BR9610527A - Novos derivados de substâncias de ciclodepsipeptìdeo pf1022 - Google Patents
Novos derivados de substâncias de ciclodepsipeptìdeo pf1022Info
- Publication number
- BR9610527A BR9610527A BR9610527-5A BR9610527A BR9610527A BR 9610527 A BR9610527 A BR 9610527A BR 9610527 A BR9610527 A BR 9610527A BR 9610527 A BR9610527 A BR 9610527A
- Authority
- BR
- Brazil
- Prior art keywords
- new derivatives
- substances
- cyclodepsipeptide
- derivatives
- new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
Patente de Invenção para "NOVOS DERIVADOS DE SUBSTâNCIAS CICLODEPSIPEPTìDEO PF1022". Novos derivados de substância PF1022, que são cilcodepsipeptideos representados pela fórmula geral (I) mostrada abaixo, ou seus sais, são úteis como agente anti-helmintico para prevenção ou tratamento de infecções parasiticas.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP24405195 | 1995-09-22 | ||
| PCT/JP1996/002730 WO1997011064A1 (en) | 1995-09-22 | 1996-09-20 | Novel cyclic depsipeptide pf1022 derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9610527A true BR9610527A (pt) | 1999-12-21 |
Family
ID=17113003
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9610527-5A BR9610527A (pt) | 1995-09-22 | 1996-09-20 | Novos derivados de substâncias de ciclodepsipeptìdeo pf1022 |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US6329338B1 (pt) |
| EP (1) | EP0903347B1 (pt) |
| KR (1) | KR19990063676A (pt) |
| CN (1) | CN1082051C (pt) |
| AT (1) | ATE299871T1 (pt) |
| AU (1) | AU727532B2 (pt) |
| BR (1) | BR9610527A (pt) |
| CA (1) | CA2232668C (pt) |
| CZ (1) | CZ295705B6 (pt) |
| DE (1) | DE69634961T2 (pt) |
| DK (1) | DK0903347T3 (pt) |
| ES (1) | ES2246496T3 (pt) |
| HU (1) | HU228004B1 (pt) |
| IL (1) | IL123776A (pt) |
| NO (1) | NO310622B1 (pt) |
| NZ (1) | NZ318515A (pt) |
| PL (1) | PL186168B1 (pt) |
| WO (1) | WO1997011064A1 (pt) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998005655A1 (en) * | 1996-08-07 | 1998-02-12 | Meiji Seika Kaisha, Ltd. | Process for producing cyclodepsipeptide compounds and novel cyclodepsipeptide |
| AU6229898A (en) * | 1997-02-19 | 1998-09-09 | Bayer Aktiengesellschaft | Derivatives of cyclodepsipeptide, pf1022 substance |
| DE19811559A1 (de) * | 1998-03-17 | 1999-09-23 | Bayer Ag | Cyclooctadepsipeptide |
| US7109018B1 (en) | 1999-09-29 | 2006-09-19 | Meiji Seika Kaisha, Ltd. | Transformant producing secondary metabolite modified with functional group and novel biosynthesis genes |
| DE10031044A1 (de) * | 2000-06-26 | 2002-01-03 | Bayer Ag | Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere |
| DE10104362A1 (de) * | 2001-02-01 | 2002-08-08 | Bayer Ag | Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit |
| DE102004055316A1 (de) * | 2004-11-16 | 2006-05-18 | Bayer Healthcare Ag | Verhinderung vertikaler Endoparasiten-Infektionen |
| DE102008022520A1 (de) | 2008-05-07 | 2009-11-12 | Bayer Animal Health Gmbh | Feste Arzneimittelformulierung mit verzögerter Freisetzung |
| DE102008030764A1 (de) | 2008-06-28 | 2009-12-31 | Bayer Animal Health Gmbh | Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden |
| DE102008031284A1 (de) * | 2008-07-02 | 2010-01-07 | Bayer Schering Pharma Aktiengesellschaft | Neue Bekämpfungsmöglichkeit der Giardiose |
| DE102008031283A1 (de) | 2008-07-02 | 2010-01-07 | Bayer Schering Pharma Aktiengesellschaft | Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten |
| DE102009012423A1 (de) | 2009-03-10 | 2010-09-16 | Bayer Animal Health Gmbh | Zubereitung auf Ölbasis |
| DE102010064245A1 (de) | 2010-12-28 | 2012-06-28 | Bayer Animal Health Gmbh | Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen |
| WO2012028556A1 (en) | 2010-08-31 | 2012-03-08 | Bayer Animal Health Gmbh | Macrocyclic lactones and their use and their combinations with other active substances |
| CN107835818B (zh) | 2015-05-20 | 2022-04-29 | 勃林格殷格翰动物保健美国公司 | 驱虫缩酚酸肽化合物 |
| KR20220003663A (ko) | 2015-12-28 | 2022-01-10 | 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 | 구충성 뎁시펩티드 화합물 |
