BR9810595A - Medicamentos, compostos de poliidroxibutilpirazina, processo para preparação dos compostos, e, utilização dos compostos. - Google Patents

Medicamentos, compostos de poliidroxibutilpirazina, processo para preparação dos compostos, e, utilização dos compostos.

Info

Publication number
BR9810595A
BR9810595A BR9810595-7A BR9810595A BR9810595A BR 9810595 A BR9810595 A BR 9810595A BR 9810595 A BR9810595 A BR 9810595A BR 9810595 A BR9810595 A BR 9810595A
Authority
BR
Brazil
Prior art keywords
radical
compounds
represent
methylene
choh
Prior art date
Application number
BR9810595-7A
Other languages
English (en)
Portuguese (pt)
Inventor
Georges Bashiardes
Jean-Christophe Carry
Michel Evers
Bruno Filoche
Serge Mignani
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of BR9810595A publication Critical patent/BR9810595A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/12Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cosmetics (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR9810595-7A 1997-07-17 1998-07-15 Medicamentos, compostos de poliidroxibutilpirazina, processo para preparação dos compostos, e, utilização dos compostos. BR9810595A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9709059A FR2766183B1 (fr) 1997-07-17 1997-07-17 Medicaments contenant des polyhydroxybutylpyrazines, les polyhydroxybutylpyrazines nouvelles et leur preparation
PCT/FR1998/001543 WO1999003841A1 (fr) 1997-07-17 1998-07-15 Polyhydroxybutylpyrazines, leur preparation et medicaments les contenant

Publications (1)

Publication Number Publication Date
BR9810595A true BR9810595A (pt) 2000-09-12

Family

ID=9509301

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9810595-7A BR9810595A (pt) 1997-07-17 1998-07-15 Medicamentos, compostos de poliidroxibutilpirazina, processo para preparação dos compostos, e, utilização dos compostos.

Country Status (25)

Country Link
US (1) US6288066B1 (cs)
EP (1) EP1001942B1 (cs)
JP (1) JP4443033B2 (cs)
KR (1) KR20010021871A (cs)
CN (1) CN1264368A (cs)
AT (1) ATE243683T1 (cs)
AU (1) AU745905B2 (cs)
BR (1) BR9810595A (cs)
CA (1) CA2296725C (cs)
CZ (1) CZ290896B6 (cs)
DE (1) DE69815854T2 (cs)
DK (1) DK1001942T3 (cs)
ES (1) ES2196595T3 (cs)
FR (1) FR2766183B1 (cs)
HU (1) HUP0004661A3 (cs)
IL (1) IL134039A0 (cs)
MX (1) MXPA00000437A (cs)
NO (1) NO20000199L (cs)
NZ (1) NZ502279A (cs)
PL (1) PL338147A1 (cs)
PT (1) PT1001942E (cs)
RU (1) RU2186773C2 (cs)
SK (1) SK462000A3 (cs)
WO (1) WO1999003841A1 (cs)
ZA (1) ZA986336B (cs)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2802816A1 (fr) * 1999-12-23 2001-06-29 Aventis Pharma Sa Association de deoxyfructosazine et d'un antidiabetique inhibiteur d'alpha-glucosidase
FR2802813A1 (fr) * 1999-12-23 2001-06-29 Aventis Pharma Sa Association de deoxyfructosazine et d'un antidiabetique de la famille des biguandes
FR2802815A1 (fr) * 1999-12-23 2001-06-29 Aventis Pharma Sa Association de deoxyfructosazine et d'un antidiabetique agoniste du recepteur gamma-active par le proliferateur de peroxisome
US6794506B2 (en) * 2000-07-21 2004-09-21 Elan Pharmaceuticals, Inc. 3-(heteroaryl) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4
MY141521A (en) * 2002-12-12 2010-05-14 Hoffmann La Roche 5-substituted-six-membered heteroaromatic glucokinase activators
DE102005047647A1 (de) * 2005-10-05 2007-04-12 Merck Patent Gmbh a,a'-Dihydroxyketonderivate und deren Verwendung als UV-Filter
US8278459B2 (en) 2007-03-19 2012-10-02 Dsm Ip Assets B.V. UV-filter compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3600052A1 (de) * 1986-01-03 1987-07-09 Merck Patent Gmbh Heterocyclische verbindungen
FR2744365B1 (fr) * 1996-02-06 1998-02-27 Inst Malgache Rech Appl Melanges isolables a partir de graines d'eugenia jambolana lamarck, leur preparation et l'utilisation de ces melanges et certains de leurs constituants comme medicaments

Also Published As

Publication number Publication date
CA2296725C (fr) 2008-11-18
JP2001510185A (ja) 2001-07-31
DE69815854T2 (de) 2004-05-13
PT1001942E (pt) 2003-11-28
HUP0004661A3 (en) 2001-12-28
EP1001942B1 (fr) 2003-06-25
NZ502279A (en) 2002-04-26
IL134039A0 (en) 2001-04-30
PL338147A1 (en) 2000-09-25
NO20000199D0 (no) 2000-01-14
ZA986336B (en) 1999-01-27
MXPA00000437A (es) 2002-04-17
CN1264368A (zh) 2000-08-23
DK1001942T3 (da) 2003-10-20
DE69815854D1 (de) 2003-07-31
RU2186773C2 (ru) 2002-08-10
SK462000A3 (en) 2000-06-12
JP4443033B2 (ja) 2010-03-31
ATE243683T1 (de) 2003-07-15
FR2766183A1 (fr) 1999-01-22
NO20000199L (no) 2000-01-14
AU8810398A (en) 1999-02-10
CZ2000121A3 (cs) 2000-05-17
HUP0004661A2 (hu) 2001-11-28
KR20010021871A (ko) 2001-03-15
CZ290896B6 (cs) 2002-11-13
EP1001942A1 (fr) 2000-05-24
CA2296725A1 (fr) 1999-01-28
US6288066B1 (en) 2001-09-11
WO1999003841A1 (fr) 1999-01-28
ES2196595T3 (es) 2003-12-16
FR2766183B1 (fr) 1999-08-27
AU745905B2 (en) 2002-04-11

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Legal Events

Date Code Title Description
TC Change of name
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A,8A E 9A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1909 DE 07/08/2007.