BRPI0415280A - methods for treating vasomotor symptoms - Google Patents
methods for treating vasomotor symptomsInfo
- Publication number
- BRPI0415280A BRPI0415280A BRPI0415280-8A BRPI0415280A BRPI0415280A BR PI0415280 A BRPI0415280 A BR PI0415280A BR PI0415280 A BRPI0415280 A BR PI0415280A BR PI0415280 A BRPI0415280 A BR PI0415280A
- Authority
- BR
- Brazil
- Prior art keywords
- methods
- vasomotor symptoms
- combination
- selective
- receptor antagonists
- Prior art date
Links
- 230000001457 vasomotor Effects 0.000 title abstract 3
- 208000024891 symptom Diseases 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 4
- 239000002767 noradrenalin uptake inhibitor Substances 0.000 abstract 4
- 229940127221 norepinephrine reuptake inhibitor Drugs 0.000 abstract 4
- 239000000674 adrenergic antagonist Substances 0.000 abstract 3
- 230000009977 dual effect Effects 0.000 abstract 1
- 239000003775 serotonin noradrenalin reuptake inhibitor Substances 0.000 abstract 1
- 229940126570 serotonin reuptake inhibitor Drugs 0.000 abstract 1
- 239000003772 serotonin uptake inhibitor Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
"MéTODOS PARA O TRATAMENTO DE SINTOMAS VASOMOTORES". A presente invenção se refere a antagonistas seletivos do receptor adrenérgiCO<244>~ 2B~ isolados, dos antagonistas seletivos do receptor adrenérgico<244>~ 2B~ em combinação com inibidores da reabsorção da norepinefrina (NRI) (como um único composto ou como uma combinação de dois ou mais compostos), ou de antagonistas seletivos do receptor adrenérgico<244>~ 2B~ em combinação com inibidores duplos de reabsorção da norepinefrina/inibidor da reabsorção da serotonina (NRI/SRI) (como um único composto ou como uma combinação de dois ou mais compostos), e a métodos para o uso dos mesmos para o tratamento de sintomas vasomotores."METHODS FOR TREATMENT OF VASOMOTOR SYMPTOMS". The present invention relates to selective β2B2-adrenergic receptor antagonists isolated from selective β2B2-adrenergic receptor antagonists in combination with norepinephrine reuptake inhibitors (NRI) (as a single compound or as a combination of two or more compounds), or selective β2B adrenergic receptor antagonists in combination with dual norepinephrine reuptake inhibitor / serotonin reuptake inhibitor (NRI / SRI) (as a single compound or as a combination two or more compounds), and methods for using them to treat vasomotor symptoms.
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51089703P | 2003-10-14 | 2003-10-14 | |
| US10/685,812 US20040152710A1 (en) | 2002-10-15 | 2003-10-14 | Use of norepinephrine reuptake modulators for preventing and treating vasomotor symptoms |
| PCT/US2003/032759 WO2004035058A1 (en) | 2002-10-15 | 2003-10-15 | Use of norepinephrine reuptake modulators for preventing and treating vasomotor symptoms |
| US10/962,897 US20050130987A1 (en) | 2003-10-14 | 2004-10-12 | Methods of treating vasomotor symptoms |
| PCT/US2004/033754 WO2005037260A2 (en) | 2003-10-14 | 2004-10-13 | Use of adrenergic alphaze antagonists for the treatment of vasomotor symptoms |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0415280A true BRPI0415280A (en) | 2006-12-19 |
Family
ID=36566007
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0415280-8A BRPI0415280A (en) | 2003-10-14 | 2004-10-13 | methods for treating vasomotor symptoms |
Country Status (4)
| Country | Link |
|---|---|
| JP (1) | JP2007515395A (en) |
| BR (1) | BRPI0415280A (en) |
| CA (1) | CA2539757A1 (en) |
| TW (1) | TW200526227A (en) |
-
2004
- 2004-10-13 CA CA002539757A patent/CA2539757A1/en not_active Abandoned
- 2004-10-13 BR BRPI0415280-8A patent/BRPI0415280A/en not_active IP Right Cessation
- 2004-10-13 JP JP2006535623A patent/JP2007515395A/en not_active Withdrawn
- 2004-10-13 TW TW093130953A patent/TW200526227A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TW200526227A (en) | 2005-08-16 |
| JP2007515395A (en) | 2007-06-14 |
| CA2539757A1 (en) | 2005-04-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE A 6A E 7A ANUIDADE(S) |
|
| B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2129 DE 25/10/2011. |