BRPI0517302A - processo de preparação de compostos de pirimidina - Google Patents
processo de preparação de compostos de pirimidinaInfo
- Publication number
- BRPI0517302A BRPI0517302A BRPI0517302-7A BRPI0517302A BRPI0517302A BR PI0517302 A BRPI0517302 A BR PI0517302A BR PI0517302 A BRPI0517302 A BR PI0517302A BR PI0517302 A BRPI0517302 A BR PI0517302A
- Authority
- BR
- Brazil
- Prior art keywords
- formula
- compound shown
- alkynyloxypyrimidine
- pyrimidine compounds
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/34—One oxygen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
PROCESSO DE PREPARAçãO DE COMPOSTOS DE PIRIMIDINA. Compostos de 4-amino-6-alquinilóxipirimid ina mostrados pela fórmula (V) que têm uma atividade de controle contra pestes podem ser preparados pelo processo que compreende a primeira etapa que produz um composto de 4-flúor-6-alquinilóxipirimidina mostrado pela fórmula (I) fazendo um composto de 4,6-diflúorpirimidina mostrado pela fórmula (II) reagir com um composto de álcool mostrado pela fórmula (III) H-0R2(III) na presença de uma amina terciária; e a segunda etapa que produz o composto de 4-amino-6-alquinilóxipirimid ina mostrado pela fórmula (V) fazendo o composto de 4-flúor-6-alquinilóxipirimidina mostrado pela fórmula (I) reagir com o composto de amina mostrado pela fórmula (IV).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2004328689 | 2004-11-12 | ||
| PCT/JP2005/020678 WO2006051891A1 (en) | 2004-11-12 | 2005-11-04 | Production method of pyrimidine compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0517302A true BRPI0517302A (pt) | 2008-10-07 |
Family
ID=36336565
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0517302-7A BRPI0517302A (pt) | 2004-11-12 | 2005-11-04 | processo de preparação de compostos de pirimidina |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US8101753B2 (pt) |
| EP (1) | EP1809610B1 (pt) |
| KR (1) | KR101195800B1 (pt) |
| CN (1) | CN101056864B (pt) |
| AR (1) | AR053097A1 (pt) |
| AT (1) | ATE521596T1 (pt) |
| BR (1) | BRPI0517302A (pt) |
| IL (1) | IL182544A (pt) |
| TW (1) | TWI367208B (pt) |
| WO (1) | WO2006051891A1 (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5061565B2 (ja) * | 2006-04-24 | 2012-10-31 | 住友化学株式会社 | ピリミジン化合物の新規製造方法 |
| JP2008280342A (ja) * | 2007-04-13 | 2008-11-20 | Sumitomo Chemical Co Ltd | 有害生物防除組成物 |
| JP2010090090A (ja) * | 2008-10-10 | 2010-04-22 | Sumitomo Chemical Co Ltd | 有害生物防除組成物及び有害生物の防除方法 |
| JP2010090089A (ja) * | 2008-10-10 | 2010-04-22 | Sumitomo Chemical Co Ltd | 有害生物防除組成物及び有害生物の防除方法 |
| CN102718701B (zh) | 2011-03-30 | 2014-05-07 | 中国中化股份有限公司 | 芳氧基二卤丙烯醚类化合物与应用 |
| CN103766334B (zh) * | 2013-12-24 | 2016-01-27 | 江苏天容集团股份有限公司 | 抗氧化剂在防治酰胺类除草剂变色方面的应用 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2937171A (en) * | 1958-06-13 | 1960-05-17 | Du Pont | Process for obtaining fluorinated organic compounds |
| IT1212140B (it) | 1987-05-08 | 1989-11-08 | Sig Gla Pharmaceuticals S P A | Processo per la preparazione del 2,4-diammino-6-(1-piperidinil)-piri mi-din-n-ossido. |
