BRPI0510084A - benzoxazina para tratamento de doenças do trato respiratório - Google Patents
benzoxazina para tratamento de doenças do trato respiratórioInfo
- Publication number
- BRPI0510084A BRPI0510084A BRPI0510084-4A BRPI0510084A BRPI0510084A BR PI0510084 A BRPI0510084 A BR PI0510084A BR PI0510084 A BRPI0510084 A BR PI0510084A BR PI0510084 A BRPI0510084 A BR PI0510084A
- Authority
- BR
- Brazil
- Prior art keywords
- respiratory tract
- benzoxazine
- treatment
- tract diseases
- relates
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Virology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
BENZOXAZINA PARA TRATAMENTO DE DOENçAS DO TRATO RESPIRATóRIO. A presente invenção refere-se ao uso dos compostos de fórmula geral <UM>1<MV>, em que os grupos R¬ 1¬, R¬ 2¬ e R¬ 3¬ podem ter os significados dados nas reivindicações e na descrição. A invenção também refere-se á produção de um medicamento para o tratamento de doenças do trato respiratório.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004019539A DE102004019539A1 (de) | 2004-04-22 | 2004-04-22 | Neue Arzneimittel zur Behandlung von Atemwegserkrankungen |
| PCT/EP2005/004075 WO2005102350A1 (de) | 2004-04-22 | 2005-04-18 | Benzoxazine zur behandlung von atemwegserkrankungen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0510084A true BRPI0510084A (pt) | 2007-10-16 |
Family
ID=34966948
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0510084-4A BRPI0510084A (pt) | 2004-04-22 | 2005-04-18 | benzoxazina para tratamento de doenças do trato respiratório |
Country Status (20)
| Country | Link |
|---|---|
| EP (1) | EP1765355B1 (pt) |
| JP (1) | JP2007533684A (pt) |
| KR (2) | KR20130042662A (pt) |
| CN (1) | CN1946406A (pt) |
| AU (1) | AU2005235420C1 (pt) |
| BR (1) | BRPI0510084A (pt) |
| CA (1) | CA2559700C (pt) |
| DE (1) | DE102004019539A1 (pt) |
| DK (1) | DK1765355T3 (pt) |
| EA (1) | EA012045B1 (pt) |
| EC (1) | ECSP066948A (pt) |
| ES (1) | ES2403184T3 (pt) |
| IL (1) | IL177663A (pt) |
| NO (1) | NO20065061L (pt) |
| NZ (1) | NZ551272A (pt) |
| PL (1) | PL1765355T3 (pt) |
| SG (1) | SG152233A1 (pt) |
| UA (1) | UA85707C2 (pt) |
| WO (1) | WO2005102350A1 (pt) |
| ZA (1) | ZA200606547B (pt) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7056916B2 (en) | 2002-11-15 | 2006-06-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Medicaments for the treatment of chronic obstructive pulmonary disease |
| DE102004024452A1 (de) * | 2004-05-14 | 2005-12-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Aerosolformulierung für die Inhalation von Betaagonisten |
| US7220742B2 (en) | 2004-05-14 | 2007-05-22 | Boehringer Ingelheim International Gmbh | Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments |
| ES2530991T3 (es) | 2005-08-15 | 2015-03-09 | Boehringer Ingelheim Int | Procedimiento para la obtención de betamiméticos |
| US20080280897A1 (en) * | 2005-11-09 | 2008-11-13 | Michael Aven | Aerosol Formulation for Inhalation |
| GB0601951D0 (en) | 2006-01-31 | 2006-03-15 | Novartis Ag | Organic compounds |
| KR20100113557A (ko) | 2008-01-11 | 2010-10-21 | 노파르티스 아게 | 키나제 억제제로서의 피리미딘 |
| WO2012034095A1 (en) | 2010-09-09 | 2012-03-15 | Irm Llc | Compounds and compositions as trk inhibitors |
| UY33597A (es) | 2010-09-09 | 2012-04-30 | Irm Llc | Compuestos y composiciones como inhibidores de la trk |
| KR20140014184A (ko) | 2011-02-25 | 2014-02-05 | 아이알엠 엘엘씨 | Trk 억제제로서의 화합물 및 조성물 |
| US9784726B2 (en) | 2013-01-08 | 2017-10-10 | Atrogi Ab | Screening method, a kit, a method of treatment and a compound for use in a method of treatment |
| JP2019536812A (ja) | 2016-12-12 | 2019-12-19 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | オロダテロールとの同時投与による間質性肺疾患の処置方法に使用するためのニンテダニブ |
| GB201714740D0 (en) | 2017-09-13 | 2017-10-25 | Atrogi Ab | New compounds and uses |
| GB201714745D0 (en) | 2017-09-13 | 2017-10-25 | Atrogi Ab | New compounds and uses |
| GB201714736D0 (en) | 2017-09-13 | 2017-10-25 | Atrogi Ab | New compounds and uses |
| GB201714734D0 (en) | 2017-09-13 | 2017-10-25 | Atrogi Ab | New compounds and uses |
