BRPI0407303A - Composição farmacêutica - Google Patents
Composição farmacêuticaInfo
- Publication number
- BRPI0407303A BRPI0407303A BR0407303-7A BRPI0407303A BRPI0407303A BR PI0407303 A BRPI0407303 A BR PI0407303A BR PI0407303 A BRPI0407303 A BR PI0407303A BR PI0407303 A BRPI0407303 A BR PI0407303A
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutical composition
- hyperinsulinemia
- preventative
- remedy
- analogues
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 208000002249 Diabetes Complications Diseases 0.000 abstract 1
- 206010012655 Diabetic complications Diseases 0.000 abstract 1
- 206010060378 Hyperinsulinaemia Diseases 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 239000003472 antidiabetic agent Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 230000003451 hyperinsulinaemic effect Effects 0.000 abstract 1
- 201000008980 hyperinsulinism Diseases 0.000 abstract 1
- 229940126904 hypoglycaemic agent Drugs 0.000 abstract 1
- 230000002503 metabolic effect Effects 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
- A61K31/5517—1,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/28—Insulins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Zoology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
"COMPOSIçãO FARMACêUTICA". Um preventivo e/ou remédio para a diabete, complicações diabéticas, hiperinsulinemia, erro metabólico do açúcar ou obesidade caracterizados por compreender uma combinação de um composto representado pela seguinte fórmula, seus análogos ou um sal destes farmaceuticamente aceitáveis com um agente hipoglicêmico.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2003031088 | 2003-02-07 | ||
| PCT/JP2004/001279 WO2004069259A1 (ja) | 2003-02-07 | 2004-02-06 | 糖尿病治療剤 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0407303A true BRPI0407303A (pt) | 2006-02-07 |
Family
ID=32844288
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0407303-7A BRPI0407303A (pt) | 2003-02-07 | 2004-02-06 | Composição farmacêutica |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US7807663B2 (pt) |
| EP (1) | EP1595544A4 (pt) |
| JP (1) | JPWO2004069259A1 (pt) |
| KR (1) | KR20050097537A (pt) |
| CN (2) | CN101822834A (pt) |
| AU (1) | AU2004210268B8 (pt) |
| BR (1) | BRPI0407303A (pt) |
| CA (1) | CA2515294A1 (pt) |
| MX (1) | MXPA05008363A (pt) |
| RU (1) | RU2358738C2 (pt) |
| WO (1) | WO2004069259A1 (pt) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI241302B (en) * | 2000-12-01 | 2005-10-11 | Ajinomoto Kk | Lactam compounds and pharmaceutical use thereof |
| AU2004261353B2 (en) | 2003-08-05 | 2009-12-10 | Novo Nordisk A/S | Novel insulin derivatives |
| WO2005042536A1 (ja) * | 2003-10-31 | 2005-05-12 | Ajinomoto Co., Inc. | 複素環を有する新規縮合多環式化合物及びその医薬用途 |
| CA2553329A1 (en) * | 2004-01-14 | 2005-07-28 | Ajinomoto Co., Inc. | New fused polycyclic compounds |
| JP5056412B2 (ja) | 2005-04-28 | 2012-10-24 | 味の素株式会社 | 新規ラクタム化合物 |
| WO2006119038A1 (en) * | 2005-04-29 | 2006-11-09 | Naturegen, Inc. | Compositions and methods for controlling glucose uptake |
| WO2007019526A2 (en) * | 2005-08-05 | 2007-02-15 | Naturegen, Inc. | Compositions and methods for controlling glucose and lipid uptake from foods |
| EP1969004B1 (en) | 2005-12-28 | 2011-08-10 | Novo Nordisk A/S | Compositions comprising an acylated insulin and zinc and method of making the said compositions |
| EP2157092A4 (en) * | 2007-04-11 | 2011-04-13 | Ajinomoto Kk | Remedy for diabetes |
| WO2008139575A1 (ja) * | 2007-04-27 | 2008-11-20 | Ajinomoto Co., Inc. | 経口投与用製剤 |
