BR112012024910A2 - composição contendo vesícula e método para sua produção - Google Patents

composição contendo vesícula e método para sua produção

Info

Publication number
BR112012024910A2
BR112012024910A2 BR112012024910A BR112012024910A BR112012024910A2 BR 112012024910 A2 BR112012024910 A2 BR 112012024910A2 BR 112012024910 A BR112012024910 A BR 112012024910A BR 112012024910 A BR112012024910 A BR 112012024910A BR 112012024910 A2 BR112012024910 A2 BR 112012024910A2
Authority
BR
Brazil
Prior art keywords
composition
vesicle
present
water
gallbladder
Prior art date
Application number
BR112012024910A
Other languages
English (en)
Inventor
Kei Watanabe
Miharu Nishida
Yuji Matsushita
Original Assignee
Shiseido Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shiseido Co Ltd filed Critical Shiseido Co Ltd
Publication of BR112012024910A2 publication Critical patent/BR112012024910A2/pt

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • A61K31/375Ascorbic acid, i.e. vitamin C; Salts thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/02Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/14Liposomes; Vesicles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/36Carboxylic acids; Salts or anhydrides thereof
    • A61K8/361Carboxylic acids having more than seven carbon atoms in an unbroken chain; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37Esters of carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37Esters of carboxylic acids
    • A61K8/375Esters of carboxylic acids the alcohol moiety containing more than one hydroxy group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A61K8/44Aminocarboxylic acids or derivatives thereof, e.g. aminocarboxylic acids containing sulfur; Salts; Esters or N-acylated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/46Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing sulfur
    • A61K8/466Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing sulfur containing sulfonic acid derivatives; Salts
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/63Steroids; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/72Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
    • A61K8/84Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
    • A61K8/86Polyethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/72Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
    • A61K8/84Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
    • A61K8/89Polysiloxanes
    • A61K8/891Polysiloxanes saturated, e.g. dimethicone, phenyl trimethicone, C24-C28 methicone or stearyl dimethicone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/72Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
    • A61K8/84Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
    • A61K8/89Polysiloxanes
    • A61K8/891Polysiloxanes saturated, e.g. dimethicone, phenyl trimethicone, C24-C28 methicone or stearyl dimethicone
    • A61K8/894Polysiloxanes saturated, e.g. dimethicone, phenyl trimethicone, C24-C28 methicone or stearyl dimethicone modified by a polyoxyalkylene group, e.g. cetyl dimethicone copolyol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/02Preparations for care of the skin for chemically bleaching or whitening the skin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Dispersion Chemistry (AREA)
  • Dermatology (AREA)
  • Cosmetics (AREA)
  • Medicinal Preparation (AREA)

Abstract

composição contendo vesícula e método para sua produção. a presente invenção refere-se a uma composição contendo vesículas tendo uma excelente estabilidade na presença de agente medicinal solúvel em água. uma composição contendo vesícula da presente invenção é caracterizada por compreender: (a) um tensoativo à base de silicone, (b) um ou mais tensoativos aniônicos selecionados de éter fosfato de polioxietileno alquila (12 a 15), taurato de acil metila e glutamato de acila, em uma quantidade de 0,001 a 0,2 % em massa, (c) um óleo polar tendo iob de 0,05 a 0,80 e/ou óleo de silicone, e (d) água contendo um agente medicinal solúvel em água em uma quantidade de 0,5 a 5% em massa com base na composição, em que (a) tensoativo com base em silicone forma vesículas; (b) os tensoativos aniônicos se ligam a uma superfície das vesículas; e (c) o óleo polar e/ou óleo de silicone está presente dentro de uma membrana de bicamada das vesículas.
BR112012024910A 2010-03-31 2011-03-25 composição contendo vesícula e método para sua produção BR112012024910A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2010082301 2010-03-31
JP2010220684 2010-09-30
PCT/JP2011/057378 WO2011122477A1 (ja) 2010-03-31 2011-03-25 ベシクル含有組成物

Publications (1)

Publication Number Publication Date
BR112012024910A2 true BR112012024910A2 (pt) 2016-07-05

Family

ID=44712184

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012024910A BR112012024910A2 (pt) 2010-03-31 2011-03-25 composição contendo vesícula e método para sua produção

Country Status (10)

