BRPI0821752A8 - Processo para preparar derivados de ácido 22-fluoracil-3-amino-acrílico - Google Patents

Processo para preparar derivados de ácido 22-fluoracil-3-amino-acrílico

Info

Publication number
BRPI0821752A8
BRPI0821752A8 BRPI0821752A BRPI0821752A BRPI0821752A8 BR PI0821752 A8 BRPI0821752 A8 BR PI0821752A8 BR PI0821752 A BRPI0821752 A BR PI0821752A BR PI0821752 A BRPI0821752 A BR PI0821752A BR PI0821752 A8 BRPI0821752 A8 BR PI0821752A8
Authority
BR
Brazil
Prior art keywords
acid derivatives
amino
preparing
acrylic acid
fluoracyl
Prior art date
Application number
BRPI0821752A
Other languages
English (en)
Inventor
Lui Norbert
Wollner Thomas
Wieschemeyer Jürgen
Dockner Michael
Heinrich Jens-Dietmar
Original Assignee
Bayer Cropscience Ag
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag, Bayer Ip Gmbh filed Critical Bayer Cropscience Ag
Publication of BRPI0821752A2 publication Critical patent/BRPI0821752A2/pt
Publication of BRPI0821752A8 publication Critical patent/BRPI0821752A8/pt
Publication of BRPI0821752B1 publication Critical patent/BRPI0821752B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/16—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions not involving the amino or carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

PROCESSO PARA PREPARAR DERIVADOS DE ÁCIDO 2-FLUORACIL-3-AMINO-ACRÍLICO. A presente invenção refere-se a um processo para preparar derivados de ácido 2-fluoracil-3-amino-acrílico através da reação de ácidos carboxílicos fluorados com derivados de ácido dialquilaminoacrílico e halogenetos de ácidos.
BRPI0821752-1A 2007-12-21 2008-12-16 Process for preparing 22-fluoracyl-3-amino acrylic acid derivatives BRPI0821752B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07150357.7 2007-12-21
EP07150357A EP2072497A1 (de) 2007-12-21 2007-12-21 Verfahren zum Herstellen von 2-Fluoracyl-3-amino-acrylsäure-Derivaten
PCT/EP2008/010689 WO2009083134A1 (de) 2007-12-21 2008-12-16 Verfahren zum herstellen von 2-fluoracyl-3-amino-acrylsäure-derivaten

Publications (3)

Publication Number Publication Date
BRPI0821752A2 BRPI0821752A2 (pt) 2015-06-16
BRPI0821752A8 true BRPI0821752A8 (pt) 2015-12-22
BRPI0821752B1 BRPI0821752B1 (pt) 2017-10-24

Family

ID=39164649

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0821752-1A BRPI0821752B1 (pt) 2007-12-21 2008-12-16 Process for preparing 22-fluoracyl-3-amino acrylic acid derivatives

Country Status (11)

Country Link
US (1) US8288582B2 (pt)
EP (2) EP2072497A1 (pt)
KR (1) KR101574143B1 (pt)
CN (1) CN101903333B (pt)
BR (1) BRPI0821752B1 (pt)
DK (1) DK2245001T3 (pt)
ES (1) ES2405549T3 (pt)
IL (1) IL205745A (pt)
MX (1) MX2010005938A (pt)
TW (1) TWI441802B (pt)
WO (1) WO2009083134A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2042482A1 (de) * 2007-09-26 2009-04-01 Bayer CropScience AG Verfahren zur Herstellung von 2-Dihalogenacyl-3-amino-acrylsäure-Derivaten
EP2263999A4 (en) * 2008-03-18 2012-11-07 Mitsui Chemicals Agro Inc METHOD FOR PRODUCING A FLUOROUS ACYL ACIDIC ACID DERIVATIVE, METHOD FOR THE PRODUCTION OF A FLUOROUS PYRAZOL CARBOXYLIC ACID DERIVATIVE AND METHOD FOR PRODUCING A FLUOROUS PYRAZOL CARBOXYLENE DERIVATIVE
JP5602131B2 (ja) 2008-05-02 2014-10-08 ビーエーエスエフ ソシエタス・ヨーロピア ハロゲン置換２−（アミノメチリデン）−３−オキソ酪酸エステルの製造方法
BRPI0911898A2 (pt) 2008-05-02 2015-10-13 Basf Se processo para preparar compostos, e, composto.
US8598222B2 (en) 2008-05-05 2013-12-03 Basf Se Method for preparing 1,3,4-substituted pyrazol compounds
EP2307384B1 (en) 2008-07-21 2012-04-25 Basf Se Process for preparing 1,3-disubstituted pyrazolecarboxylic esters
MX2017017140A (es) * 2015-06-26 2018-03-09 Bayer Cropscience Ag Proceso para la preparacion de pirazoles sustituidos que contienen grupos haloalcoxi-y haloalquiltio a partir de a,a-dihaloalquilaminas y quetiminas.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE59005903D1 (de) * 1989-09-01 1994-07-07 Gretag Imaging Ag Photoelektrischer Abtaster.
DE4302156A1 (de) 1993-01-27 1994-07-28 Bayer Ag Verfahren zur Herstellung von Aminomethylenverbindungen
DE19822912A1 (de) * 1998-05-22 1999-11-25 Degussa Verfahren zur Herstellung von 3-Amino-2-oxo-pyrrolidinen, neue Zwischenprodukte und deren Verwendung
KR20000035081A (ko) * 1998-11-10 2000-06-26 마크 에스. 아들러 2-(트리할로아세틸)-3-(치환된 아미노)-2-프로페노에이트 제조방법
DE10161978A1 (de) 2001-12-17 2003-06-26 Bayer Ag Verfahren zur Herstellung von 2-Halogenacyl-3-amino-acrylsäure-derivate
DE10349500A1 (de) * 2003-10-23 2005-06-02 Bayer Cropscience Ag Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern
CN101405270B (zh) * 2006-03-22 2013-01-16 霍夫曼-拉罗奇有限公司 作为11-β-HSD-1的吡唑类

