BRPI0407480A - Cristal de intermediário sintético de carbapenem - Google Patents

Cristal de intermediário sintético de carbapenem

Info

Publication number
BRPI0407480A
BRPI0407480A BR0407480-7A BRPI0407480A BRPI0407480A BR PI0407480 A BRPI0407480 A BR PI0407480A BR PI0407480 A BRPI0407480 A BR PI0407480A BR PI0407480 A BRPI0407480 A BR PI0407480A
Authority
BR
Brazil
Prior art keywords
carbapenem
synthetic intermediate
crystal
intermediate crystal
synthetic
Prior art date
Application number
BR0407480-7A
Other languages
English (en)
Inventor
Masaaki Uenaka
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of BRPI0407480A publication Critical patent/BRPI0407480A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C07D477/10—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D477/12—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
    • C07D477/16—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
    • C07D477/20—Sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"CRISTAL DE INTERMEDIáRIO SINTéTICO DE CARBAPENEM". A presente invenção refere-se a um cristal de intermediários sintéticos de carbapenem, que é útil para um método industrial para produção, que é fornecido. Um solvato do composto (I) da fórmula: ou um cristal deste.
BR0407480-7A 2003-02-14 2004-02-12 Cristal de intermediário sintético de carbapenem BRPI0407480A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2003036233 2003-02-14
PCT/JP2004/001477 WO2004072073A1 (ja) 2003-02-14 2004-02-12 カルバペネム合成中間体の結晶

Publications (1)

Publication Number Publication Date
BRPI0407480A true BRPI0407480A (pt) 2006-02-07

Family

ID=32866319

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0407480-7A BRPI0407480A (pt) 2003-02-14 2004-02-12 Cristal de intermediário sintético de carbapenem

Country Status (11)

Country Link
US (1) US7767809B2 (pt)
EP (1) EP1595883A4 (pt)
JP (1) JP4404316B2 (pt)
KR (1) KR101089529B1 (pt)
CN (1) CN100378099C (pt)
AU (1) AU2004212402B2 (pt)
BR (1) BRPI0407480A (pt)
CA (1) CA2515741C (pt)
MX (1) MXPA05008439A (pt)
TW (1) TWI319401B (pt)
WO (1) WO2004072073A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030153191A1 (en) * 2000-03-31 2003-08-14 Izumi Saitoh Novel crystal form of pyrrolidylthiocarbapenem derivative
EP1852436A4 (en) * 2005-02-15 2010-02-24 Shionogi & Co PROCESS FOR PRODUCING CARBAPENEME DERIVATIVE AND CRYSTALLINE INTERMEDIATE THEREOF
US7932381B2 (en) * 2005-02-15 2011-04-26 Shionogi & Co., Ltd. Process for producing carbapenem derivative and intermediate crystal therefor
JP2008007418A (ja) * 2006-06-27 2008-01-17 Tokuyama Corp 安定な結晶構造を有するベンゾオキサジン化合物の製造方法
CN101747333B (zh) * 2008-11-28 2012-07-04 上海医药工业研究院 一种多尼培南的中间体化合物的制备方法
CN101747251B (zh) * 2008-11-28 2013-01-16 上海医药工业研究院 一种多尼培南的中间体的结晶及其制备方法
WO2015167148A1 (ko) 2014-04-28 2015-11-05 제이더블유중외제약 주식회사 도리페넴의 신규한 결정 및 이의 제조방법

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5317016A (en) 1991-08-20 1994-05-31 Shionogi Seiyaku Kabushiki Kaisha Pyrrolidylthiocarbapenem derivative
US5539102A (en) 1992-02-21 1996-07-23 Shionogi Seiyaku Kabushiki Kaisha Production method for sulfamide
US7932381B2 (en) * 2005-02-15 2011-04-26 Shionogi & Co., Ltd. Process for producing carbapenem derivative and intermediate crystal therefor

Also Published As

Publication number Publication date
EP1595883A1 (en) 2005-11-16
KR101089529B1 (ko) 2011-12-05
US20060229285A1 (en) 2006-10-12
AU2004212402A1 (en) 2004-08-26
AU2004212402B2 (en) 2009-11-26
CA2515741C (en) 2014-04-01
TWI319401B (en) 2010-01-11
JP4404316B2 (ja) 2010-01-27
JPWO2004072073A1 (ja) 2006-06-01
TW200504066A (en) 2005-02-01
CN100378099C (zh) 2008-04-02
EP1595883A4 (en) 2008-11-26
US7767809B2 (en) 2010-08-03
KR20050099548A (ko) 2005-10-13
CN1747954A (zh) 2006-03-15
MXPA05008439A (es) 2005-10-19
WO2004072073A1 (ja) 2004-08-26
CA2515741A1 (en) 2004-08-26

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: PARA: INT. CL. C07D 477/00; A61P 31/00

Ipc: C07D 477/00 (2011.01), A61P 31/00 (2011.01)

B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]