Country Link
US (1) US20130028950A1 (pt)
EP (1) EP2561862B1 (pt)
JP (1) JP4980474B2 (pt)
KR (1) KR101344557B1 (pt)
CN (1) CN102811708B (pt)
BR (1) BR112012024910A2 (pt)
ES (1) ES2546986T3 (pt)
RU (1) RU2517710C1 (pt)
TW (1) TWI412378B (pt)
WO (1) WO2011122477A1 (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5977107B2 (ja) * 2012-07-18 2016-08-24 花王株式会社 ベシクル組成物の製造方法
CN104093392A (zh) * 2012-02-13 2014-10-08 花王株式会社 囊泡组合物的制造方法
JP5988263B2 (ja) * 2012-09-18 2016-09-07 国立大学法人京都大学 複数の被内包リポソームを内包するリポソーム及びその製造方法
JP5690373B2 (ja) 2013-04-26 2015-03-25 株式会社 資生堂 水性組成物
CN103751072B (zh) * 2014-02-19 2015-04-22 珀莱雅化妆品股份有限公司 一种能恢复皮肤微生态的非离子表面活性剂囊泡及其制备方法
KR101655956B1 (ko) * 2014-10-30 2016-09-08 서울과학기술대학교 산학협력단 유성 화장품의 제거를 위한 w/o 마이크로에멀전 조성물
KR101664877B1 (ko) * 2015-06-26 2016-10-12 주식회사 코리아나화장품 니트로지방산을 함유하는 니오좀을 포함하는 화장료 조성물
CN111263628B (zh) * 2017-10-26 2023-09-08 株式会社资生堂 含囊泡的组合物
PT3700506T (pt) 2017-10-27 2021-09-29 Xyon Health Inc Formulações tópicas para tratar distúrbios dermatológicos incluindo calvíce de padrão masculino
WO2019235331A1 (ja) * 2018-06-06 2019-12-12 株式会社 資生堂 部分架橋もしくは架橋型ジメチルポリシロキサンを用いた水中油型乳化化粧料
CN116761579A (zh) * 2020-12-25 2023-09-15 株式会社资生堂 水包油型乳化化妆品
JP7695825B2 (ja) * 2021-06-10 2025-06-19 株式会社 資生堂 変臭定量化方法、変臭定量化装置、及び変臭定量化プログラム
KR102764695B1 (ko) 2021-08-05 2025-02-11 (주)아모레퍼시픽 난용성 성분이 안정화된 나노베지클을 포함하는 수중유형 화장료 조성물

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US5229104A (en) * 1991-04-29 1993-07-20 Richardson-Vicks Inc. Artificial tanning compositions containing positively charged paucilamellar vesicles
FR2725369B1 (fr) * 1994-10-07 1997-01-03 Oreal Composition cosmetique ou dermatologique constituee d'une emulsion huile dans eau a base de globules huileux pourvus d'un enrobage cristal liquide lamellaire
JP3483988B2 (ja) * 1995-06-01 2004-01-06 株式会社資生堂 皮膚外用剤
JP4246980B2 (ja) * 2001-09-11 2009-04-02 花王株式会社 皮膚外用剤
CN1720021A (zh) * 2002-12-04 2006-01-11 陶氏康宁公司 基于硅氧烷表面活性剂的极性有机油的泡囊和微乳液组合物
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JP4611831B2 (ja) * 2005-07-26 2011-01-12 株式会社資生堂 油中水型皮膚外用剤
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JP5121179B2 (ja) 2006-07-25 2013-01-16 株式会社 資生堂 ベシクル含有組成物及びその製造方法
JP5254645B2 (ja) * 2007-03-13 2013-08-07 株式会社コーセー ベシクル組成物及び該ベシクル組成物を配合した皮膚外用剤
BRPI0811575B1 (pt) 2007-05-15 2016-09-13 Shiseido Co Ltd composição contendo vesículas e método de produção da mesma
JP2009242326A (ja) * 2008-03-31 2009-10-22 Shiseido Co Ltd 美白液状化粧料
JP4395537B2 (ja) * 2008-04-09 2010-01-13 株式会社資生堂 ベシクル及びそれを含む化粧料

Also Published As

Publication number Publication date
JP4980474B2 (ja) 2012-07-18
JP2012092084A (ja) 2012-05-17
EP2561862A1 (en) 2013-02-27
KR101344557B1 (ko) 2013-12-26
TWI412378B (zh) 2013-10-21
HK1175996A1 (en) 2013-07-19
TW201201849A (en) 2012-01-16
EP2561862B1 (en) 2015-08-05
RU2517710C1 (ru) 2014-05-27
CN102811708B (zh) 2014-11-05
CN102811708A (zh) 2012-12-05
US20130028950A1 (en) 2013-01-31
EP2561862A4 (en) 2013-10-30
WO2011122477A1 (ja) 2011-10-06
KR20130040829A (ko) 2013-04-24
ES2546986T3 (es) 2015-09-30

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Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2622 DE 06-04-2021 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.