| WO2008139574A1 (ja) * | 2007-04-27 | 2008-11-20 | Ajinomoto Co., Inc. | ラクタム化合物の結晶形およびその製造方法 |
| WO2008136394A1 (ja) * | 2007-04-27 | 2008-11-13 | Ajinomoto Co., Inc. | ラクタム化合物の製造方法及びその製造中間体 |
| JP5552046B2 (ja) | 2007-06-13 | 2014-07-16 | ノボ・ノルデイスク・エー/エス | インスリン誘導体を含有する薬学的製剤 |
| CN102202683A (zh) | 2008-10-30 | 2011-09-28 | 诺沃-诺迪斯克有限公司 | 用少于每日一次的注射频率注射胰岛素来治疗糖尿病 |
| DK2632478T3 (da) | 2010-10-27 | 2019-10-07 | Novo Nordisk As | Behandling af diabetes melitus under anvendelse af insulinindsprøjtninger indgivet med varierende indsprøjtningsintervaller |
| KR101904920B1 (ko) * | 2012-05-18 | 2018-10-08 | (주)아모레퍼시픽 | 보글리보스를 포함하는 피부 미백용 조성물 |
| EP2991672A1 (en) | 2013-04-30 | 2016-03-09 | Novo Nordisk A/S | Novel administration regime |
| US10335464B1 (en) | 2018-06-26 | 2019-07-02 | Novo Nordisk A/S | Device for titrating basal insulin |
| CN114096269B (zh) | 2019-07-12 | 2024-06-11 | 诺和诺德股份有限公司 | 高浓度胰岛素制剂 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2961377A (en) * | 1957-08-05 | 1960-11-22 | Us Vitamin Pharm Corp | Oral anti-diabetic compositions and methods |
| US3174901A (en) * | 1963-01-31 | 1965-03-23 | Jan Marcel Didier Aron Samuel | Process for the oral treatment of diabetes |
| NL132376C (pt) * | 1966-02-10 | |||
| US4062950A (en) * | 1973-09-22 | 1977-12-13 | Bayer Aktiengesellschaft | Amino sugar derivatives |
| FR2774591B1 (fr) * | 1998-02-12 | 2000-05-05 | Lipha | Composition pharmaceutique comprenant l'association metformine et fibrate et son utilisation pour la preparation de medicaments destines a reduire l'hyperglycemie |
| US20020099186A1 (en) * | 2000-11-29 | 2002-07-25 | Synsorb Biotech, Inc. | Processes for the preparation of alphaGal(1-3)betaGal(1-4)Glc-OR |
| TWI241302B (en) * | 2000-12-01 | 2005-10-11 | Ajinomoto Kk | Lactam compounds and pharmaceutical use thereof |
| WO2005042536A1 (ja) | 2003-10-31 | 2005-05-12 | Ajinomoto Co., Inc. | 複素環を有する新規縮合多環式化合物及びその医薬用途 |
-
2004
- 2004-02-06 MX MXPA05008363A patent/MXPA05008363A/es active IP Right Grant
- 2004-02-06 BR BR0407303-7A patent/BRPI0407303A/pt not_active IP Right Cessation
- 2004-02-06 RU RU2005127870/15A patent/RU2358738C2/ru not_active IP Right Cessation
- 2004-02-06 EP EP04708897A patent/EP1595544A4/en not_active Withdrawn
- 2004-02-06 CA CA002515294A patent/CA2515294A1/en not_active Abandoned
- 2004-02-06 CN CN201010167277A patent/CN101822834A/zh active Pending
- 2004-02-06 KR KR1020057014352A patent/KR20050097537A/ko not_active Ceased
- 2004-02-06 JP JP2005504900A patent/JPWO2004069259A1/ja active Pending
- 2004-02-06 AU AU2004210268A patent/AU2004210268B8/en not_active Ceased
- 2004-02-06 CN CN2004800094107A patent/CN1771040B/zh not_active Expired - Fee Related
- 2004-02-06 WO PCT/JP2004/001279 patent/WO2004069259A1/ja not_active Ceased
-
2005
- 2005-08-08 US US11/198,511 patent/US7807663B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US7807663B2 (en) | 2010-10-05 |
| EP1595544A4 (en) | 2009-05-06 |
| RU2358738C2 (ru) | 2009-06-20 |
| CN1771040B (zh) | 2010-06-16 |
| CA2515294A1 (en) | 2004-08-19 |
| MXPA05008363A (es) | 2005-12-06 |
| CN101822834A (zh) | 2010-09-08 |
| AU2004210268A1 (en) | 2004-08-19 |
| AU2004210268B8 (en) | 2009-06-04 |
| US20050272641A1 (en) | 2005-12-08 |
| EP1595544A1 (en) | 2005-11-16 |
| KR20050097537A (ko) | 2005-10-07 |
| JPWO2004069259A1 (ja) | 2006-05-25 |
| WO2004069259A1 (ja) | 2004-08-19 |
| RU2005127870A (ru) | 2006-03-10 |
| CN1771040A (zh) | 2006-05-10 |
| AU2004210268B2 (en) | 2009-05-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 8A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2144 DE 07/02/2012. |