BR112012024910A2 - composição contendo vesícula e método para sua produção - Google Patents
composição contendo vesícula e método para sua produçãoInfo
- Publication number
- BR112012024910A2 BR112012024910A2 BR112012024910A BR112012024910A BR112012024910A2 BR 112012024910 A2 BR112012024910 A2 BR 112012024910A2 BR 112012024910 A BR112012024910 A BR 112012024910A BR 112012024910 A BR112012024910 A BR 112012024910A BR 112012024910 A2 BR112012024910 A2 BR 112012024910A2
- Authority
- BR
- Brazil
- Prior art keywords
- composition
- vesicle
- present
- water
- gallbladder
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
- A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
- A61K31/375—Ascorbic acid, i.e. vitamin C; Salts thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/02—Cosmetics or similar toiletry preparations characterised by special physical form
- A61K8/14—Liposomes; Vesicles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
- A61K8/36—Carboxylic acids; Salts or anhydrides thereof
- A61K8/361—Carboxylic acids having more than seven carbon atoms in an unbroken chain; Salts or anhydrides thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
- A61K8/37—Esters of carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
- A61K8/37—Esters of carboxylic acids
- A61K8/375—Esters of carboxylic acids the alcohol moiety containing more than one hydroxy group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
- A61K8/44—Aminocarboxylic acids or derivatives thereof, e.g. aminocarboxylic acids containing sulfur; Salts; Esters or N-acylated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/46—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing sulfur
- A61K8/466—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing sulfur containing sulfonic acid derivatives; Salts
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/63—Steroids; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
- A61K8/84—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
- A61K8/86—Polyethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
- A61K8/84—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
- A61K8/89—Polysiloxanes
- A61K8/891—Polysiloxanes saturated, e.g. dimethicone, phenyl trimethicone, C24-C28 methicone or stearyl dimethicone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
- A61K8/84—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
- A61K8/89—Polysiloxanes
- A61K8/891—Polysiloxanes saturated, e.g. dimethicone, phenyl trimethicone, C24-C28 methicone or stearyl dimethicone
- A61K8/894—Polysiloxanes saturated, e.g. dimethicone, phenyl trimethicone, C24-C28 methicone or stearyl dimethicone modified by a polyoxyalkylene group, e.g. cetyl dimethicone copolyol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/127—Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/02—Preparations for care of the skin for chemically bleaching or whitening the skin
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Birds (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Emergency Medicine (AREA)
- Dispersion Chemistry (AREA)
- Dermatology (AREA)
- Cosmetics (AREA)
- Medicinal Preparation (AREA)
Abstract
composição contendo vesícula e método para sua produção. a presente invenção refere-se a uma composição contendo vesículas tendo uma excelente estabilidade na presença de agente medicinal solúvel em água. uma composição contendo vesícula da presente invenção é caracterizada por compreender: (a) um tensoativo à base de silicone, (b) um ou mais tensoativos aniônicos selecionados de éter fosfato de polioxietileno alquila (12 a 15), taurato de acil metila e glutamato de acila, em uma quantidade de 0,001 a 0,2 % em massa, (c) um óleo polar tendo iob de 0,05 a 0,80 e/ou óleo de silicone, e (d) água contendo um agente medicinal solúvel em água em uma quantidade de 0,5 a 5% em massa com base na composição, em que (a) tensoativo com base em silicone forma vesículas; (b) os tensoativos aniônicos se ligam a uma superfície das vesículas; e (c) o óleo polar e/ou óleo de silicone está presente dentro de uma membrana de bicamada das vesículas.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2010082301 | 2010-03-31 | ||
| JP2010220684 | 2010-09-30 | ||
| PCT/JP2011/057378 WO2011122477A1 (ja) | 2010-03-31 | 2011-03-25 | ベシクル含有組成物 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112012024910A2 true BR112012024910A2 (pt) | 2016-07-05 |
Family
ID=44712184
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012024910A BR112012024910A2 (pt) | 2010-03-31 | 2011-03-25 | composição contendo vesícula e método para sua produção |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20130028950A1 (pt) |
