BRPI0823136A2 - Processo para a preparação de fenilalaninas substituídas - Google Patents

Processo para a preparação de fenilalaninas substituídas

Info

Publication number: BRPI0823136A2
Authority: BR; Brazil
Prior art keywords: preparation; substituted phenylalanines; phenylalanines; substituted
Prior art date: 2008-10-24

Application number

BRPI0823136-2A

Other languages

English (en)

Inventor

Hugh Alfred Burgoon

Ramanaiah C Kanamarlapudi

Iain Fraser Pickersgill

Zhi-Cai Shi

Wenxue Wu

Haiming Zhang

Matthew Mangzhu Zhao

Original Assignee

Lexicon Pharmaceuticals Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-10-24

Filing date

2008-10-24

Publication date

2015-06-16

2008-10-24 Application filed by Lexicon Pharmaceuticals Inc filed Critical Lexicon Pharmaceuticals Inc

2015-06-16 Publication of BRPI0823136A2 publication Critical patent/BRPI0823136A2/pt

Links

235000008729 phenylalanine Nutrition 0.000 title 1
150000002994 phenylalanines Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C43/00—Ethers; Compounds having groups, groups or groups
- C07C43/02—Ethers
- C07C43/20—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring
- C07C43/23—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring containing hydroxy or O-metal groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)

BRPI0823136-2A 2008-10-24 2008-10-24 Processo para a preparação de fenilalaninas substituídas BRPI0823136A2 (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/US2008/081054 WO2010047712A1 (en)	2008-10-24	2008-10-24	Process for the preparation of substituted phenylalanines

Publications (1)

Publication Number	Publication Date
BRPI0823136A2 true BRPI0823136A2 (pt)	2015-06-16

Family

ID=40785295

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0823136-2A BRPI0823136A2 (pt)	2008-10-24	2008-10-24	Processo para a preparação de fenilalaninas substituídas

Country Status (11)

Country	Link
EP (1)	EP2358685A1 (pt)
JP (1)	JP2012506427A (pt)
KR (1)	KR20110074875A (pt)
CN (1)	CN102203069A (pt)
AU (1)	AU2008363274A1 (pt)
BR (1)	BRPI0823136A2 (pt)
CA (1)	CA2741563A1 (pt)
IL (1)	IL211996A0 (pt)
MX (1)	MX2011004168A (pt)
RU (1)	RU2011120822A (pt)
WO (1)	WO2010047712A1 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2015089137A1 (en) *	2013-12-11	2015-06-18	Karos Pharmaceuticals, Inc.	Acylguanidines as tryptophan hydroxylase inhibitors
BR112020018094A2 (pt)	2018-03-08	2020-12-22	Incyte Corporation	Compostos de aminopirazina diol como inibidores de pi3k-¿
US11046658B2 (en)	2018-07-02	2021-06-29	Incyte Corporation	Aminopyrazine derivatives as PI3K-γ inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK1984344T3 (da) *	2005-12-29	2013-01-14	Lexicon Pharmaceuticals Inc	Multicykliske aminosyrederivater og fremgangsmåder til anvendelse heraf
UA99270C2 (en) *	2006-12-12	2012-08-10	Лексикон Фармасьютикалз, Инк.	4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds and methods of their use

2008
- 2008-10-24 RU RU2011120822/04A patent/RU2011120822A/ru unknown
- 2008-10-24 AU AU2008363274A patent/AU2008363274A1/en not_active Abandoned
- 2008-10-24 CA CA2741563A patent/CA2741563A1/en not_active Abandoned
- 2008-10-24 EP EP08876427A patent/EP2358685A1/en not_active Withdrawn
- 2008-10-24 WO PCT/US2008/081054 patent/WO2010047712A1/en not_active Ceased
- 2008-10-24 KR KR1020117009174A patent/KR20110074875A/ko not_active Withdrawn
- 2008-10-24 BR BRPI0823136-2A patent/BRPI0823136A2/pt not_active IP Right Cessation
- 2008-10-24 CN CN2008801316930A patent/CN102203069A/zh active Pending
- 2008-10-24 MX MX2011004168A patent/MX2011004168A/es not_active Application Discontinuation
- 2008-10-24 JP JP2011533149A patent/JP2012506427A/ja not_active Withdrawn
2011
- 2011-03-29 IL IL211996A patent/IL211996A0/en unknown

Also Published As

Publication number	Publication date
CN102203069A (zh)	2011-09-28
EP2358685A1 (en)	2011-08-24
RU2011120822A (ru)	2012-11-27
CA2741563A1 (en)	2010-04-29
KR20110074875A (ko)	2011-07-04
IL211996A0 (en)	2011-06-30
JP2012506427A (ja)	2012-03-15
WO2010047712A1 (en)	2010-04-29
AU2008363274A1 (en)	2010-04-29
MX2011004168A (es)	2011-05-23

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Legal Events

Date	Code	Title	Description
2015-12-01	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES.
2016-04-05	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2343 DE 01-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.