BRPI0511296A - sensibilização à outra terapia anticáncer e/ou melhora de um efeito colateral de outra terapia anticáncer por tratamento com um composto anticáncer ativado por gst - Google Patents
sensibilização à outra terapia anticáncer e/ou melhora de um efeito colateral de outra terapia anticáncer por tratamento com um composto anticáncer ativado por gstInfo
- Publication number
- BRPI0511296A BRPI0511296A BRPI0511296-6A BRPI0511296A BRPI0511296A BR PI0511296 A BRPI0511296 A BR PI0511296A BR PI0511296 A BRPI0511296 A BR PI0511296A BR PI0511296 A BRPI0511296 A BR PI0511296A
- Authority
- BR
- Brazil
- Prior art keywords
- anticancer
- gst
- therapy
- compound
- activated
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 9
- 238000011319 anticancer therapy Methods 0.000 title abstract 8
- 230000001093 anti-cancer Effects 0.000 title abstract 7
- 230000000694 effects Effects 0.000 title abstract 4
- 238000011282 treatment Methods 0.000 title abstract 3
- 206010070834 Sensitisation Diseases 0.000 title 1
- 230000008313 sensitization Effects 0.000 title 1
- 241000124008 Mammalia Species 0.000 abstract 4
- 230000001235 sensitizing effect Effects 0.000 abstract 3
- 238000000034 method Methods 0.000 abstract 2
- QCQCHGYLTSGIGX-GHXANHINSA-N 4-[[(3ar,5ar,5br,7ar,9s,11ar,11br,13as)-5a,5b,8,8,11a-pentamethyl-3a-[(5-methylpyridine-3-carbonyl)amino]-2-oxo-1-propan-2-yl-4,5,6,7,7a,9,10,11,11b,12,13,13a-dodecahydro-3h-cyclopenta[a]chrysen-9-yl]oxy]-2,2-dimethyl-4-oxobutanoic acid Chemical compound N([C@@]12CC[C@@]3(C)[C@]4(C)CC[C@H]5C(C)(C)[C@@H](OC(=O)CC(C)(C)C(O)=O)CC[C@]5(C)[C@H]4CC[C@@H]3C1=C(C(C2)=O)C(C)C)C(=O)C1=CN=CC(C)=C1 QCQCHGYLTSGIGX-GHXANHINSA-N 0.000 abstract 1
- 238000001815 biotherapy Methods 0.000 abstract 1
- 238000002512 chemotherapy Methods 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 230000002708 enhancing effect Effects 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 238000009126 molecular therapy Methods 0.000 abstract 1
- 238000001959 radiotherapy Methods 0.000 abstract 1
- 238000009097 single-agent therapy Methods 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/06—Tripeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/28—Compounds containing heavy metals
- A61K31/282—Platinum compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/475—Quinolines; Isoquinolines having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Immunology (AREA)
- Gastroenterology & Hepatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
SENSIBILIZAçãO à OUTRA TERAPIA ANTICáNCER E/OU MELHORA DE UM EFEITO COLATERAL DE OUTRA TERAPIA ANTICáNCER POR TRATAMENTO COM UM COMPOSTO ANTICáNCER ATIVADO POR GST. A presente invenção refere-se ao uso de um composto anticâncer ativado por GST na fabricação de um medicamento para sensibilizar um mamífero, especialmente um ser humano, para outra terapia anticâncer (isto é, uma terapia anticâncer que não é tratamento com um composto anticâncer ativado por GST - incluindo quimioterapia, terapia alvejada molecular, terapia biológica, radioterapia, cada empregado como monoterapia ou duas ou mais usadas em combinação), ou para melhorar um efeito colateral de outra terapia anticâncer em um mamífero, especialmente um ser humano. Composições contendo um composto anticâncer ativado por GST para estes usos. Um método de sensibilizar um mamífero, especialmente um ser humano, para outra terapia anticâncer, administrando-se uma quantidade eficaz sensibilizadora de um composto anticâncer ativado por GST. Um método de melhorar um efeito colateral de outra terapia anticâncer em um mamífero, especialmente um ser humano, administrando-se uma quantidade eficaz melhoradora de um composto anticâncer ativado por GST. O composto anticâncer ativado por GST é preferivelmente um composto da Patente dos Estados Unidos n<0> 5.556.942, e mais preferivelmente canfosfamida, especialmente como o sal de cloridrato.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US57279004P | 2004-05-20 | 2004-05-20 | |
