BRPI0605901A - formas polimórficas de maleato de tegaserode - Google Patents

formas polimórficas de maleato de tegaserode

Info

Publication number
BRPI0605901A
BRPI0605901A BRPI0605901-5A BRPI0605901A BRPI0605901A BR PI0605901 A BRPI0605901 A BR PI0605901A BR PI0605901 A BRPI0605901 A BR PI0605901A BR PI0605901 A BRPI0605901 A BR PI0605901A
Authority
BR
Brazil
Prior art keywords
tegaserode
maleate
polymorphic forms
polymorphic
processes
Prior art date
Application number
BRPI0605901-5A
Other languages
English (en)
Inventor
Santiago Ini
Tamas Koltai
Michael Pinchasov
Sofia Gorohovsky
Gustavo Frenkel
Original Assignee
Teva Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharma filed Critical Teva Pharma
Publication of BRPI0605901A publication Critical patent/BRPI0605901A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

FORMAS POLIMóRFICAS DE MALEATO DE TEGASERODE. São fornecidas formas cristalinas de maleato de tegaserode e processos para sua preparação.
BRPI0605901-5A 2005-06-22 2006-06-22 formas polimórficas de maleato de tegaserode BRPI0605901A (pt)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US69330105P 2005-06-22 2005-06-22
US70404805P 2005-07-28 2005-07-28
US72172905P 2005-09-28 2005-09-28
US72925805P 2005-10-20 2005-10-20
US77306606P 2006-02-13 2006-02-13
US79281106P 2006-04-17 2006-04-17
PCT/US2006/024348 WO2007002314A2 (en) 2005-06-22 2006-06-22 Polymorphic forms of tegaserod maleate

Publications (1)

Publication Number Publication Date
BRPI0605901A true BRPI0605901A (pt) 2007-12-18

Family

ID=37192322

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0605901-5A BRPI0605901A (pt) 2005-06-22 2006-06-22 formas polimórficas de maleato de tegaserode

Country Status (7)

Country Link
US (1) US20070112057A1 (pt)
EP (1) EP1893195A2 (pt)
JP (2) JP2008514734A (pt)
KR (1) KR20070062504A (pt)
BR (1) BRPI0605901A (pt)
MX (1) MX2007002113A (pt)
WO (1) WO2007002314A2 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20050253A1 (es) * 2003-07-24 2005-06-03 Novartis Ag Modificaciones estables de maleato de hidrogeno de tegaserod
US20070225507A1 (en) * 2006-01-18 2007-09-27 Gustavo Frenkel Process for preparing a crystalline form of Tegaserod maleate
EP1956002A1 (en) * 2007-02-07 2008-08-13 Chemo Ibérica, S.A. New tegaserod maleate polymorphs and process for their preparation
EP2146958A1 (en) * 2007-05-17 2010-01-27 Generics Ýuk¨Limited Process for the preparation of form a of tegaserod
TWI665190B (zh) 2013-11-15 2019-07-11 阿克比治療有限公司 ｛［５－（３－氯苯基）－３－羥基吡啶－２－羰基］胺基｝乙酸之固體型式，其組合物及用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR027261A1 (es) * 2000-02-02 2003-03-19 Upjohn Co Linezolid forma cristalina ii
JP4414237B2 (ja) * 2002-03-20 2010-02-10 テバ ファーマシューティカル インダストリーズ リミティド ケチアピンヘミフマレートの結晶形
JP4298212B2 (ja) * 2002-03-29 2009-07-15 大日本印刷株式会社 塩酸エピナスチン高融点型結晶の製造法
WO2004085393A1 (en) * 2003-03-25 2004-10-07 Hetero Drugs Limited Novel crystalline forms of tegaserod maleate
PE20050253A1 (es) * 2003-07-24 2005-06-03 Novartis Ag Modificaciones estables de maleato de hidrogeno de tegaserod

Also Published As

Publication number Publication date
MX2007002113A (es) 2007-04-27
KR20070062504A (ko) 2007-06-15
JP2007297377A (ja) 2007-11-15
WO2007002314A3 (en) 2007-06-28
EP1893195A2 (en) 2008-03-05
US20070112057A1 (en) 2007-05-17
WO2007002314A9 (en) 2007-08-23
WO2007002314A2 (en) 2007-01-04
JP2008514734A (ja) 2008-05-08

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]