| DE4137291A1 (de) * | 1991-11-13 | 1993-05-19 | Bayer Ag | Verfahren zur kontinuierlichen umsetzung von halogenpyrimidinen mit aminen |
| BR0113970A (pt) * | 2000-09-19 | 2003-07-01 | Sumitomo Chemical Co | Compostos de pirimidina e seu uso |
| JP2003034682A (ja) * | 2000-09-19 | 2003-02-07 | Sumitomo Chem Co Ltd | ピリミジン化合物及びその用途 |
| EP1193031A1 (en) | 2000-09-29 | 2002-04-03 | Infineon Technologies SC300 GmbH & Co. KG | Arrangement for polishing disk-like objects |
| JP4186484B2 (ja) * | 2002-03-12 | 2008-11-26 | 住友化学株式会社 | ピリミジン化合物およびその用途 |
| TWI312272B (en) | 2003-05-12 | 2009-07-21 | Sumitomo Chemical Co | Pyrimidine compound and pests controlling composition containing the same |
-
2005
- 2005-09-15 TW TW094131894A patent/TWI367208B/zh not_active IP Right Cessation
- 2005-10-14 AR ARP050104316A patent/AR053097A1/es not_active Application Discontinuation
- 2005-11-04 CN CN2005800387808A patent/CN101056864B/zh not_active Expired - Fee Related
- 2005-11-04 US US11/577,377 patent/US8101753B2/en not_active Expired - Fee Related
- 2005-11-04 WO PCT/JP2005/020678 patent/WO2006051891A1/en not_active Ceased
- 2005-11-04 EP EP05803375A patent/EP1809610B1/en not_active Expired - Lifetime
- 2005-11-04 KR KR1020077009998A patent/KR101195800B1/ko not_active Expired - Fee Related
- 2005-11-04 AT AT05803375T patent/ATE521596T1/de not_active IP Right Cessation
- 2005-11-04 BR BRPI0517302-7A patent/BRPI0517302A/pt not_active IP Right Cessation
-
2007
- 2007-04-12 IL IL182544A patent/IL182544A/en not_active IP Right Cessation
-
2011
- 2011-12-15 US US13/327,387 patent/US20120088914A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP1809610A4 (en) | 2009-11-18 |
| WO2006051891A1 (en) | 2006-05-18 |
| US20080039445A1 (en) | 2008-02-14 |
| CN101056864A (zh) | 2007-10-17 |
| TWI367208B (en) | 2012-07-01 |
| ATE521596T1 (de) | 2011-09-15 |
| CN101056864B (zh) | 2010-12-22 |
| EP1809610B1 (en) | 2011-08-24 |
| IL182544A (en) | 2011-04-28 |
| TW200621726A (en) | 2006-07-01 |
| EP1809610A1 (en) | 2007-07-25 |
| US8101753B2 (en) | 2012-01-24 |
| US20120088914A1 (en) | 2012-04-12 |
| IL182544A0 (en) | 2007-09-20 |
| AR053097A1 (es) | 2007-04-25 |
| KR20070083909A (ko) | 2007-08-24 |
| KR101195800B1 (ko) | 2012-11-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B06H | Technical and formal requirements: requirement cancelled [chapter 6.8 patent gazette] |
Free format text: REF. A RPI NO 2154 DE 17/04/2012. ANULACAO DA EXIGENCIA 6.6 POR TER SIDO INDEVIDA. REQUERENTE NAO APRESENTOU RESPOSTA A EXIGENCIA CONFORME DISPOE A RESOLUCAO 207 DE 24/04/2009, ENTRETANTO, A RESPOSTA CONSTA NO FORMULARIO DE DEPOSITO. |
|
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 9A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2279 DE 09/09/2014. |
|
| B11D | Dismissal acc. art. 38, par 2 of ipl - failure to pay fee after grant in time | ||
| B11N | Dismissal: publication cancelled [chapter 11.14 patent gazette] |
Free format text: PUBLICACAO ANULADA REFERENTE RPI/2328 DE 18/08/2015, POR TER SIDO INDEVIDA. |