Also Published As

Publication number Publication date
BRPI0821752B1 (pt) 2017-10-24
TW200940483A (en) 2009-10-01
CN101903333B (zh) 2013-11-06
ES2405549T3 (es) 2013-05-31
DK2245001T3 (da) 2013-06-17
EP2245001B1 (de) 2013-03-20
KR20100099237A (ko) 2010-09-10
IL205745A0 (en) 2010-11-30
MX2010005938A (es) 2010-07-19
KR101574143B1 (ko) 2016-02-19
IL205745A (en) 2014-01-30
CN101903333A (zh) 2010-12-01
BRPI0821752A2 (pt) 2015-06-16
EP2245001A1 (de) 2010-11-03
EP2072497A1 (de) 2009-06-24
US8288582B2 (en) 2012-10-16
WO2009083134A1 (de) 2009-07-09
TWI441802B (zh) 2014-06-21
US20100274049A1 (en) 2010-10-28

Similar Documents

Publication Publication Date Title
BRPI0817747A8 (pt) Processo para a preparação de derivados de ácido 2-di-halogenoacil-3-amino-acrílico
BRPI0914917A2 (pt) processo para a produção de ácidos carboxílicos livres.
BRPI1011506B8 (pt) processo para a fabricação de moduladores de regulador de condutância de transmembrana de fibrose cística
BR112012000210A2 (pt) processo para a produção de heterodímeoros de ácido glutâmico.
BRPI0919826A2 (pt) Micro-organismo para a producao de acido succinico.
BRPI0823162A2 (pt) Processo destinado à produção de ácido forsfórico de alta pureza
BR112012028395A2 (pt) processo para preparar ditiina-tetracarboxi-diimidas
PT2639222T (pt) Processo de produção de ácidos cicloalquilcarboxamido-piridina-benzoicos
BR112013002925A2 (pt) processo para a síntese de ácido 2,5-furandicarboxílico
BRPI0921013A2 (pt) processo para a síntese de um ômega-aminoácido (éster).
BR112012011961A2 (pt) processo para produzir cloretos de ácido 5-flúor-1-alquil-3-fluoralquil-1h-pirazol-4-carboxílico
BRPI0822106A2 (pt) "processo para preparação de ácido metacrílico de alta pureza."
BR112012001105A2 (pt) produção de ácido acético por meio de carbonilação com uma reação e vaporização instantânea melhoradas
BR112012015490A2 (pt) adoçantes e processo para a sua produção
BRPI0905147A8 (pt) processo para síntese de ivabradina e seus sais de adição com um ácido farmaceuticamente aceitável
BRPI0909369A2 (pt) processo contínuo para preparação de amidas de ácidos carboxílicos alifáticos inferiores
BR112015031913A2 (pt) processo para a fabricação de amino-benzoxazinonas 4-propargilatadas e sua utilização
BRPI0909560A2 (pt) processo de preparação de derivaods de ácido 1-(2-halo-bifenil-4-il)-ciclopropano carboxílico
BR112012020824A2 (pt) processo para produção de corpos moldados revestidos.
BR112012002641A2 (pt) processo de preparação de amidas de ácido carboxílico pirazol
BRPI0907872A2 (pt) Processo para produção de ácido dicarboxílico
CR20110208A (es) Proceso para la preparación de benzonorbornenos
BR112012001274A2 (pt) processo para produção de ácidos decancarboxílicos
BRPI1009635A2 (pt) ''processo de produção de cristais de ácido adípico''
MX2010005938A (es) Procedimiento para la preparacion de derivados de acido 2-fluoroacil-3-amino-acrilico.

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 4A ANUIDADE. PAGAR RESTAURACAO.

B25A Requested transfer of rights approved

Owner name: BAYER INTELLECTUAL PROPERTY GMBH (DE)

B08H Application fees: decision cancelled [chapter 8.8 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2343 DE 01/12/2015.

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]
B25G Requested change of headquarter approved
B25A Requested transfer of rights approved