BRPI0411195A - método para a preparação de uma oxazinona fundida e método para a preparação de um composto - Google Patents
método para a preparação de uma oxazinona fundida e método para a preparação de um compostoInfo
- Publication number
- BRPI0411195A BRPI0411195A BRPI0411195-8A BRPI0411195A BRPI0411195A BR PI0411195 A BRPI0411195 A BR PI0411195A BR PI0411195 A BRPI0411195 A BR PI0411195A BR PI0411195 A BRPI0411195 A BR PI0411195A
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- compound
- formula
- carboxylic acid
- fused oxazinone
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 7
- 238000000034 method Methods 0.000 title abstract 7
- FBXGQDUVJBKEAJ-UHFFFAOYSA-N 4h-oxazin-3-one Chemical compound O=C1CC=CON1 FBXGQDUVJBKEAJ-UHFFFAOYSA-N 0.000 title abstract 4
- 150000001732 carboxylic acid derivatives Chemical class 0.000 abstract 4
- VYFOAVADNIHPTR-UHFFFAOYSA-N isatoic anhydride Chemical compound NC1=CC=CC=C1CO VYFOAVADNIHPTR-UHFFFAOYSA-N 0.000 abstract 3
- YBBRCQOCSYXUOC-UHFFFAOYSA-N sulfuryl dichloride Chemical compound ClS(Cl)(=O)=O YBBRCQOCSYXUOC-UHFFFAOYSA-N 0.000 abstract 3
- 150000003512 tertiary amines Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
"MéTODO PARA A PREPARAçãO DE UMA OXAZINONA FUNDIDA E MéTODO PARA A PREPARAçãO DE UM COMPOSTO". Trata-se de um método para a preparação de uma oxazinona fundida no qual um ácido carboxílico é colocado em contato com um cloreto de sulfonila e um anidrido isatóico na presença de uma amina terciária, sendo que a razão molar nominal entre o dito cloreto de sulfonila e o dito ácido carboxílico é de cerca de 1,0 a 1,5 e a razão molar nominal entre o dito anidrido isatóico e o dito ácido carboxílico é de cerca de 0,8 a 1,2. Também é apresentado um método para a preparação de um composto da fórmula (III), ao usar um composto da fórmula (Ia), o qual é caracterizado pela preparação da oxazinona fundida da fórmula (Ia) pelo método acima, ao usar um composto da fórmula LS(O)~ 2~CI como o cloreto de sulfonila, um composto da fórmula (2<39>) como o ácido carboxílico, e um composto da fórmula (5<39>) como o anidrido isatóico, em que L, X, Y e R¬ 1¬ a R¬ 9¬ são tal como definido na descrição.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47787703P | 2003-06-12 | 2003-06-12 | |
| PCT/US2004/019068 WO2004111030A1 (en) | 2003-06-12 | 2004-06-10 | Method for preparing fused oxazinones |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0411195A true BRPI0411195A (pt) | 2006-07-25 |
Family
ID=33551774
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0411195-8A BRPI0411195A (pt) | 2003-06-12 | 2004-06-10 | método para a preparação de uma oxazinona fundida e método para a preparação de um composto |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US7276601B2 (pt) |
| EP (1) | EP1631564A1 (pt) |
| JP (1) | JP4543043B2 (pt) |
| KR (1) | KR20060008336A (pt) |
| CN (1) | CN100376565C (pt) |
| BR (1) | BRPI0411195A (pt) |
| IL (1) | IL172234A (pt) |
| TW (1) | TWI313686B (pt) |
| WO (1) | WO2004111030A1 (pt) |
| ZA (1) | ZA200508771B (pt) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2424840T3 (es) | 2003-01-28 | 2013-10-09 | E.I. Du Pont De Nemours And Company | Insecticidas tipo ciano antranilamida |
| AR048669A1 (es) * | 2004-03-03 | 2006-05-17 | Syngenta Ltd | Derivados biciclicos de bisamida |
| TWI363756B (en) | 2004-12-07 | 2012-05-11 | Du Pont | Method for preparing n-phenylpyrazole-1-carboxamides |
| AR054187A1 (es) * | 2005-04-20 | 2007-06-06 | Syngenta Participations Ag | Derivados de antranilamida con propiedades insecticidas |
| AU2006283181A1 (en) * | 2005-08-24 | 2007-03-01 | E. I. Du Pont De Nemours And Company | Anthranilamides for controlling invertebrate pests |
| UY30090A1 (es) | 2006-01-16 | 2007-08-31 | Syngenta Participations Ag | Insecticidas novedosos |
| PL2066662T3 (pl) | 2006-09-21 | 2013-05-31 | Kyorin Seiyaku Kk | Inhibitory hydrolaz serynowych |
| CN102134238A (zh) * | 2010-01-25 | 2011-07-27 | 中化蓝天集团有限公司 | 一种含一氟甲氧基吡唑的4h-苯并[1,3]噁嗪-4-酮类化合物、其制备方法及应用 |
| CA2894399A1 (en) | 2012-12-06 | 2014-06-12 | Quanticel Pharmaceuticals, Inc. | Histone demethylase inhibitors |
| CA3129876A1 (en) | 2019-02-18 | 2020-08-27 | Pi Industries Ltd. | A process for preparing anthranilic diamides and intermediates thereof |
| TW202222162A (zh) | 2020-09-26 | 2022-06-16 | 印度商皮埃企業有限公司 | 鄰胺苯甲酸/醯胺化合物及其中間體的合成方法 |
| EP4380363A1 (en) | 2021-08-05 | 2024-06-12 | Syngenta Crop Protection AG | Method for controlling diamide resistant pests & compounds therefor |
| US20240327395A1 (en) * | 2021-11-02 | 2024-10-03 | Tagros Chemicals India Pvt Ltd | A process for preparing benzoxazinone compounds |