| PCT/US2005/017960 WO2005112973A1 (en) | 2004-05-20 | 2005-05-19 | Sensitization to another anticancer therapy and/or amelioration of a side effect of another anticancer therapy by treatment with a gst-activated anticancer compound |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0511296A true BRPI0511296A (pt) | 2007-12-04 |
Family
ID=34970551
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0511296-6A BRPI0511296A (pt) | 2004-05-20 | 2005-05-19 | sensibilização à outra terapia anticáncer e/ou melhora de um efeito colateral de outra terapia anticáncer por tratamento com um composto anticáncer ativado por gst |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US20050261202A1 (pt) |
| EP (1) | EP1755632A1 (pt) |
| JP (1) | JP2007538105A (pt) |
| KR (1) | KR101174685B1 (pt) |
| CN (1) | CN1953762B (pt) |
| AR (1) | AR048971A1 (pt) |
| AU (1) | AU2005245004B2 (pt) |
| BR (1) | BRPI0511296A (pt) |
| CA (1) | CA2566850A1 (pt) |
| MX (1) | MXPA06013375A (pt) |
| TW (1) | TW200538149A (pt) |
| WO (1) | WO2005112973A1 (pt) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0011903D0 (en) * | 2000-05-18 | 2000-07-05 | Astrazeneca Ab | Combination chemotherapy |
| TWI323662B (en) * | 2002-11-15 | 2010-04-21 | Telik Inc | Combination cancer therapy with a gst-activated anticancer compound and another anticancer therapy |
| TW200538149A (en) | 2004-05-20 | 2005-12-01 | Telik Inc | Sensitization to another anticancer therapy and/or amelioration of a side effect of another anticancer therapy by treatment with a GST-activated anticancer compound |
| CU23511B6 (es) * | 2006-02-28 | 2010-04-13 | Biorec B V | Combinación farmacéutica para el tratamiento y/o quimiosensibilización de tumores refractarios a drogas anticancerígenas |
| ES2293834B1 (es) | 2006-07-20 | 2009-02-16 | Consejo Superior Investig. Cientificas | Compuesto con actividad inhibidora de las interacciones ubc13-uev, composiciones farmaceuticas que lo comprenden y sus aplicaciones terapeuticas. |
| US8173686B2 (en) | 2006-11-06 | 2012-05-08 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8178564B2 (en) * | 2006-11-06 | 2012-05-15 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8168661B2 (en) | 2006-11-06 | 2012-05-01 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8168662B1 (en) | 2006-11-06 | 2012-05-01 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| JP5424887B2 (ja) * | 2006-11-08 | 2014-02-26 | チョンシー ユー | ペプチド及び関連化合物の経皮送達システム |
| US20110033528A1 (en) * | 2009-08-05 | 2011-02-10 | Poniard Pharmaceuticals, Inc. | Stabilized picoplatin oral dosage form |
| JP5337143B2 (ja) * | 2007-04-14 | 2013-11-06 | サザン リサーチ インスティテュート | 化学療法剤と放射線とを併用した新形成の治療方法 |
| TW200916094A (en) * | 2007-06-27 | 2009-04-16 | Poniard Pharmaceuticals Inc | Stabilized picoplatin dosage form |
| US20100260832A1 (en) * | 2007-06-27 | 2010-10-14 | Poniard Pharmaceuticals, Inc. | Combination therapy for ovarian cancer |
| TW200920347A (en) * | 2007-07-16 | 2009-05-16 | Poniard Pharmaceuticals Inc | Oral formulations for picoplatin |
| US8252773B2 (en) * | 2007-11-02 | 2012-08-28 | Ziopharm Oncology, Inc. | Combination therapy with organic arsenicals |
| ES2332167B1 (es) | 2007-12-04 | 2010-10-25 | Universidad Autonoma De Madrid | Empleo de trefoil factor-family 3 (tff3) en el pronostico de sujetos diagnosticados con cancer colorectal. |
| ES2332557B1 (es) | 2007-12-04 | 2011-02-02 | Universidad Autonoma De Madrid | Huella genomica para el pronostico de la evolucion de adenocarcinoma colorectal. |
| US20110053879A1 (en) * | 2008-02-08 | 2011-03-03 | Poniard Pharmaceuticals, Inc. | Picoplatin and amrubicin to treat lung cancer |
| EP2252246B1 (en) * | 2008-03-14 | 2014-06-18 | Bionumerik Pharmaceuticals, Inc. | Chemoprotective methods and compositions |
| ES2338843B1 (es) | 2008-07-02 | 2011-01-24 | Centro De Investigaciones Energeticas, Medioambientales Y Tecnologicas | Huella genomica de cancer de mama. |
| EP2169078A1 (en) | 2008-09-26 | 2010-03-31 | Fundacion Gaiker | Methods and kits for the diagnosis and the staging of colorectal cancer |