| EP (1) | EP2561862B1 (pt) |
| JP (1) | JP4980474B2 (pt) |
| KR (1) | KR101344557B1 (pt) |
| CN (1) | CN102811708B (pt) |
| BR (1) | BR112012024910A2 (pt) |
| ES (1) | ES2546986T3 (pt) |
| RU (1) | RU2517710C1 (pt) |
| TW (1) | TWI412378B (pt) |
| WO (1) | WO2011122477A1 (pt) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5977107B2 (ja) * | 2012-07-18 | 2016-08-24 | 花王株式会社 | ベシクル組成物の製造方法 |
| CN104093392A (zh) * | 2012-02-13 | 2014-10-08 | 花王株式会社 | 囊泡组合物的制造方法 |
| JP5988263B2 (ja) * | 2012-09-18 | 2016-09-07 | 国立大学法人京都大学 | 複数の被内包リポソームを内包するリポソーム及びその製造方法 |
| JP5690373B2 (ja) | 2013-04-26 | 2015-03-25 | 株式会社 資生堂 | 水性組成物 |
| CN103751072B (zh) * | 2014-02-19 | 2015-04-22 | 珀莱雅化妆品股份有限公司 | 一种能恢复皮肤微生态的非离子表面活性剂囊泡及其制备方法 |
| KR101655956B1 (ko) * | 2014-10-30 | 2016-09-08 | 서울과학기술대학교 산학협력단 | 유성 화장품의 제거를 위한 w/o 마이크로에멀전 조성물 |
| KR101664877B1 (ko) * | 2015-06-26 | 2016-10-12 | 주식회사 코리아나화장품 | 니트로지방산을 함유하는 니오좀을 포함하는 화장료 조성물 |
| CN111263628B (zh) * | 2017-10-26 | 2023-09-08 | 株式会社资生堂 | 含囊泡的组合物 |
| PT3700506T (pt) | 2017-10-27 | 2021-09-29 | Xyon Health Inc | Formulações tópicas para tratar distúrbios dermatológicos incluindo calvíce de padrão masculino |
| WO2019235331A1 (ja) * | 2018-06-06 | 2019-12-12 | 株式会社 資生堂 | 部分架橋もしくは架橋型ジメチルポリシロキサンを用いた水中油型乳化化粧料 |
| CN116761579A (zh) * | 2020-12-25 | 2023-09-15 | 株式会社资生堂 | 水包油型乳化化妆品 |
| JP7695825B2 (ja) * | 2021-06-10 | 2025-06-19 | 株式会社 資生堂 | 変臭定量化方法、変臭定量化装置、及び変臭定量化プログラム |
| KR102764695B1 (ko) | 2021-08-05 | 2025-02-11 | (주)아모레퍼시픽 | 난용성 성분이 안정화된 나노베지클을 포함하는 수중유형 화장료 조성물 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5229104A (en) * | 1991-04-29 | 1993-07-20 | Richardson-Vicks Inc. | Artificial tanning compositions containing positively charged paucilamellar vesicles |
| FR2725369B1 (fr) * | 1994-10-07 | 1997-01-03 | Oreal | Composition cosmetique ou dermatologique constituee d'une emulsion huile dans eau a base de globules huileux pourvus d'un enrobage cristal liquide lamellaire |
| JP3483988B2 (ja) * | 1995-06-01 | 2004-01-06 | 株式会社資生堂 | 皮膚外用剤 |
| JP4246980B2 (ja) * | 2001-09-11 | 2009-04-02 | 花王株式会社 | 皮膚外用剤 |
| CN1720021A (zh) * | 2002-12-04 | 2006-01-11 | 陶氏康宁公司 | 基于硅氧烷表面活性剂的极性有机油的泡囊和微乳液组合物 |
| JP2004269430A (ja) * | 2003-03-10 | 2004-09-30 | Ichimaru Pharcos Co Ltd | 毛髪処理用組成物及び損傷毛用毛髪化粧料 |
| US20070243241A1 (en) * | 2004-04-20 | 2007-10-18 | Shaow Lin | Silicone Vesicles Containing Actives |
| US8012387B2 (en) * | 2004-04-20 | 2011-09-06 | Dow Corning Corporation | Silicone vesicles |
| JP4611831B2 (ja) * | 2005-07-26 | 2011-01-12 | 株式会社資生堂 | 油中水型皮膚外用剤 |
| US20080226708A1 (en) * | 2005-11-01 | 2008-09-18 | Shaow Burn Lin | Silicone Vesicles Containing Actives |
| JP5121179B2 (ja) | 2006-07-25 | 2013-01-16 | 株式会社 資生堂 | ベシクル含有組成物及びその製造方法 |
| JP5254645B2 (ja) * | 2007-03-13 | 2013-08-07 | 株式会社コーセー | ベシクル組成物及び該ベシクル組成物を配合した皮膚外用剤 |
| BRPI0811575B1 (pt) | 2007-05-15 | 2016-09-13 | Shiseido Co Ltd | composição contendo vesículas e método de produção da mesma |
| JP2009242326A (ja) * | 2008-03-31 | 2009-10-22 | Shiseido Co Ltd | 美白液状化粧料 |
| JP4395537B2 (ja) * | 2008-04-09 | 2010-01-13 | 株式会社資生堂 | ベシクル及びそれを含む化粧料 |
-
2011
- 2011-03-25 BR BR112012024910A patent/BR112012024910A2/pt not_active IP Right Cessation
- 2011-03-25 EP EP11762708.3A patent/EP2561862B1/en active Active
- 2011-03-25 RU RU2012144575/04A patent/RU2517710C1/ru not_active IP Right Cessation
- 2011-03-25 KR KR1020127027086A patent/KR101344557B1/ko not_active Expired - Fee Related
- 2011-03-25 WO PCT/JP2011/057378 patent/WO2011122477A1/ja not_active Ceased
- 2011-03-25 US US13/637,394 patent/US20130028950A1/en not_active Abandoned
- 2011-03-25 CN CN201180016924.5A patent/CN102811708B/zh active Active
- 2011-03-25 ES ES11762708.3T patent/ES2546986T3/es active Active
- 2011-03-25 JP JP2011067914A patent/JP4980474B2/ja active Active
- 2011-03-29 TW TW100110716A patent/TWI412378B/zh not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| JP4980474B2 (ja) | 2012-07-18 |
| JP2012092084A (ja) | 2012-05-17 |
| EP2561862A1 (en) | 2013-02-27 |
| KR101344557B1 (ko) | 2013-12-26 |
| TWI412378B (zh) | 2013-10-21 |
| HK1175996A1 (en) | 2013-07-19 |
| TW201201849A (en) | 2012-01-16 |
| EP2561862B1 (en) | 2015-08-05 |
| RU2517710C1 (ru) | 2014-05-27 |
| CN102811708B (zh) | 2014-11-05 |
| CN102811708A (zh) | 2012-12-05 |
| US20130028950A1 (en) | 2013-01-31 |
| EP2561862A4 (en) | 2013-10-30 |
| WO2011122477A1 (ja) | 2011-10-06 |
| KR20130040829A (ko) | 2013-04-24 |
| ES2546986T3 (es) | 2015-09-30 |
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| B350 | Update of information on the portal [chapter 15.35 patent gazette] | ||
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