BRPI0906632A2 - Imidazolinil metil aril sulfonamidas - Google Patents

Imidazolinil metil aril sulfonamidas

Info

Publication number
BRPI0906632A2
BRPI0906632A2 BRPI0906632-2A BRPI0906632A BRPI0906632A2 BR PI0906632 A2 BRPI0906632 A2 BR PI0906632A2 BR PI0906632 A BRPI0906632 A BR PI0906632A BR PI0906632 A2 BRPI0906632 A2 BR PI0906632A2
Authority
BR
Brazil
Prior art keywords
methyl aryl
aryl sulfonamides
imidazolinyl
imidazolinyl methyl
methods
Prior art date
Application number
BRPI0906632-2A
Other languages
English (en)
Inventor
Robert Greenhouse
Counde O'yang
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BRPI0906632A2 publication Critical patent/BRPI0906632A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D233/24—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
BRPI0906632-2A 2008-02-04 2009-01-26 Imidazolinil metil aril sulfonamidas BRPI0906632A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2584108P 2008-02-04 2008-02-04
PCT/EP2009/050841 WO2009098136A1 (en) 2008-02-04 2009-01-26 Novel imidazolinylmethyl aryl sulfonamides

Publications (1)

Publication Number Publication Date
BRPI0906632A2 true BRPI0906632A2 (pt) 2015-07-14

Family

ID=40679581

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0906632-2A BRPI0906632A2 (pt) 2008-02-04 2009-01-26 Imidazolinil metil aril sulfonamidas

Country Status (12)

Country Link
US (2) US20090197934A1 (pt)
EP (1) EP2238116B1 (pt)
JP (1) JP2011511026A (pt)
KR (1) KR20100096262A (pt)
CN (1) CN101925581A (pt)
AT (1) ATE525360T1 (pt)
AU (1) AU2009211506A1 (pt)
BR (1) BRPI0906632A2 (pt)
CA (1) CA2711728A1 (pt)
IL (1) IL206611A0 (pt)
MX (1) MX2010007929A (pt)
WO (1) WO2009098136A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20220401415A1 (en) * 2019-10-25 2022-12-22 Curasen Therapeutics, Inc. Methods for treating neurological disorders with alpha1a-ar partial agonists
KR20230058066A (ko) * 2020-08-27 2023-05-02 큐라센 테라퓨틱스, 인코포레이티드 α1A-아드레날린성 수용체 작용제 및 사용 방법
CN112624975A (zh) * 2020-11-27 2021-04-09 华南农业大学 一种妥拉唑林半抗原、人工抗原、抗体及其制备和应用
CN117229291B (zh) * 2023-11-10 2024-03-15 山东大学 内体-溶酶体转运靶向嵌合体降解剂及其制备方法与应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG72827A1 (en) * 1997-06-23 2000-05-23 Hoffmann La Roche Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
EP1501817A1 (en) * 2002-04-23 2005-02-02 F. Hoffmann-La Roche Ag Imidazolinylmethyl aralkylsulfonamides
EP2238114A1 (en) * 2008-02-04 2010-10-13 F. Hoffmann-La Roche AG Novel imidazolinylmethyl aryl sulfonamides
MX2010007967A (es) * 2008-02-04 2010-08-09 Hoffmann La Roche N-[3-bromo-2-cloro-4-(4,5-dihidro-1h-imidazol-2-ilmetil)-fenil]-m etansulfoamida como agonista parcial alfa-1 a adrenergico para el tratamiento de la incontinencia.

Also Published As

Publication number Publication date
AU2009211506A1 (en) 2009-08-13
EP2238116A1 (en) 2010-10-13
EP2238116B1 (en) 2011-09-21
CN101925581A (zh) 2010-12-22
CA2711728A1 (en) 2009-07-13
IL206611A0 (en) 2010-12-30
KR20100096262A (ko) 2010-09-01
US20090197934A1 (en) 2009-08-06
ATE525360T1 (de) 2011-10-15
MX2010007929A (es) 2010-08-09
JP2011511026A (ja) 2011-04-07
US20110230535A1 (en) 2011-09-22
WO2009098136A1 (en) 2009-08-13

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.