BRPI0816909A2 - Processo para produção de intermediários de monobactama em ponte. - Google Patents

Processo para produção de intermediários de monobactama em ponte.

Info

Publication number
BRPI0816909A2
BRPI0816909A2 BRPI0816909A BRPI0816909A2 BR PI0816909 A2 BRPI0816909 A2 BR PI0816909A2 BR PI0816909 A BRPI0816909 A BR PI0816909A BR PI0816909 A2 BRPI0816909 A2 BR PI0816909A2
Authority
BR
Brazil
Prior art keywords
intermediates
production
bridged monobactam
monobactam
bridged
Prior art date
Application number
Other languages
English (en)
Inventor
Marc Muller
Xiaoping Wu
Lin Xu
Original Assignee
Basilea Pharmaceutica Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basilea Pharmaceutica Ag filed Critical Basilea Pharmaceutica Ag
Publication of BRPI0816909A2 publication Critical patent/BRPI0816909A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/40Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
    • C07C271/42Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/54Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/22Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BRPI0816909 2007-09-17 2008-09-15 Processo para produção de intermediários de monobactama em ponte. BRPI0816909A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07116603 2007-09-17
PCT/EP2008/062258 WO2009037229A1 (en) 2007-09-17 2008-09-15 Process for the manufacture of bridged monobactam intermediates

Publications (1)

Publication Number Publication Date
BRPI0816909A2 true BRPI0816909A2 (pt) 2015-03-17

Family

ID=39027525

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0816909 BRPI0816909A2 (pt) 2007-09-17 2008-09-15 Processo para produção de intermediários de monobactama em ponte.

Country Status (16)

Country Link
US (2) US8450477B2 (pt)
EP (1) EP2197881B1 (pt)
JP (1) JP5551072B2 (pt)
KR (1) KR101421774B1 (pt)
CN (1) CN101801974B (pt)
AU (1) AU2008300616B2 (pt)
BR (1) BRPI0816909A2 (pt)
CA (1) CA2698441C (pt)
CY (1) CY1114147T1 (pt)
DK (1) DK2197881T3 (pt)
ES (1) ES2419255T3 (pt)
MX (1) MX2010002642A (pt)
PL (1) PL2197881T3 (pt)
PT (1) PT2197881E (pt)
WO (1) WO2009037229A1 (pt)
ZA (1) ZA201001694B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014184503A1 (fr) 2013-05-16 2014-11-20 Universite De Strasbourg Composés dendritiques comprenant un agent chélatant, fluorochrome ou agent de reconnaissance, compositions les comprenant et leurs utilisations
CN103554112B (zh) * 2013-11-07 2016-04-13 中国科学院昆明植物研究所 顺式稠环的β-内酰胺化合物的合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA826089B (en) * 1981-08-27 1983-07-27 Hoffmann La Roche Beta-lactams
CA1262128A (en) 1981-08-27 1989-10-03 Christian N. Hubschwerlen .beta.-lactams
DK0508234T3 (da) * 1991-04-11 1996-10-28 Hoffmann La Roche Beta-lactamer
CA2143519A1 (en) * 1994-03-11 1995-09-12 F. Hoffmann-La Roche Ag Beta-lactams
TW358097B (en) * 1996-05-24 1999-05-11 Hoffmann La Roche Beta-lactams and their process and pharmaceutical compositions
CN103724330B (zh) 2005-12-07 2015-08-19 巴斯利尔药物股份公司 单环-内酰胺类抗生素与β-内酰胺酶抑制剂的有效的联合应用

Also Published As

Publication number Publication date
MX2010002642A (es) 2010-03-26
US8877961B2 (en) 2014-11-04
EP2197881B1 (en) 2013-04-17
CY1114147T1 (el) 2016-07-27
US20110178291A1 (en) 2011-07-21
DK2197881T3 (da) 2013-06-24
US20130274503A1 (en) 2013-10-17
ZA201001694B (en) 2010-10-27
CA2698441C (en) 2012-04-03
CN101801974A (zh) 2010-08-11
US8450477B2 (en) 2013-05-28
AU2008300616B2 (en) 2013-02-14
KR20100074157A (ko) 2010-07-01
EP2197881A1 (en) 2010-06-23
CA2698441A1 (en) 2009-03-26
HK1142900A1 (en) 2010-12-17
CN101801974B (zh) 2013-08-28
WO2009037229A1 (en) 2009-03-26
PL2197881T3 (pl) 2013-09-30
KR101421774B1 (ko) 2014-07-30
JP5551072B2 (ja) 2014-07-16
PT2197881E (pt) 2013-06-28
AU2008300616A1 (en) 2009-03-26
JP2010539211A (ja) 2010-12-16
ES2419255T3 (es) 2013-08-20

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2479 DE 10-07-2018 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.