BRPI0417158A - composto, composição farmacêutica, uso de um composto, método para prevenir, tratar ou melhorar uma doença ou condição associada com angiogênese desregulada, e, métodos para tratar ou melhorar cáncer, para reduzir o potencial metastático de um tumor, e para tratar ou melhorar tumores, e uma condição ou doença - Google Patents

composto, composição farmacêutica, uso de um composto, método para prevenir, tratar ou melhorar uma doença ou condição associada com angiogênese desregulada, e, métodos para tratar ou melhorar cáncer, para reduzir o potencial metastático de um tumor, e para tratar ou melhorar tumores, e uma condição ou doença

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Publication number
BRPI0417158A
BRPI0417158A BRPI0417158-6A BRPI0417158A BRPI0417158A BR PI0417158 A BRPI0417158 A BR PI0417158A BR PI0417158 A BRPI0417158 A BR PI0417158A BR PI0417158 A BRPI0417158 A BR PI0417158A
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BR
Brazil
Prior art keywords
treating
ameliorating
disease
compound
condition
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BRPI0417158-6A
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English (en)
Inventor
Jef Fensholdt
Jacob Thorhauge
Bjarne Norremark
Original Assignee
Leo Pharma As
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Publication date
Application filed by Leo Pharma As filed Critical Leo Pharma As
Publication of BRPI0417158A publication Critical patent/BRPI0417158A/pt

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Abstract

"COMPOSTO, COMPOSIçãO FARMACêUTICA, USO DE UM COMPOSTO, MéTODO PARA PREVENIR, TRATAR OU MELHORAR UMA DOENçA OU CONDIçãO ASSOCIADA COM ANGIOGêNESE DESREGULADA, E, METODOS PARA TRATAR OU MELHORAR CáNCER, PARA REDUZIR O POTENCIAL METASTáTICO DE UM TUMOR, E PARA TRATAR OU MELHORAR TUMORES, E UMA CONDIçãO OU DOENçA". A invenção refere-se a compostos de fórmula geral I, sendo que D, E, F, G, W, Y R~ 1~, A, R~ 9~, X, B, R~ 8~ são como definido aqui, e sais, hidratos, ou solvatos farmaceuticamente aceitáveis dos mesmos, para uso sozinhos ou em combinação com um ou mais outros compostos farmaceuticamente ativos na terapia, para tratar doenças associadas com angiogêneseI desregulada, como, câncer.
BRPI0417158-6A 2003-12-03 2004-12-02 composto, composição farmacêutica, uso de um composto, método para prevenir, tratar ou melhorar uma doença ou condição associada com angiogênese desregulada, e, métodos para tratar ou melhorar cáncer, para reduzir o potencial metastático de um tumor, e para tratar ou melhorar tumores, e uma condição ou doença BRPI0417158A (pt)

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US52626203P 2003-12-03 2003-12-03
PCT/DK2004/000840 WO2005054179A2 (en) 2003-12-03 2004-12-02 Hydroxamic acid esters and pharmaceutical use thereof

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US (1) US8034811B2 (pt)
EP (1) EP1697312B1 (pt)
JP (1) JP2007513098A (pt)
KR (1) KR20070026337A (pt)
CN (1) CN1906155B (pt)
AR (1) AR046785A1 (pt)
AT (1) ATE517081T1 (pt)
AU (1) AU2004295022A1 (pt)
BR (1) BRPI0417158A (pt)
CA (1) CA2549242A1 (pt)
IL (1) IL175480A0 (pt)
MX (1) MXPA06006210A (pt)
NO (1) NO20062905L (pt)
NZ (1) NZ547231A (pt)
RU (1) RU2357952C2 (pt)
TW (1) TW200529815A (pt)
UA (1) UA89035C2 (pt)
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EP1697312B1 (en) 2011-07-20
MXPA06006210A (es) 2006-08-25
CN1906155A (zh) 2007-01-31
US8034811B2 (en) 2011-10-11
CA2549242A1 (en) 2005-06-16
US20070244117A1 (en) 2007-10-18
JP2007513098A (ja) 2007-05-24
ATE517081T1 (de) 2011-08-15
EP1697312A2 (en) 2006-09-06
UA89035C2 (ru) 2009-12-25
RU2357952C2 (ru) 2009-06-10
AR046785A1 (es) 2005-12-21
NO20062905L (no) 2006-06-21
KR20070026337A (ko) 2007-03-08
TW200529815A (en) 2005-09-16
AU2004295022A1 (en) 2005-06-16
IL175480A0 (en) 2006-09-05
NZ547231A (en) 2010-02-26
ZA200603873B (en) 2008-10-29
CN1906155B (zh) 2010-06-23
HK1098127A1 (en) 2007-07-13
WO2005054179A3 (en) 2005-08-04
WO2005054179A2 (en) 2005-06-16

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