| RU2627065C2 (ru) | 2009-05-08 | 2017-08-03 | Текфилдз Байокем Ко., Лтд. | Пролекарственные композиции с высокой степенью проникновения на основе пептидов и родственных пептидам соединений |
| ES2661216T3 (es) * | 2009-06-05 | 2018-03-28 | Cavion, Inc. | Método combinado para tratar el cáncer o un estado precanceroso |
| SG183114A1 (en) | 2010-03-01 | 2012-09-27 | Tau Therapeutics Llc | Cancer diagnosis and imaging |
| US20120251496A1 (en) * | 2011-03-31 | 2012-10-04 | Telik, Inc. | Ezatiostat for treating multiple myeloma |
| US20120288554A1 (en) * | 2011-05-12 | 2012-11-15 | Telik, Inc. | Canfosfamide monotherapy for treating multiple myeloma |
| WO2013092960A1 (en) | 2011-12-22 | 2013-06-27 | Fundacion Gaiker | Methods and kits for the diagnosis of colorectal cancer |
| SG10201610869TA (en) | 2012-06-26 | 2017-02-27 | Del Mar Pharmaceuticals | Methods for treating tyrosine-kinase-inhibitor-resistant malignancies in patients with genetic polymorphisms or ahi1 dysregulations or mutations employing dianhydrogalactitol, diacetyldianhydrogalacti |
| JP6340162B2 (ja) | 2012-12-20 | 2018-06-06 | 日東電工株式会社 | アポトーシス誘導剤 |
| KR20160061911A (ko) | 2013-04-08 | 2016-06-01 | 데니스 엠. 브라운 | 최적하 투여된 화학 화합물의 치료 효과 |
| CN106573062B (zh) | 2014-06-17 | 2020-08-25 | 日东电工株式会社 | 细胞凋亡诱导剂 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5556942A (en) * | 1991-04-29 | 1996-09-17 | Terrapin Technologies, Inc. | Glutathione S-transferase-activated compounds |
| US5767147A (en) * | 1995-04-21 | 1998-06-16 | The Regents Of The University Of California | Inhibition of glutathione transferase by haloenol lactones |
| EP0831877B1 (en) | 1995-06-07 | 2004-10-27 | Telik, Inc. | Metabolic effects of certain glutathione analogs |
| US5880097A (en) * | 1996-01-04 | 1999-03-09 | Terrapin Techologies, Inc. | Tethered prodrugs |
| US6281223B1 (en) * | 1999-04-13 | 2001-08-28 | Supergen, Inc. | Radioenhanced camptothecin derivative cancer treatments |
| TWI323662B (en) * | 2002-11-15 | 2010-04-21 | Telik Inc | Combination cancer therapy with a gst-activated anticancer compound and another anticancer therapy |
| TW200538149A (en) | 2004-05-20 | 2005-12-01 | Telik Inc | Sensitization to another anticancer therapy and/or amelioration of a side effect of another anticancer therapy by treatment with a GST-activated anticancer compound |
-
2005
- 2005-05-10 TW TW094115086A patent/TW200538149A/zh unknown
- 2005-05-19 CN CN2005800158989A patent/CN1953762B/zh not_active Expired - Fee Related
- 2005-05-19 AR ARP050102064A patent/AR048971A1/es not_active Application Discontinuation
- 2005-05-19 JP JP2007527521A patent/JP2007538105A/ja active Pending
- 2005-05-19 WO PCT/US2005/017960 patent/WO2005112973A1/en not_active Ceased
- 2005-05-19 CA CA002566850A patent/CA2566850A1/en not_active Abandoned
- 2005-05-19 BR BRPI0511296-6A patent/BRPI0511296A/pt not_active IP Right Cessation
- 2005-05-19 EP EP05752058A patent/EP1755632A1/en not_active Withdrawn
- 2005-05-19 AU AU2005245004A patent/AU2005245004B2/en not_active Ceased
- 2005-05-19 MX MXPA06013375A patent/MXPA06013375A/es active IP Right Grant
- 2005-05-19 US US11/133,833 patent/US20050261202A1/en not_active Abandoned
-
2006
- 2006-12-08 KR KR1020067025870A patent/KR101174685B1/ko not_active Expired - Fee Related
-
2007
- 2007-10-15 US US11/872,662 patent/US8207121B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20050261202A1 (en) | 2005-11-24 |
| KR20070012542A (ko) | 2007-01-25 |
| KR101174685B1 (ko) | 2012-08-16 |
| US20080166428A1 (en) | 2008-07-10 |
| TW200538149A (en) | 2005-12-01 |
| EP1755632A1 (en) | 2007-02-28 |
| CA2566850A1 (en) | 2005-12-01 |
| CN1953762A (zh) | 2007-04-25 |
| WO2005112973A1 (en) | 2005-12-01 |
| MXPA06013375A (es) | 2007-03-01 |
| JP2007538105A (ja) | 2007-12-27 |
| AU2005245004B2 (en) | 2011-08-04 |
| AR048971A1 (es) | 2006-06-14 |
| CN1953762B (zh) | 2012-04-25 |
| US8207121B2 (en) | 2012-06-26 |
| AU2005245004A1 (en) | 2005-12-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 9A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2260 DE 29/04/2014. |