| GB201903832D0 (en) | 2019-03-20 | 2019-05-01 | Atrogi Ab | New compounds and methods |
| GB202205895D0 (en) | 2022-04-22 | 2022-06-08 | Atrogi Ab | New medical uses |
| EP4651867A1 (en) | 2023-01-20 | 2025-11-26 | Atrogi AB | Beta 2-adrenergic receptor agonists for treatment or prevention of muscle wasting |
| GB202302225D0 (en) | 2023-02-16 | 2023-04-05 | Atrogi Ab | New medical uses |
| GB202303229D0 (en) | 2023-03-06 | 2023-04-19 | Atrogi Ab | New medical uses |
| GB202403169D0 (en) | 2024-03-05 | 2024-04-17 | Atrogi Ab | New medical uses |
| WO2025238248A1 (en) | 2024-05-17 | 2025-11-20 | Atrogi Ab | USE OF β2-ADRENERGIC RECEPTOR AGONISTS IN TREATING MUSCLE WASTING |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4460581A (en) * | 1982-10-12 | 1984-07-17 | Boehringer Ingelheim Kg | (1-Hydroxy-2-amino-alkyl)-substituted benzoxazinones and benzoxazolinones |
| CN1426401A (zh) * | 2000-04-27 | 2003-06-25 | 贝林格尔英格海姆法玛公司 | 新的长效倍他米美类药物(betamimetics)其制备方法,及其作为药物组合物的用途 |
| DE10130371A1 (de) * | 2001-06-23 | 2003-01-02 | Boehringer Ingelheim Pharma | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika, Corticosteroiden und Betamimetika |
| DE10253282A1 (de) * | 2002-11-15 | 2004-05-27 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Arzneimittel zur Behandlung von chronisch obstruktiver Lungenerkrankung |
-
2004
- 2004-04-22 DE DE102004019539A patent/DE102004019539A1/de not_active Withdrawn
-
2005
- 2005-04-18 ES ES05740045T patent/ES2403184T3/es not_active Expired - Lifetime
- 2005-04-18 PL PL05740045T patent/PL1765355T3/pl unknown
- 2005-04-18 DK DK05740045.9T patent/DK1765355T3/da active
- 2005-04-18 EP EP05740045A patent/EP1765355B1/de not_active Expired - Lifetime
- 2005-04-18 CA CA2559700A patent/CA2559700C/en not_active Expired - Lifetime
- 2005-04-18 EA EA200601837A patent/EA012045B1/ru not_active IP Right Cessation
- 2005-04-18 KR KR1020137008584A patent/KR20130042662A/ko not_active Ceased
- 2005-04-18 AU AU2005235420A patent/AU2005235420C1/en not_active Ceased
- 2005-04-18 SG SG200902504-0A patent/SG152233A1/en unknown
- 2005-04-18 UA UAA200612036A patent/UA85707C2/ru unknown
- 2005-04-18 WO PCT/EP2005/004075 patent/WO2005102350A1/de not_active Ceased
- 2005-04-18 CN CNA200580012623XA patent/CN1946406A/zh active Pending
- 2005-04-18 BR BRPI0510084-4A patent/BRPI0510084A/pt not_active IP Right Cessation
- 2005-04-18 JP JP2007508807A patent/JP2007533684A/ja active Pending
- 2005-04-18 KR KR1020067024543A patent/KR101338947B1/ko not_active Expired - Fee Related
- 2005-04-18 NZ NZ551272A patent/NZ551272A/en not_active IP Right Cessation
-
2006
- 2006-08-07 ZA ZA200606547A patent/ZA200606547B/xx unknown
- 2006-08-23 IL IL177663A patent/IL177663A/en not_active IP Right Cessation
- 2006-10-23 EC EC2006006948A patent/ECSP066948A/es unknown
- 2006-11-02 NO NO20065061A patent/NO20065061L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20070054599A (ko) | 2007-05-29 |
| KR101338947B1 (ko) | 2013-12-10 |
| CA2559700C (en) | 2013-06-11 |
| CA2559700A1 (en) | 2005-11-03 |
| AU2005235420A1 (en) | 2005-11-03 |
| NZ551272A (en) | 2010-10-29 |
| EA012045B1 (ru) | 2009-08-28 |
| KR20130042662A (ko) | 2013-04-26 |
| ECSP066948A (es) | 2006-12-20 |
| SG152233A1 (en) | 2009-05-29 |
| DK1765355T3 (da) | 2013-04-08 |
| IL177663A (en) | 2014-04-30 |
| UA85707C2 (ru) | 2009-02-25 |
| DE102004019539A1 (de) | 2005-11-10 |
| AU2005235420B2 (en) | 2010-10-28 |
| AU2005235420C1 (en) | 2011-02-24 |
| EP1765355B1 (de) | 2013-03-06 |
| JP2007533684A (ja) | 2007-11-22 |
| CN1946406A (zh) | 2007-04-11 |
| WO2005102350A1 (de) | 2005-11-03 |
| EP1765355A1 (de) | 2007-03-28 |
| IL177663A0 (en) | 2006-12-31 |
| ES2403184T3 (es) | 2013-05-16 |
| EA200601837A1 (ru) | 2007-04-27 |
| ZA200606547B (en) | 2008-04-30 |
| NO20065061L (no) | 2006-11-07 |
| PL1765355T3 (pl) | 2013-08-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 11A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2385 DE 20-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |