BRPI0510126A - derivados de piperidina como moduladores do receptor de quimiocina ccr5 - Google Patents

derivados de piperidina como moduladores do receptor de quimiocina ccr5

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Publication number
BRPI0510126A
BRPI0510126A BRPI0510126-3A BRPI0510126A BRPI0510126A BR PI0510126 A BRPI0510126 A BR PI0510126A BR PI0510126 A BRPI0510126 A BR PI0510126A BR PI0510126 A BRPI0510126 A BR PI0510126A
Authority
BR
Brazil
Prior art keywords
receptor modulators
piperidine derivatives
chemokine receptor
ccr5 chemokine
ccr5
Prior art date
Application number
BRPI0510126-3A
Other languages
English (en)
Inventor
Faull Alan
Tucker Howard
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35197429&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0510126(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from SE0401057A external-priority patent/SE0401057D0/xx
Priority claimed from SE0500057A external-priority patent/SE0500057D0/sv
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0510126A publication Critical patent/BRPI0510126A/pt

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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Abstract

DERIVADOS DE PIPERIDINA COMO MODULADORES DO RECEPTOR DE QUIMIOCINA CCR5 A presente invenção refere-se a compostos de fórmula (I): a composições os compreendendo, a processos para a sua preparação e ao seu uso em terapia médica (por exemplo, na modulação da atividade do receptor CCR5 em um animal de sangue quente).
BRPI0510126-3A 2004-04-23 2005-04-20 derivados de piperidina como moduladores do receptor de quimiocina ccr5 BRPI0510126A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0401057A SE0401057D0 (sv) 2004-04-23 2004-04-23 Chemical Compounds
SE0500057A SE0500057D0 (sv) 2005-01-10 2005-01-10 Chemical compounds
PCT/SE2005/000574 WO2005101989A2 (en) 2004-04-23 2005-04-20 Piperidine derivatives as modulators of chemokine receptor ccr5

Publications (1)

Publication Number Publication Date
BRPI0510126A true BRPI0510126A (pt) 2007-06-26

Family

ID=35197429

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0510126-3A BRPI0510126A (pt) 2004-04-23 2005-04-20 derivados de piperidina como moduladores do receptor de quimiocina ccr5

Country Status (16)

Country Link
US (2) US7615555B2 (pt)
EP (1) EP1742934A2 (pt)
JP (1) JP2007533735A (pt)
KR (1) KR20070007345A (pt)
AR (1) AR048834A1 (pt)
AU (1) AU2005235169B2 (pt)
BR (1) BRPI0510126A (pt)
CA (1) CA2562417A1 (pt)
IL (1) IL178650A0 (pt)
MX (1) MXPA06012045A (pt)
NO (1) NO20065319L (pt)
RU (1) RU2368608C2 (pt)
SA (1) SA05260099B1 (pt)
TW (1) TW200610761A (pt)
UY (1) UY28870A1 (pt)
WO (1) WO2005101989A2 (pt)

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CA2721099C (en) 2008-04-11 2017-04-25 Janssen Pharmaceutica Nv Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene a4 hydrolase
US8217060B2 (en) 2009-05-15 2012-07-10 Janssen Pharmaceutica, Nv Benzimidazole derivatives useful as TRP M8 receptor modulators
EP2456309B1 (en) 2009-07-24 2015-12-23 GlaxoSmithKline LLC Azabicyclo[3.2.1]octyl derivatives for use in the treatment of HIV.
CN102241664B (zh) * 2010-05-13 2014-11-12 上海医药工业研究院 芳烷二胺类衍生物及其作为抗抑郁症药物的应用
SG185615A1 (en) 2010-05-17 2012-12-28 Array Biopharma Inc Piperidinyl-substituted lactams as gpr119 modulators
US20140309226A1 (en) * 2011-11-16 2014-10-16 Array Biopharma Inc. Piperidinyl-substituted cyclic ureas as gpr119 modulators
JP6303250B2 (ja) 2012-12-21 2018-04-04 石原産業株式会社 有害生物防除剤
WO2014102594A2 (en) 2012-12-27 2014-07-03 Purdue Pharma L.P. Substituted benzimidazole-type piperidine compounds and uses thereof
US10556899B2 (en) * 2018-02-09 2020-02-11 Sci Pharmtech, Inc. Method for preparing Maraviroc
WO2025064788A2 (en) * 2023-09-20 2025-03-27 Cidara Therapeutics, Inc. Ccr5 conjugates and uses thereof

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