BRPI0908951A2 - compostos de minociclina e método de uso dos mesmos - Google Patents

compostos de minociclina e método de uso dos mesmos

Info

Publication number
BRPI0908951A2
BRPI0908951A2 BRPI0908951A BRPI0908951A BRPI0908951A2 BR PI0908951 A2 BRPI0908951 A2 BR PI0908951A2 BR PI0908951 A BRPI0908951 A BR PI0908951A BR PI0908951 A BRPI0908951 A BR PI0908951A BR PI0908951 A2 BRPI0908951 A2 BR PI0908951A2
Authority
BR
Brazil
Prior art keywords
minocycline compounds
minocycline
compounds
avaible
abstract
Prior art date
Application number
BRPI0908951A
Other languages
English (en)
Inventor
Dennis P Molnar
Ken S Tanaka
Robert D Arbeit
Sean Johnston
Thomas J Bigger
Original Assignee
Paratek Pharm Innc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41056527&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0908951(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Paratek Pharm Innc filed Critical Paratek Pharm Innc
Publication of BRPI0908951A2 publication Critical patent/BRPI0908951A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/65Tetracyclines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

abstract not avaible
BRPI0908951A 2008-03-05 2009-03-05 compostos de minociclina e método de uso dos mesmos BRPI0908951A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6818008P 2008-03-05 2008-03-05
PCT/US2009/001451 WO2009111064A2 (en) 2008-03-05 2009-03-05 Minocycline compounds and methods of use thereof

Publications (1)

Publication Number Publication Date
BRPI0908951A2 true BRPI0908951A2 (pt) 2017-01-17

Family

ID=41056527

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0908951A BRPI0908951A2 (pt) 2008-03-05 2009-03-05 compostos de minociclina e método de uso dos mesmos

Country Status (12)

Country Link
US (9) US20090253660A1 (pt)
EP (1) EP2262754A4 (pt)
JP (1) JP2011513404A (pt)
KR (1) KR20100126469A (pt)
CN (1) CN102015602A (pt)
AU (1) AU2009220171A1 (pt)
BR (1) BRPI0908951A2 (pt)
CA (1) CA2717703A1 (pt)
CL (1) CL2010000188A1 (pt)
MX (1) MX2010009693A (pt)
RU (1) RU2010140682A (pt)
WO (1) WO2009111064A2 (pt)

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US8636982B2 (en) 2007-08-07 2014-01-28 Foamix Ltd. Wax foamable vehicle and pharmaceutical compositions thereof
WO2009090495A2 (en) 2007-12-07 2009-07-23 Foamix Ltd. Oil and liquid silicone foamable carriers and formulations
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PT2271348T (pt) * 2008-03-28 2018-04-16 Paratek Pharm Innc Formulação de comprimido oral de composto de tetraciclina
TW202332671A (zh) 2008-05-19 2023-08-16 美商Prtk Spv2公司 四環素化合物之甲苯磺酸鹽及同素異形體
WO2010125470A2 (en) 2009-04-28 2010-11-04 Foamix Ltd. Foamable vehicle and pharmaceutical compositions comprising aprotic polar solvents and uses thereof
CA2769677A1 (en) 2009-07-29 2011-02-03 Foamix Ltd. Non surface active agent non polymeric agent hydro-alcoholic foamable compositions, breakable foams and their uses
WO2011013009A2 (en) 2009-07-29 2011-02-03 Foamix Ltd. Non surfactant hydro-alcoholic foamable compositions, breakable foams and their uses
US9849142B2 (en) 2009-10-02 2017-12-26 Foamix Pharmaceuticals Ltd. Methods for accelerated return of skin integrity and for the treatment of impetigo
MX359879B (es) 2009-10-02 2018-10-12 Foamix Pharmaceuticals Ltd Composiciones tópicas de tetraciclina.
EP3574908B8 (en) * 2011-05-12 2024-09-11 Almirall LLC Pharmaceutical composition for oral administration comprising crystalline salts of (4s, 4as, 5ar, 12as)-4-dimethylamino-3,10,12,12a-tetrahydroxy-7-[(methoxy(methyl)amino)-methyl]-1,11-dioxo-1,4,4a,5,5a,6,11,12a-octahydro-naphthacene-2carboxylic acid amide
KR20240051297A (ko) * 2015-03-24 2024-04-19 파라테크 파마슈티컬스, 인크. 생물방어를 위한 미노시클린 화합물
GB201509326D0 (en) 2015-05-29 2015-07-15 Antibio Tx Aps Novel use
MX2018013271A (es) * 2016-05-02 2019-03-28 Paratek Pharm Innc Compuestos 9-aminometil minociclina y metodos para utilizarlos en el tratamiento de infeccion de vias urinarias (ivu).
TWI746610B (zh) * 2016-08-03 2021-11-21 美商派瑞泰Spv2有限公司 9-胺甲基米諾四環素化合物及其用途
CA2978573A1 (en) 2016-09-08 2018-03-08 Foamix Pharmaceuticals Ltd. Compositions and methods for treating rosacea and acne
GB201615693D0 (en) 2016-09-15 2016-11-02 Combinatorx Infection Ltd Combinations
US10383884B2 (en) * 2016-11-01 2019-08-20 Paratek Pharmaceuticals, Inc. 9-aminomethyl minocycline compounds and use thereof in treating community-acquired bacterial pneumonia (CABP)
LT3917616T (lt) 2019-01-31 2025-08-11 Takeda Pharmaceutical Company Limited Heterocikliniai junginiai ir jų naudojimas
US11419834B2 (en) 2019-02-25 2022-08-23 Rhode Island Hospital Methods for treating diseases or infections caused by or associated with H. pylori using a halogenated salicylanilide
GB201902580D0 (en) * 2019-02-26 2019-04-10 Healx Ltd Treatment
JP2023530415A (ja) * 2020-06-11 2023-07-18 パラテック ファーマシューティカルズ,インコーポレイテッド オマダサイクリンの結晶形態、その合成方法及びその使用方法
PT117254B (pt) 2021-05-26 2024-04-18 Hovione Farm S A Método de síntese de compostos 9-aminometil tetraciclinas

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Also Published As

Publication number Publication date
JP2011513404A (ja) 2011-04-28
CN102015602A (zh) 2011-04-13
MX2010009693A (es) 2010-12-20
WO2009111064A3 (en) 2010-03-11
US20210121483A1 (en) 2021-04-29
EP2262754A4 (en) 2012-03-14
US20090253660A1 (en) 2009-10-08
CL2010000188A1 (es) 2011-04-01
KR20100126469A (ko) 2010-12-01
US9724358B2 (en) 2017-08-08
EP2262754A2 (en) 2010-12-22
US20240131037A1 (en) 2024-04-25
US20240226119A9 (en) 2024-07-11
RU2010140682A (ru) 2012-04-10
US20160228459A1 (en) 2016-08-11
US20200289532A1 (en) 2020-09-17
WO2009111064A2 (en) 2009-09-11
US20180015108A1 (en) 2018-01-18
CA2717703A1 (en) 2009-09-11
AU2009220171A1 (en) 2009-09-11
US9265740B2 (en) 2016-02-23
US10124014B2 (en) 2018-11-13
US20150087711A1 (en) 2015-03-26
US20250213595A1 (en) 2025-07-03
US20190142850A1 (en) 2019-05-16

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]