BRPI0410398A - processo para sintetizar intermediários inibidores de beta-lactamase - Google Patents
processo para sintetizar intermediários inibidores de beta-lactamaseInfo
- Publication number
- BRPI0410398A BRPI0410398A BRPI0410398-0A BRPI0410398A BRPI0410398A BR PI0410398 A BRPI0410398 A BR PI0410398A BR PI0410398 A BRPI0410398 A BR PI0410398A BR PI0410398 A BRPI0410398 A BR PI0410398A
- Authority
- BR
- Brazil
- Prior art keywords
- lactamase inhibitor
- synthesizing beta
- intermediates
- inhibitor intermediates
- beta
- Prior art date
Links
- 239000003781 beta lactamase inhibitor Substances 0.000 title abstract 3
- 229940126813 beta-lactamase inhibitor Drugs 0.000 title abstract 3
- 239000000543 intermediate Substances 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 3
- 230000002194 synthesizing effect Effects 0.000 title 1
- 229940126085 β‑Lactamase Inhibitor Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
"PROCESSO PARA SINTETIZAR INTERMEDIáRIOS INIBIDORES DE BETA-LACTAMASE". A presente invenção refere-se a um processo para a preparação de carboxaldeídos de heteroarila bicíclica tendo a fórmula estrutural I onde X e Y são definidos no relatório descritivo. Os carboxaldeídos de heteroarila bicíclica são úteis como intermediários na preparação de inibidores de <225>lactamase.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47145803P | 2003-05-16 | 2003-05-16 | |
| PCT/US2004/014834 WO2004104006A2 (en) | 2003-05-16 | 2004-05-12 | PROCESS FOR SYNTHESIZING β-LACTAMASE INHIBITOR IN INTERMEDIATES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0410398A true BRPI0410398A (pt) | 2006-07-04 |
Family
ID=33476847
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0410398-0A BRPI0410398A (pt) | 2003-05-16 | 2004-05-12 | processo para sintetizar intermediários inibidores de beta-lactamase |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US7276611B2 (pt) |
| EP (1) | EP1626975A2 (pt) |
| JP (1) | JP2006528978A (pt) |
| CN (1) | CN1823074A (pt) |
| AR (1) | AR044341A1 (pt) |
| AU (1) | AU2004240925A1 (pt) |
| BR (1) | BRPI0410398A (pt) |
| CA (1) | CA2525504A1 (pt) |
| CL (1) | CL2004001038A1 (pt) |
| MX (1) | MXPA05012110A (pt) |
| TW (1) | TW200510430A (pt) |
| WO (1) | WO2004104006A2 (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7115595B2 (en) * | 2000-12-27 | 2006-10-03 | Dainippon Sumitomo Pharma Co., Ltd. | Carbapenem compounds |
| JPWO2004089954A1 (ja) | 2003-04-08 | 2006-07-06 | 大日本住友製薬株式会社 | 新規なカルバペネム化合物 |
| US7276611B2 (en) * | 2003-05-16 | 2007-10-02 | Wyeth Holdings Corporation | Process for synthesizing beta-lactamase inhibitor intermediates |
| CN1823069A (zh) * | 2003-05-16 | 2006-08-23 | 惠氏控股公司 | 合成β－内酰胺酶抑制剂中间体的方法 |
| MXPA06002125A (es) * | 2003-08-25 | 2006-05-31 | Revaax Pharmaceuticals Llc | Composiciones orales de cefazolin neuroterapeutico. |
| TW201245185A (en) | 2011-04-01 | 2012-11-16 | Lundbeck & Co As H | New positive allosteric modulators of nicotinic acetylcholine receptor |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2118181B (en) | 1982-04-08 | 1986-07-30 | Erba Farmitalia | Substituted penem derivatives and new process for their preparation |
| US7276611B2 (en) * | 2003-05-16 | 2007-10-02 | Wyeth Holdings Corporation | Process for synthesizing beta-lactamase inhibitor intermediates |
| CN1823069A (zh) * | 2003-05-16 | 2006-08-23 | 惠氏控股公司 | 合成β－内酰胺酶抑制剂中间体的方法 |
-
2004
- 2004-05-12 US US10/844,243 patent/US7276611B2/en not_active Expired - Fee Related
- 2004-05-12 TW TW093113266A patent/TW200510430A/zh unknown
- 2004-05-12 MX MXPA05012110A patent/MXPA05012110A/es not_active Application Discontinuation
- 2004-05-12 CA CA002525504A patent/CA2525504A1/en not_active Abandoned
- 2004-05-12 JP JP2006532981A patent/JP2006528978A/ja active Pending
- 2004-05-12 CN CNA2004800201170A patent/CN1823074A/zh active Pending
- 2004-05-12 EP EP04751978A patent/EP1626975A2/en not_active Withdrawn
- 2004-05-12 BR BRPI0410398-0A patent/BRPI0410398A/pt not_active Application Discontinuation
- 2004-05-12 AU AU2004240925A patent/AU2004240925A1/en not_active Abandoned
- 2004-05-12 WO PCT/US2004/014834 patent/WO2004104006A2/en not_active Ceased
- 2004-05-13 CL CL200401038A patent/CL2004001038A1/es unknown
- 2004-05-14 AR ARP040101657A patent/AR044341A1/es unknown
-
2007
- 2007-06-18 US US11/820,575 patent/US20080009634A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004104006A2 (en) | 2004-12-02 |
| TW200510430A (en) | 2005-03-16 |
| CA2525504A1 (en) | 2004-12-02 |
| US20080009634A1 (en) | 2008-01-10 |
| CL2004001038A1 (es) | 2005-03-04 |
| EP1626975A2 (en) | 2006-02-22 |
| AU2004240925A1 (en) | 2004-12-02 |
| AR044341A1 (es) | 2005-09-07 |
| US20040242874A1 (en) | 2004-12-02 |
| US7276611B2 (en) | 2007-10-02 |
| JP2006528978A (ja) | 2006-12-28 |
| CN1823074A (zh) | 2006-08-23 |
| WO2004104006A3 (en) | 2005-01-27 |
| MXPA05012110A (es) | 2006-02-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired |