BRPI0912995A2 - compostos tricíclicos contendo nitrogênio e sua utilização como agentes antibacterianos - Google Patents

compostos tricíclicos contendo nitrogênio e sua utilização como agentes antibacterianos

Info

Publication number
BRPI0912995A2
BRPI0912995A2 BRPI0912995A BRPI0912995A BRPI0912995A2 BR PI0912995 A2 BRPI0912995 A2 BR PI0912995A2 BR PI0912995 A BRPI0912995 A BR PI0912995A BR PI0912995 A BRPI0912995 A BR PI0912995A BR PI0912995 A2 BRPI0912995 A2 BR PI0912995A2
Authority
BR
Brazil
Prior art keywords
nitrogen
antibacterial agents
tricyclic compounds
containing tricyclic
compounds
Prior art date
Application number
BRPI0912995A
Other languages
English (en)
Inventor
Alan Joseph Hennessy
Carlos Alemparte-Gallardo
Christopher Barfoot
David Barros-Aguirre
Jose Maria Fiandor Roman
Modesto Jesus Remuinan-Blanco
Monica Cacho-Izquierdo
Neil David Pearson
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of BRPI0912995A2 publication Critical patent/BRPI0912995A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0912995A 2008-05-23 2009-05-20 compostos tricíclicos contendo nitrogênio e sua utilização como agentes antibacterianos BRPI0912995A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP08382018 2008-05-23
EP08382044 2008-10-17
EP08382057 2008-10-17
PCT/EP2009/056177 WO2009141398A1 (en) 2008-05-23 2009-05-20 Tricyclic nitrogen containing compounds and their use as antibacterials

Publications (1)

Publication Number Publication Date
BRPI0912995A2 true BRPI0912995A2 (pt) 2015-10-13

Family

ID=40874958

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0912995A BRPI0912995A2 (pt) 2008-05-23 2009-05-20 compostos tricíclicos contendo nitrogênio e sua utilização como agentes antibacterianos

Country Status (24)

Country Link
US (1) US8097628B2 (pt)
EP (1) EP2300476B1 (pt)
JP (1) JP5474941B2 (pt)
KR (1) KR20110016947A (pt)
CN (1) CN102105473B (pt)
AR (1) AR071869A1 (pt)
AU (1) AU2009248786B2 (pt)
BR (1) BRPI0912995A2 (pt)
CA (1) CA2725726A1 (pt)
CL (1) CL2009001267A1 (pt)
CO (1) CO6321284A2 (pt)
CR (1) CR11838A (pt)
DO (1) DOP2010000342A (pt)
EA (1) EA018817B1 (pt)
ES (1) ES2455496T3 (pt)
IL (1) IL209270A (pt)
MA (1) MA32406B1 (pt)
MX (1) MX2010012732A (pt)
NZ (1) NZ589062A (pt)
PE (1) PE20091927A1 (pt)
TW (1) TW201008941A (pt)
UY (1) UY31839A (pt)
WO (1) WO2009141398A1 (pt)
ZA (1) ZA201007945B (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2009248774B2 (en) 2008-05-23 2012-05-31 Novartis Ag Derivatives of quinolines and quinoxalines as protein tyrosine kinase inhibitors
JP2012505866A (ja) * 2008-10-17 2012-03-08 グラクソ グループ リミテッド 抗菌剤として使用される三環式窒素化合物
JP5857040B2 (ja) 2010-05-04 2016-02-10 アルカーメス ファーマ アイルランド リミテッド 酸化ラクタム化合物の合成方法
EP2844655A1 (en) 2012-05-02 2015-03-11 Lupin Limited Substituted pyridine compounds as crac modulators
CN103113291B (zh) * 2013-02-04 2015-03-04 浙江大学 一种3位烯基吡啶衍生物的合成方法
AR101674A1 (es) 2014-08-22 2017-01-04 Glaxosmithkline Ip Dev Ltd Uso de un compuesto tricíclico que contiene nitrógeno
EP3468975B1 (en) 2016-06-08 2020-04-01 Aziende Chimiche Riunite Angelini Francesco A.C.R. New antibacterial compounds
WO2021198981A1 (en) 2020-04-01 2021-10-07 Janssen Biopharma, Inc. Antiviral compounds and uses thereof
KR20250006204A (ko) 2022-04-25 2025-01-10 니뽄 신야쿠 가부시키가이샤 Ddr1 키나아제 저해제로서의 화합물 및 의약

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007071936A1 (en) * 2005-12-22 2007-06-28 Glaxo Group Limited Heterocyclic compounds, their preparation and their use as antibacterials
ATE481406T1 (de) * 2006-04-06 2010-10-15 Glaxo Group Ltd Pyrrolochinoxalinonderivate als antibakterielle mittel
PT2137196E (pt) * 2007-04-20 2010-12-16 Glaxo Group Ltd Compostos tricíclicos contendo azoto como agentes antibacterianos
GB0707706D0 (en) * 2007-04-20 2007-05-30 Glaxo Group Ltd Compounds

Also Published As

Publication number Publication date
US8097628B2 (en) 2012-01-17
MA32406B1 (fr) 2011-06-01
CL2009001267A1 (es) 2010-12-31
IL209270A0 (en) 2011-01-31
TW201008941A (en) 2010-03-01
MX2010012732A (es) 2010-12-07
EA018817B1 (ru) 2013-10-30
EA201071352A1 (ru) 2011-06-30
AU2009248786A1 (en) 2009-11-26
IL209270A (en) 2013-09-30
UY31839A (es) 2009-12-14
US20090306089A1 (en) 2009-12-10
CA2725726A1 (en) 2009-11-26
CN102105473B (zh) 2013-05-08
NZ589062A (en) 2012-06-29
ZA201007945B (en) 2011-08-31
CO6321284A2 (es) 2011-09-20
EP2300476B1 (en) 2014-01-08
PE20091927A1 (es) 2010-01-21
KR20110016947A (ko) 2011-02-18
ES2455496T3 (es) 2014-04-15
EP2300476A1 (en) 2011-03-30
CR11838A (es) 2011-03-25
AU2009248786B2 (en) 2013-04-04
WO2009141398A1 (en) 2009-11-26
AR071869A1 (es) 2010-07-21
JP5474941B2 (ja) 2014-04-16
JP2011520943A (ja) 2011-07-21
CN102105473A (zh) 2011-06-22
DOP2010000342A (es) 2010-11-30

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]