BR9912980A - Composição farmacêutica administrável oralmente, utilização de compostos, tablete de mascar e processos para evitar a sìndrome de vazamento anal de óleo - Google Patents

Composição farmacêutica administrável oralmente, utilização de compostos, tablete de mascar e processos para evitar a sìndrome de vazamento anal de óleo

Info

Publication number
BR9912980A
BR9912980A BR9912980-9A BR9912980A BR9912980A BR 9912980 A BR9912980 A BR 9912980A BR 9912980 A BR9912980 A BR 9912980A BR 9912980 A BR9912980 A BR 9912980A
Authority
BR
Brazil
Prior art keywords
pharmaceutical composition
compounds
processes
orally administrable
oil leakage
Prior art date
Application number
BR9912980-9A
Other languages
English (en)
Other versions
BR9912980B1 (pt
Inventor
Manuela Hug
Hans-Peter Maerki
Marcel Meier
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR9912980A publication Critical patent/BR9912980A/pt
Publication of BR9912980B1 publication Critical patent/BR9912980B1/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Nutrition Science (AREA)
  • Zoology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Physiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Jellies, Jams, And Syrups (AREA)
  • General Preparation And Processing Of Foods (AREA)

Abstract

<B><MU>COMPOSIçãO FARMACêUTICA ADMINISTRáVEL ORALMENTE, UTILIZAçãO DE COMPOSTOS, TABLETE DE MASCAR E PROCESSOS PARA EVITAR A SìNDROME DE VAZAMENTO ANAL DE óLEO<MV><D> Expõe-se uma composição farmacêutica administrável oralmente que contém um inibidor de lípase gastrintestinal, um (ou mais) aditivo(s) do grupo que consiste de espessadores e emulsionadores fracamente digeríveis, fracamente fermentáveis, hidrófilos e/ou hidrocolóides, e excipientes auxiliares.
BRPI9912980-9B1A 1998-08-14 1999-08-02 Composição farmacêutica administrável oralmente, tablete de mascar contendo a mesma e utilização da mesma BR9912980B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP98115311 1998-08-14
EP99109516 1999-05-12
PCT/EP1999/005607 WO2000009122A1 (en) 1998-08-14 1999-08-02 Pharmaceutical compositions containing lipase inhibitors

Publications (2)

Publication Number Publication Date
BR9912980A true BR9912980A (pt) 2001-05-08
BR9912980B1 BR9912980B1 (pt) 2013-10-22

Family

ID=26149537

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9912980-9B1A BR9912980B1 (pt) 1998-08-14 1999-08-02 Composição farmacêutica administrável oralmente, tablete de mascar contendo a mesma e utilização da mesma

Country Status (19)

Country Link
US (1) US6358522B1 (pt)
EP (1) EP1105122B1 (pt)
JP (1) JP3774118B2 (pt)
KR (1) KR20010079635A (pt)
CN (1) CN1170534C (pt)
AR (1) AR035001A1 (pt)
AT (1) ATE293970T1 (pt)
AU (1) AU761351B2 (pt)
BR (1) BR9912980B1 (pt)
CA (1) CA2340056C (pt)
CO (1) CO5130009A1 (pt)
DE (1) DE69924999T2 (pt)
DK (1) DK1105122T3 (pt)
ES (1) ES2242413T3 (pt)
MA (1) MA26671A1 (pt)
PE (1) PE20000953A1 (pt)
PT (1) PT1105122E (pt)
TR (1) TR200100471T2 (pt)
WO (1) WO2000009122A1 (pt)