| WO2023110710A1 (en) | 2021-12-13 | 2023-06-22 | Syngenta Crop Protection Ag | Method for controlling diamide resistant pests & compounds therefor |
| WO2024133426A1 (en) | 2022-12-21 | 2024-06-27 | Syngenta Crop Protection Ag | Method for controlling diamide resistant pests and compounds therefor |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY138097A (en) * | 2000-03-22 | 2009-04-30 | Du Pont | Insecticidal anthranilamides |
| US20040102324A1 (en) * | 2002-02-28 | 2004-05-27 | Annis Gary David | Heterocyclic diamide invertebrate pest control agents |
| RU2299198C2 (ru) * | 2001-05-21 | 2007-05-20 | Е.И.Дюпон Де Немур Энд Компани | Диамиды антраниловой кислоты, способ борьбы с насекомыми, композиция для борьбы с насекомыми |
| TWI356822B (en) * | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| TWI312274B (en) * | 2001-08-13 | 2009-07-21 | Du Pont | Method for controlling particular insect pests by applying anthranilamide compounds |
| AR036872A1 (es) * | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| US7038057B2 (en) * | 2001-08-13 | 2006-05-02 | E.I. Du Pont De Nemours And Company | Substituted 1H-dihydropyrazoles, their preparation and use |
| AU2002331706B2 (en) * | 2001-08-15 | 2009-01-22 | E.I. Du Pont De Nemours And Company | Ortho-substituted aryl amides for controlling invertebrate pests |
| BR0212183B1 (pt) * | 2001-08-16 | 2014-10-21 | Du Pont | composto de antranilamida substituída, seus n-óxidos e sais, método para o controle de uma praga invertebrada e composição para o controle de uma praga invertebrada |
| TWI283164B (en) * | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| WO2003027099A1 (en) * | 2001-09-21 | 2003-04-03 | E. I. Du Pont De Nemours And Company | Arthropodicidal anthranilamides |
| US20040110777A1 (en) * | 2001-12-03 | 2004-06-10 | Annis Gary David | Quinazolinones and pyridinylpyrimidinones for controlling invertebrate pests |
| BR0307178A (pt) * | 2002-01-22 | 2004-12-07 | Du Pont | Composto, composição e método para controle de pragas invertebradas |
| WO2003062221A1 (en) * | 2002-01-22 | 2003-07-31 | E.I. Du Pont De Nemours And Company | Diamide invertebrate pest control agents |
| AU2003245466A1 (en) * | 2002-06-11 | 2003-12-22 | E.I. Du Pont De Nemours And Company | Insecticidal amides with nitrogen-containing benzo-fused bicyclic ring systems |
| BR0311707A (pt) | 2002-06-13 | 2005-03-15 | Du Pont | Composto, composição e método de controle de pelo menos uma praga invertebrada |
| TWI343376B (en) * | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
| TWI326283B (en) * | 2002-07-31 | 2010-06-21 | Du Pont | Method for preparing fused oxazinones |
| AU2003282711A1 (en) | 2002-10-04 | 2004-05-04 | E.I. Du Pont De Nemours And Company | Anthranilamide insecticides |
| MXPA05005025A (es) | 2002-11-15 | 2005-08-03 | Du Pont | Nuevos insecticidas de antranilamida. |
| ES2424840T3 (es) | 2003-01-28 | 2013-10-09 | E.I. Du Pont De Nemours And Company | Insecticidas tipo ciano antranilamida |
| TWI367882B (en) | 2003-03-26 | 2012-07-11 | Du Pont | Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates |
-
2004
- 2004-06-10 EP EP04755313A patent/EP1631564A1/en not_active Ceased
- 2004-06-10 CN CNB2004800163408A patent/CN100376565C/zh not_active Expired - Lifetime
- 2004-06-10 JP JP2006533800A patent/JP4543043B2/ja not_active Expired - Fee Related
- 2004-06-10 WO PCT/US2004/019068 patent/WO2004111030A1/en not_active Ceased
- 2004-06-10 US US10/554,090 patent/US7276601B2/en not_active Expired - Lifetime
- 2004-06-10 KR KR1020057023611A patent/KR20060008336A/ko not_active Ceased
- 2004-06-10 BR BRPI0411195-8A patent/BRPI0411195A/pt not_active IP Right Cessation
- 2004-06-10 ZA ZA200508771A patent/ZA200508771B/en unknown
- 2004-06-11 TW TW093116971A patent/TWI313686B/zh not_active IP Right Cessation
-
2005
- 2005-11-29 IL IL172234A patent/IL172234A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CN1805950A (zh) | 2006-07-19 |
| US20060241304A1 (en) | 2006-10-26 |
| JP4543043B2 (ja) | 2010-09-15 |
| EP1631564A1 (en) | 2006-03-08 |
| TWI313686B (en) | 2009-08-21 |
| ZA200508771B (en) | 2008-04-30 |
| TW200504058A (en) | 2005-02-01 |
| US7276601B2 (en) | 2007-10-02 |
| AU2004247738A1 (en) | 2004-12-23 |
| IL172234A (en) | 2012-07-31 |
| CN100376565C (zh) | 2008-03-26 |
| JP2007501867A (ja) | 2007-02-01 |
| IL172234A0 (en) | 2006-04-10 |
| WO2004111030A1 (en) | 2004-12-23 |
| KR20060008336A (ko) | 2006-01-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 12A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2385 DE 20-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |