 기를 갖는 인자 ｘａ의 억제제
TWI327566B (en) * 2001-08-13 2010-07-21 Du Pont Novel substituted ihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use
DE60236600D1 (de) 2001-08-13 2010-07-15 Du Pont Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung
SI1599463T1 (sl) * 2003-01-28 2013-10-30 E.I. Du Pont De Nemours And Company Ciano antranilamidni insekticidi
TW200526588A (en) * 2003-11-17 2005-08-16 Smithkline Beecham Corp Chemical compounds
DE102006032168A1 (de) 2006-06-13 2007-12-20 Bayer Cropscience Ag Anthranilsäurediamid-Derivate mit heteroaromatischen Substituenten
EP2243777A1 (de) * 2009-04-03 2010-10-27 Bayer CropScience AG Verfahren zum Herstellen von Pyridyl-substituierten Pyrazolen
JP5753855B2 (ja) * 2009-12-15 2015-07-22 バイエル・クロップサイエンス・アーゲーＢａｙｅｒ Ｃｒｏｐｓｃｉｅｎｃｅ Ａｇ 新規ジオキソラン及びジオキサン誘導体並びにそれらを製造する方法

Also Published As

Publication number Publication date
KR20120096078A (ko) 2012-08-29
TW201144288A (en) 2011-12-16
CN102753531A (zh) 2012-10-24
US20110152532A1 (en) 2011-06-23
JP2013513635A (ja) 2013-04-22
CN102753531B (zh) 2015-07-01
EP2513063A1 (de) 2012-10-24
IL220211A (en) 2016-02-29
TWI504590B (zh) 2015-10-21
ES2437923T3 (es) 2014-01-15
DK2513063T3 (da) 2014-01-06
IL220211A0 (en) 2012-07-31
EP2513063B1 (de) 2013-11-06
MX2012006723A (es) 2012-06-28
KR101758201B1 (ko) 2017-07-14
BR112012014683B1 (pt) 2017-11-07
WO2011073101A1 (de) 2011-06-23
US8586753B2 (en) 2013-11-19
JP5753856B2 (ja) 2015-07-22

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Legal Events

Date Code Title Description
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 10/12/2010, OBSERVADAS AS CONDICOES LEGAIS.