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AR025609A1 (es) 1999-09-13 2002-12-04 Hoffmann La Roche Formulaciones lipidas solidas
AR025587A1 (es) 1999-09-13 2002-12-04 Hoffmann La Roche Formulaciones en dispersion que contienen inhibidores de lipasa
EP1132389A1 (en) 2000-03-06 2001-09-12 Vernalis Research Limited New aza-indolyl derivatives for the treatment of obesity
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RU2241462C2 (ru) * 2000-07-28 2004-12-10 Ф. Хоффманн-Ля Рош Аг Новая фармацевтическая композиция
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AU2167002A (en) 2000-10-16 2002-06-11 Hoffmann La Roche Indoline derivatives and their use as 5-ht2 receptor ligands
GB0030710D0 (en) 2000-12-15 2001-01-31 Hoffmann La Roche Piperazine derivatives
KR100539143B1 (ko) 2000-12-27 2005-12-26 에프. 호프만-라 로슈 아게 인돌 유도체 및 그의 5-ｈｔ2ｂ 및 5-ｈｔ2ｃ 수용체리간드로서의 용도
GB0106177D0 (en) 2001-03-13 2001-05-02 Hoffmann La Roche Piperazine derivatives
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US6730319B2 (en) * 2001-06-06 2004-05-04 Hoffmann-La Roche Inc. Pharmaceutical compositions having depressed melting points
US7049345B2 (en) * 2001-06-29 2006-05-23 Genzyme Corporation Fat-binding polymers
US7041280B2 (en) * 2001-06-29 2006-05-09 Genzyme Corporation Aryl boronate functionalized polymers for treating obesity
US6787558B2 (en) 2001-09-28 2004-09-07 Hoffmann-La Roche Inc. Quinoline derivatives
GB0202015D0 (en) 2002-01-29 2002-03-13 Hoffmann La Roche Piperazine Derivatives
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MXPA04008379A (es) 2002-02-28 2004-11-26 Hoffmann La Roche Derivados de tiazol como antagonistas del receptor de neuropeptido y (npy).
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EP1560816A1 (en) 2002-07-05 2005-08-10 F. Hoffmann-La Roche Ag Quinazoline derivatives
RU2324685C2 (ru) 2002-08-07 2008-05-20 Ф.Хоффманн-Ля Рош Аг Производные тиазола, способ их получения и применение, фармацевтическая композиция, обладающая свойствами антагонистов рецепторов npy
RU2296759C2 (ru) 2002-09-12 2007-04-10 Ф.Хоффманн-Ля Рош Аг N-замещенные 1н-индол-5-пропионовые кислоты, фармацевтическая композиция, содержащая эти соединения, и их применение (варианты)
RU2315767C2 (ru) 2002-11-25 2008-01-27 Ф.Хоффманн-Ля Рош Аг Индолилпроизводные, способ их получения, фармацевтическая композиция, способ лечения и/или профилактики заболеваний
US8372430B2 (en) 2002-12-17 2013-02-12 The Procter & Gamble Company Compositions, methods, and kits useful for the alleviation of gastrointestinal effects
GB0314967D0 (en) 2003-06-26 2003-07-30 Hoffmann La Roche Piperazine derivatives
RU2321586C2 (ru) 2003-08-12 2008-04-10 Ф.Хоффманн-Ля Рош Аг Производные тиазола в качестве антагонистов npy
RU2006107444A (ru) 2003-08-12 2007-09-20 Ф.Хоффманн-Ля Рош Аг (Ch) 2-амино-5-бензоилтиазолы в качестве антагонистов npy
CN101171252B (zh) 2005-05-03 2011-06-01 霍夫曼-拉罗奇有限公司 作为5-ht2配体的四环氮杂吡嗪并二氢吲哚类化合物
ES2434072T3 (es) * 2005-06-09 2013-12-13 Norgine Bv Preparación sólida de 2-hexadeciloxi-6-metil-4H-3,1-benzoxacin-4-ona
AU2006281435A1 (en) 2005-08-18 2007-02-22 F. Hoffmann-La Roche Ag Thiazolyl piperidine derivatives useful as H3 receptor modulators
ES2359739T3 (es) 2005-11-30 2011-05-26 F. Hoffmann-La Roche Ag Derivados de indol-2-il-amida 1,5-sustituida.
CN101316835A (zh) 2005-11-30 2008-12-03 霍夫曼-拉罗奇有限公司 5-取代的吲哚-2-甲酰胺衍生物
CN101316838B (zh) 2005-11-30 2013-01-30 霍夫曼-拉罗奇有限公司 用作h3调节剂的1,1-二氧代-硫代吗啉基吲哚基甲酮衍生物
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EP2032554A1 (en) 2006-05-30 2009-03-11 F. Hoffmann-Roche AG Piperidinyl pyrimidine derivatives
US7514433B2 (en) 2006-08-03 2009-04-07 Hoffmann-La Roche Inc. 1H-indole-6-yl-piperazin-1-yl-methanone derivatives
US20080146559A1 (en) 2006-12-08 2008-06-19 Li Chen 4,5,6,7-Tetrahydro-Thieno [2,3-C] Pyridine Derivatives
BRPI0810278B1 (pt) * 2007-05-16 2017-10-24 Buckman Laboratories International, Inc. Method for one of the size reductions of contaminants, number or quantity of measurable particles and / or the treatment of organic fiber contaminants in paper manufacturing systems
BRPI0814532A2 (pt) 2007-07-25 2015-01-27 Hoffmann La Roche Compostos, processo para a sua manufatura, composições farmacêuticas que os compreendem, método para o tratamento e/ou prevenção de enfermidades que estão associadas com a modulação dos receptores de h3, e uso desses compostos para a preparação de medicamentos.
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Also Published As

Publication number Publication date
JP2002522491A (ja) 2002-07-23
EP1105122B1 (en) 2005-04-27
CN1170534C (zh) 2004-10-13
DK1105122T3 (da) 2005-08-08
AU761351B2 (en) 2003-06-05
AR035001A1 (es) 2004-04-14
CA2340056A1 (en) 2000-02-24
ES2242413T3 (es) 2005-11-01
PE20000953A1 (es) 2000-09-26
JP3774118B2 (ja) 2006-05-10
PT1105122E (pt) 2005-08-31
DE69924999T2 (de) 2006-05-04
AU5418599A (en) 2000-03-06
CN1312713A (zh) 2001-09-12
CA2340056C (en) 2007-01-09
EP1105122A1 (en) 2001-06-13
ATE293970T1 (de) 2005-05-15
CO5130009A1 (es) 2002-02-27
TR200100471T2 (tr) 2001-07-23
KR20010079635A (ko) 2001-08-22
WO2000009122A1 (en) 2000-02-24
MA26671A1 (fr) 2004-12-20
US6358522B1 (en) 2002-03-19
DE69924999D1 (de) 2005-06-02
BR9912980B1 (pt) 2013-10-22

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DE INT.CL: A61K 31/365, A61K 9/00, A61K 45/08, A61K 47/38, A61P 3/04, A61P 30/04, A61P 43/00

Ipc: A61K 31/365 (2008.04), A61K 9/00 (2008.04), A61K 4

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFERIMENTO DO PRESENTE PEDIDO UMA VEZ QUE ESTE CONTRARIA O DISPOSTO NOS ARTIGOS 8O, 10 ( VIII ), 11, 13 E 25 DA LPI

B12B Appeal against refusal [chapter 12.2 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 22/10/2013, OBSERVADAS AS CONDICOES LEGAIS.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

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B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2594 DE 24-09-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.