BRPI0411837A - pirazolopirimidinas - Google Patents

pirazolopirimidinas

Info

Publication number
BRPI0411837A
BRPI0411837A BRPI0411837-5A BRPI0411837A BRPI0411837A BR PI0411837 A BRPI0411837 A BR PI0411837A BR PI0411837 A BRPI0411837 A BR PI0411837A BR PI0411837 A BRPI0411837 A BR PI0411837A
Authority
BR
Brazil
Prior art keywords
sup
pyrazolopyrimidines
producing
materials
methods
Prior art date
Application number
BRPI0411837-5A
Other languages
English (en)
Inventor
Olaf Gebauer
Ulrich Heinemann
Stefan Herrmann
Oliver Guth
Hans-Ludwig Elbe
Herbert Gayer
J Rg Nico Greul
Stefan Hillebrand
Ronald Ebbert
Ulrike Wachendorff Neumann
Peter Dahmen
Karl-Heinz Kuck
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10339360A external-priority patent/DE10339360A1/de
Priority claimed from DE2003157570 external-priority patent/DE10357570A1/de
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BRPI0411837A publication Critical patent/BRPI0411837A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/55—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pest Control & Pesticides (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

"PIRAZOLOPIRIMIDINAS". A presente invenção refere-se a novas pirazolopirimidinas da fórmula (I), na qual R¬ 1¬, R¬ 2¬, R¬ 3¬, R¬ 4¬, X e Hal têm os significados especificados na descrição, vários processos para a produção desses materiais e seu emprego para o combate de microorganismos indesejáveis. Novos produtos intermediários das fórmulas (II), (X), (XII-a) e (XII-b) e processos para a produção desses materiais.
BRPI0411837-5A 2003-06-27 2004-06-18 pirazolopirimidinas BRPI0411837A (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE10328996 2003-06-27
DE10339360A DE10339360A1 (de) 2003-06-27 2003-08-27 Pyrazolopyrimidine
DE2003157570 DE10357570A1 (de) 2003-12-10 2003-12-10 Pyrazolopyrimidine
PCT/EP2004/006609 WO2005000851A1 (de) 2003-06-27 2004-06-18 Pyrazolopyrimidine

Publications (1)

Publication Number Publication Date
BRPI0411837A true BRPI0411837A (pt) 2006-08-08

Family

ID=33555888

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0411837-5A BRPI0411837A (pt) 2003-06-27 2004-06-18 pirazolopirimidinas

Country Status (11)

Country Link
US (1) US20070037828A1 (pt)
EP (1) EP1641800B1 (pt)
JP (1) JP2007506665A (pt)
KR (1) KR20060027809A (pt)
AT (1) ATE388138T1 (pt)
AU (1) AU2004251845A1 (pt)
BR (1) BRPI0411837A (pt)
CA (1) CA2530378A1 (pt)
DE (1) DE502004006422D1 (pt)
MX (1) MXPA05013902A (pt)
WO (1) WO2005000851A1 (pt)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10357565A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE102004008807A1 (de) 2004-02-20 2005-09-08 Bayer Cropscience Ag Pyrazolopyrimidine
DE102005007534A1 (de) * 2005-02-17 2006-08-31 Bayer Cropscience Ag Pyrazolopyrimidine
JP2007008864A (ja) * 2005-06-30 2007-01-18 Bayer Cropscience Ag ピラゾロピリミジン誘導体及び農園芸用殺菌剤
WO2007024680A1 (en) 2005-08-22 2007-03-01 Amgen Inc. Pyrazolopyridine and pyrazolopyrimidine compounds useful as kinase enzymes modulators
WO2007101859A1 (de) * 2006-03-07 2007-09-13 Basf Se Substituierte pyrazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
WO2008046856A2 (de) * 2006-10-18 2008-04-24 Basf Se Fungizide zusammensetzungen
EP2014661A1 (de) * 2007-06-13 2009-01-14 Bayer CropScience AG Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate
ES2688584T3 (es) 2014-02-25 2018-11-05 Saudi Basic Industries Corporation Proceso para producir btx a partir de una fuente de hidrocarburo mixto usando coquización
EA039640B1 (ru) 2014-02-25 2022-02-21 Сауди Бейсик Индастриз Корпорейшн Способ получения продукта бтк из смешанного углеводородного источника при использовании пиролиза
SG11201606519WA (en) 2014-02-25 2016-09-29 Saudi Basic Ind Corp Process and installation for the conversion of crude oil to petrochemicals having an improved ethylene and btx yield
ES2681801T3 (es) 2014-02-25 2018-09-17 Saudi Basic Industries Corporation Proceso para producir BTX a partir de una fuente mixta de hidrocarburos mediante el uso de craqueo catalítico
KR102467347B1 (ko) 2016-04-15 2022-11-14 바이엘 애니멀 헬스 게엠베하 피라졸로피리미딘 유도체
KR102912267B1 (ko) * 2023-04-20 2026-01-15 한국화학연구원 신규한 헤테로고리 화합물 또는 이의 약학적으로 허용가능한 염 및 이를 유효성분으로 포함하는 바이러스성 질환의 예방 또는 치료용 약학적 조성물

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3130633A1 (de) * 1981-08-01 1983-02-17 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)pyrimidine und diese enthaltende fungizide
US4908056A (en) * 1986-04-25 1990-03-13 E. I. Du Pont De Nemours And Company Heterocyclic acyl sulfonamides
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
US5817663A (en) * 1996-10-07 1998-10-06 American Cyanamid Company Pentafluorophenylazolopyrimidines
JP2001019693A (ja) * 1999-06-14 2001-01-23 American Cyanamid Co 殺菌・殺カビ性６−フェニル−ピラゾロピリミジン
GB0126914D0 (en) * 2001-11-08 2002-01-02 Syngenta Ltd Fungicides
DE10223917A1 (de) * 2002-05-29 2003-12-11 Bayer Cropscience Ag Pyrazolopyrimidine

Also Published As

Publication number Publication date
MXPA05013902A (es) 2006-02-24
US20070037828A1 (en) 2007-02-15
WO2005000851A1 (de) 2005-01-06
CA2530378A1 (en) 2005-01-06
EP1641800A1 (de) 2006-04-05
AU2004251845A1 (en) 2005-01-06
DE502004006422D1 (en) 2008-04-17
EP1641800B1 (de) 2008-03-05
KR20060027809A (ko) 2006-03-28
JP2007506665A (ja) 2007-03-22
ATE388138T1 (de) 2008-03-15

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE 5A., 6A. E 7A. ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE AS 5A, 6A E 7A ANUIDADES.