BRPI0511532A - composto, uso do mesmo, composição farmacêutica, e, métodos para a terapia de distúrbios gastrointestinais funcionais e de sìndrome do intestino irritável em um animal de sangue quente, e para a preparação de um composto - Google Patents

composto, uso do mesmo, composição farmacêutica, e, métodos para a terapia de distúrbios gastrointestinais funcionais e de sìndrome do intestino irritável em um animal de sangue quente, e para a preparação de um composto

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Publication number
BRPI0511532A
BRPI0511532A BRPI0511532-9A BRPI0511532A BRPI0511532A BR PI0511532 A BRPI0511532 A BR PI0511532A BR PI0511532 A BRPI0511532 A BR PI0511532A BR PI0511532 A BRPI0511532 A BR PI0511532A
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BR
Brazil
Prior art keywords
compound
therapy
preparation
methods
pharmaceutical composition
Prior art date
Application number
BRPI0511532-9A
Other languages
English (en)
Inventor
Shujuan Jin
Ziping Liu
Claire Milburn
Miroslaw Tomaszewski
Christopher Walpole
Zhong-Yong Wei
Hua Yang
Original Assignee
Astrazeneca Ab
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32589801&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0511532(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0511532A publication Critical patent/BRPI0511532A/pt

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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/28—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton
    • C07C237/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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    • A61P25/22—Anxiolytics
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • C07C237/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having carbon atoms of carboxamide groups, amino groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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  • Organic Chemistry (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • General Health & Medical Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
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  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

COMPOSTO, USO DO MESMO, COMPOSIçãO FARMACEUTICA, E, MéTODOS PARA A TERAPIA DE DISTURBIOS GASTROENTESTINAIS FUNCIONAIS DE SINDROME DO INTESTINO IRRITáVEL EM UM ANIMAL DE SANGUE QUENTE, E PARA A PREPARAçãO DE UM COMPOSTO. Compostos da formula I ou sais farmaceuticamente aceitáveis dos mesmos: (I) em que R¬ 1¬, R¬ 2¬, R¬ 3¬, R¬ 4¬, m e n são como definidos no relatório, assim como sais e composições farmaceuticas que incluem os compostos, são preparados. Eles são uteis em terapia, em particular para o controle da dor.
BRPI0511532-9A 2004-05-25 2005-05-20 composto, uso do mesmo, composição farmacêutica, e, métodos para a terapia de distúrbios gastrointestinais funcionais e de sìndrome do intestino irritável em um animal de sangue quente, e para a preparação de um composto BRPI0511532A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0401342A SE0401342D0 (sv) 2004-05-25 2004-05-25 Therapeutic compounds
PCT/SE2005/000754 WO2005115972A1 (en) 2004-05-25 2005-05-20 Therapeutic compounds

Publications (1)

Publication Number Publication Date
BRPI0511532A true BRPI0511532A (pt) 2008-01-02

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BRPI0511532-9A BRPI0511532A (pt) 2004-05-25 2005-05-20 composto, uso do mesmo, composição farmacêutica, e, métodos para a terapia de distúrbios gastrointestinais funcionais e de sìndrome do intestino irritável em um animal de sangue quente, e para a preparação de um composto

Country Status (16)

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US (1) US20090018116A1 (pt)
EP (1) EP1756044A1 (pt)
JP (1) JP2008500337A (pt)
CN (1) CN1989100A (pt)
AR (1) AR049898A1 (pt)
AU (1) AU2005247835A1 (pt)
BR (1) BRPI0511532A (pt)
CA (1) CA2565066A1 (pt)
IL (1) IL179145A0 (pt)
MX (1) MXPA06013536A (pt)
NO (1) NO20065904L (pt)
SE (1) SE0401342D0 (pt)
TW (1) TW200539856A (pt)
UY (1) UY28922A1 (pt)
WO (1) WO2005115972A1 (pt)
ZA (1) ZA200609542B (pt)

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Publication number Priority date Publication date Assignee Title
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