| EP3541789A1 (en) | 2016-11-16 | 2019-09-25 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic depsipeptide compounds |
| CN111757880A (zh) | 2017-11-07 | 2020-10-09 | 拜耳动物保健有限责任公司 | 用于合成环状缩肽的方法 |
| JP7164608B2 (ja) | 2017-11-29 | 2022-11-01 | ゾエティス・サービシーズ・エルエルシー | 内部寄生性デプシペプチド |
| EP3790876B1 (en) | 2018-05-10 | 2025-04-30 | Zoetis Services LLC | Endoparasitic depsipeptides |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH477172A (de) * | 1965-05-18 | 1969-08-31 | Agripat Sa | Beifuttermittel |
| DK431083A (da) * | 1982-09-22 | 1984-03-23 | Meiji Seika Co | Fremgangsmaade til fremstilling af hydroxylaminderivater |
| NO176766C (no) * | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
| CA2132199C (en) * | 1992-03-17 | 2000-01-18 | Hitoshi Nishiyama | Depsipeptide derivative, production thereof and use thereof |
| JP2873894B2 (ja) * | 1992-10-19 | 1999-03-24 | 明治製菓株式会社 | 環状デプシペプチドおよびその製造法 |
| CN1073560C (zh) * | 1993-02-19 | 2001-10-24 | 明治制果株式会社 | 环缩酚酸肽pf1022衍生物 |
| DE4317432A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
| DE4317457A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
| JPH07233068A (ja) * | 1993-12-27 | 1995-09-05 | Meiji Seika Kaisha Ltd | 高コレステロール血症、高脂血症又は動脈硬化症の治療薬 |
-
1996
- 1996-09-20 NZ NZ318515A patent/NZ318515A/xx not_active IP Right Cessation
- 1996-09-20 ES ES96931283T patent/ES2246496T3/es not_active Expired - Lifetime
- 1996-09-20 AU AU70019/96A patent/AU727532B2/en not_active Expired
- 1996-09-20 DK DK96931283T patent/DK0903347T3/da active
- 1996-09-20 EP EP96931283A patent/EP0903347B1/en not_active Expired - Lifetime
- 1996-09-20 PL PL96326024A patent/PL186168B1/pl unknown
- 1996-09-20 BR BR9610527-5A patent/BR9610527A/pt not_active Application Discontinuation
- 1996-09-20 US US09/043,558 patent/US6329338B1/en not_active Expired - Lifetime
- 1996-09-20 KR KR1019980702138A patent/KR19990063676A/ko not_active Ceased
- 1996-09-20 IL IL12377696A patent/IL123776A/en not_active IP Right Cessation
- 1996-09-20 WO PCT/JP1996/002730 patent/WO1997011064A1/ja not_active Ceased
- 1996-09-20 CZ CZ1998855A patent/CZ295705B6/cs not_active IP Right Cessation
- 1996-09-20 HU HU0001164A patent/HU228004B1/hu unknown
- 1996-09-20 DE DE69634961T patent/DE69634961T2/de not_active Expired - Lifetime
- 1996-09-20 AT AT96931283T patent/ATE299871T1/de active
- 1996-09-20 CN CN96198101A patent/CN1082051C/zh not_active Expired - Lifetime
- 1996-09-20 CA CA2232668A patent/CA2232668C/en not_active Expired - Lifetime
-
1998
- 1998-03-19 NO NO19981250A patent/NO310622B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| PL326024A1 (en) | 1998-08-17 |
| EP0903347B1 (en) | 2005-07-20 |
| HUP0001164A3 (en) | 2001-04-28 |
| AU727532B2 (en) | 2000-12-14 |
| CA2232668C (en) | 2011-10-18 |
| CA2232668A1 (en) | 1997-03-27 |
| PL186168B1 (pl) | 2003-11-28 |
| EP0903347A4 (pt) | 1999-03-24 |
| MX9802268A (es) | 1998-08-30 |
| NZ318515A (en) | 2000-05-26 |
| JP4001381B1 (pt) | 2007-10-31 |
| DE69634961T2 (de) | 2006-04-20 |
| AU7001996A (en) | 1997-04-09 |
| NO310622B1 (no) | 2001-07-30 |
| IL123776A0 (en) | 1998-10-30 |
| EP0903347A1 (en) | 1999-03-24 |
| KR19990063676A (ko) | 1999-07-26 |
| CZ85598A3 (cs) | 1998-08-12 |
| DK0903347T3 (da) | 2005-11-21 |
| CN1201456A (zh) | 1998-12-09 |
| CN1082051C (zh) | 2002-04-03 |
| DE69634961D1 (de) | 2005-08-25 |
| HU228004B1 (en) | 2012-08-28 |
| CZ295705B6 (cs) | 2005-10-12 |
| IL123776A (en) | 2002-09-12 |
| NO981250L (no) | 1998-05-22 |
| US6329338B1 (en) | 2001-12-11 |
| NO981250D0 (no) | 1998-03-19 |
| WO1997011064A1 (en) | 1997-03-27 |
| ES2246496T3 (es) | 2006-02-16 |
| HUP0001164A2 (hu) | 2000-11-28 |
| ATE299871T1 (de) | 2005-08-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B25A | Requested transfer of rights approved |
Owner name: BAYER AKTIENGSELLSCHAFT (DE) Free format text: TRANSFERIDO DE: MEIJI SHEIKA KAISHA, LTD. |
|
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PRESENTE PEDIDO COM BASE NO DISPOSTO NOS ARTIGOS 8O E 13O DA LPI 9.279/96 |
|
| B12B | Appeal against refusal [chapter 12.2 patent gazette] |