BRPI0413682A - compostos, composição farmacêutica e respectivos métodos de preparação, de tratamento de infecção microbiana e de extermìnio de microrganismo e usos - Google Patents
compostos, composição farmacêutica e respectivos métodos de preparação, de tratamento de infecção microbiana e de extermìnio de microrganismo e usosInfo
- Publication number
- BRPI0413682A BRPI0413682A BRPI0413682-9A BRPI0413682A BRPI0413682A BR PI0413682 A BRPI0413682 A BR PI0413682A BR PI0413682 A BRPI0413682 A BR PI0413682A BR PI0413682 A BRPI0413682 A BR PI0413682A
- Authority
- BR
- Brazil
- Prior art keywords
- compounds
- methods
- extermination
- microorganism
- pharmaceutical composition
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 6
- 238000000034 method Methods 0.000 title abstract 4
- 208000015181 infectious disease Diseases 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- 230000000813 microbial effect Effects 0.000 title abstract 2
- 244000005700 microbiome Species 0.000 title abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- QAZLUNIWYYOJPC-UHFFFAOYSA-M sulfenamide Chemical compound [Cl-].COC1=C(C)C=[N+]2C3=NC4=CC=C(OC)C=C4N3SCC2=C1C QAZLUNIWYYOJPC-UHFFFAOYSA-M 0.000 abstract 1
- 230000002194 synthesizing effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Crystallography & Structural Chemistry (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Epidemiology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
"COMPOSTOS, COMPOSIçãO FARMACêUTICA E RESPECTIVOS MéTODOS DE PREPARAçãO DE TRATAMENTO DE INFECçãO MICROBIANA E DE EXTERMìNIO DE MICROORGANISMO E USOS". São apresentados compostos de óxido de sulfenamida da fórmula geral (I), em que A, R~ 1~, R~ 2~, X~ 1~, X~ 1~<39>, X~ 2~, X~ 2~<39>, X~ 3~, X~ 4~, X~ 4~<39>, X~ 5~ e X~ 5~<39> definem muitas variáveis e em que q é O ou 1 e p é 1 ou 2. Os compostos apresentados nos exemplos são os compostos de óxido de sulfenamida galactofuranosil e glucofuranosil, em que a variável A é o oxigenio. Também são apresentados métodos de síntese dos compostos de fórmula geral (I), composições farmacêuticas que os contenham e métodos de uso no tratamento de pacientes que estejam sofrendo de infecção microbiana.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2003904500A AU2003904500A0 (en) | 2003-08-21 | Novel compounds II | |
| AU2003904501A AU2003904501A0 (en) | 2003-08-21 | Novel compounds III | |
| PCT/AU2004/001110 WO2005019236A1 (en) | 2003-08-21 | 2004-08-20 | Novel sulfenamide oxides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0413682A true BRPI0413682A (pt) | 2006-10-24 |
Family
ID=34218927
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0413682-9A BRPI0413682A (pt) | 2003-08-21 | 2004-08-20 | compostos, composição farmacêutica e respectivos métodos de preparação, de tratamento de infecção microbiana e de extermìnio de microrganismo e usos |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1664071A1 (pt) |
| JP (1) | JP2007502778A (pt) |
| BR (1) | BRPI0413682A (pt) |
| CA (1) | CA2535800A1 (pt) |
| MX (1) | MXPA06001974A (pt) |
| RU (1) | RU2006108577A (pt) |
| WO (1) | WO2005019236A1 (pt) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7601716B2 (en) | 2006-05-01 | 2009-10-13 | Cephalon, Inc. | Pyridopyrazines and derivatives thereof as ALK and c-Met inhibitors |
| CN102282155B (zh) | 2008-12-02 | 2017-06-09 | 日本波涛生命科学公司 | 磷原子修饰的核酸的合成方法 |
| RU2612521C2 (ru) | 2009-07-06 | 2017-03-09 | Онтории, Инк. | Новые пролекарства нуклеиновых кислот и способы их применения |
| JP5868324B2 (ja) | 2010-09-24 | 2016-02-24 | 株式会社Wave Life Sciences Japan | 不斉補助基 |
| CN103796657B (zh) | 2011-07-19 | 2017-07-11 | 波涛生命科学有限公司 | 合成官能化核酸的方法 |
| PL2872485T3 (pl) | 2012-07-13 | 2021-05-31 | Wave Life Sciences Ltd. | Asymetryczna grupa pomocnicza |
| BR112016016400A2 (pt) | 2014-01-16 | 2017-10-03 | Wave Life Sciences Ltd | Composições de oligonucleotídeos quiralmente controlados, seu uso, sua composição farmacêutica, e métodos |
| CA3033867A1 (en) | 2016-08-17 | 2018-02-22 | Solstice Biologics, Ltd. | Polynucleotide constructs |
| US11597744B2 (en) | 2017-06-30 | 2023-03-07 | Sirius Therapeutics, Inc. | Chiral phosphoramidite auxiliaries and methods of their use |
| BR112022010924A2 (pt) | 2019-12-06 | 2022-09-06 | Vertex Pharma | Tetra-hidrofuranos substituídos como moduladores de canais de sódio |
| JP2023527792A (ja) | 2020-05-27 | 2023-06-30 | アキシャル セラピューティクス，インク． | Ｔｌｒ２調節剤化合物、医薬組成物、及びそれらの使用 |
| SMT202500481T1 (it) | 2021-06-04 | 2026-01-12 | Vertex Pharma | N-(idrossialchil(etero)aril)tetraidrofuran carbossammidi come modulatori di canali del sodio |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005523904A (ja) * | 2002-02-22 | 2005-08-11 | グリフィス ユニバーシティ | 抗菌剤 |
-
2004
- 2004-08-20 EP EP04761147A patent/EP1664071A1/en not_active Withdrawn
- 2004-08-20 RU RU2006108577/04A patent/RU2006108577A/ru not_active Application Discontinuation
- 2004-08-20 BR BRPI0413682-9A patent/BRPI0413682A/pt not_active Application Discontinuation
- 2004-08-20 CA CA002535800A patent/CA2535800A1/en not_active Abandoned
- 2004-08-20 JP JP2006523486A patent/JP2007502778A/ja active Pending
- 2004-08-20 WO PCT/AU2004/001110 patent/WO2005019236A1/en not_active Ceased
- 2004-08-20 MX MXPA06001974A patent/MXPA06001974A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EP1664071A1 (en) | 2006-06-07 |
| CA2535800A1 (en) | 2005-03-03 |
| RU2006108577A (ru) | 2007-09-27 |
| JP2007502778A (ja) | 2007-02-15 |
| WO2005019236A1 (en) | 2005-03-03 |
| MXPA06001974A (es) | 2006-05-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired |