BRPI0919295A2 - 1h-benzimidazol-5-carboxamidas como agentes anti-inflamatórios. - Google Patents

1h-benzimidazol-5-carboxamidas como agentes anti-inflamatórios.

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Publication number
BRPI0919295A2
BRPI0919295A2 BRPI0919295A BRPI0919295A BRPI0919295A2 BR PI0919295 A2 BRPI0919295 A2 BR PI0919295A2 BR PI0919295 A BRPI0919295 A BR PI0919295A BR PI0919295 A BRPI0919295 A BR PI0919295A BR PI0919295 A2 BRPI0919295 A2 BR PI0919295A2
Authority
BR
Brazil
Prior art keywords
carboxamides
benzimidazole
inflammatory agents
inflammatory
agents
Prior art date
Application number
BRPI0919295A
Other languages
English (en)
Inventor
Dirk Stenkamp
Henning Priepke
Henri Doods
Juergen Mack
Kirsten Arndt
Klaus Klinder
Norbert Hauel
Raimund Kuelzer
Roland Pfau
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40344110&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0919295(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of BRPI0919295A2 publication Critical patent/BRPI0919295A2/pt

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    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30Nitrogen atoms not forming part of a nitro radical
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
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    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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BRPI0919295A 2008-09-25 2009-09-25 1h-benzimidazol-5-carboxamidas como agentes anti-inflamatórios. BRPI0919295A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9998708P 2008-09-25 2008-09-25
EP08165120 2008-09-25
PCT/EP2009/062421 WO2010034796A1 (en) 2008-09-25 2009-09-25 1h-benz imidazole-5-carboxamides as anti-inflammatory agents

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BRPI0919295A2 true BRPI0919295A2 (pt) 2015-12-15

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Family Applications (3)

Application Number Title Priority Date Filing Date
BRPI0919738A BRPI0919738A2 (pt) 2008-09-25 2009-09-25 3h-imidazo[4,5-c] piridino-6-carboxamidas como agentes anti-inflamatórios
BRPI0919292A BRPI0919292A2 (pt) 2008-09-25 2009-09-25 3h-imidazo[4,5-b] piridina-6-carboxamidas como agentes anti-inflamatórios
BRPI0919295A BRPI0919295A2 (pt) 2008-09-25 2009-09-25 1h-benzimidazol-5-carboxamidas como agentes anti-inflamatórios.

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AU2009295816A1 (en) 2010-04-01
AR073403A1 (es) 2010-11-03
US20110312935A1 (en) 2011-12-22
CA2738083A1 (en) 2010-04-01
CN102164911A (zh) 2011-08-24
US8598190B2 (en) 2013-12-03
EP2350073A1 (en) 2011-08-03
US8703796B2 (en) 2014-04-22
NZ591846A (en) 2012-11-30
NZ591847A (en) 2013-01-25
US20120115902A1 (en) 2012-05-10
CN102164924A (zh) 2011-08-24
JP2012503627A (ja) 2012-02-09
WO2010034799A1 (en) 2010-04-01
KR20110056530A (ko) 2011-05-30
AU2009295814A1 (en) 2010-04-01
KR20110065478A (ko) 2011-06-15
JP2012503630A (ja) 2012-02-09
AU2009295815A1 (en) 2010-04-01
CN102224143A (zh) 2011-10-19
TW201018669A (en) 2010-05-16
US20110275656A1 (en) 2011-11-10
JP2012503628A (ja) 2012-02-09
RU2011116133A (ru) 2012-10-27
WO2010034797A1 (en) 2010-04-01
BRPI0919738A2 (pt) 2015-12-08
AR073684A1 (es) 2010-11-24
WO2010034798A1 (en) 2010-04-01
UY32138A (es) 2010-04-30
MX2011002948A (es) 2011-04-26
EP2361252A1 (en) 2011-08-31
KR20110056533A (ko) 2011-05-30
RU2011116131A (ru) 2012-10-27
BRPI0919292A2 (pt) 2017-05-30
JP5591807B2 (ja) 2014-09-17
CA2737839A1 (en) 2010-04-01
EP2334664A1 (en) 2011-06-22
ZA201101041B (en) 2011-10-26
TW201016682A (en) 2010-05-01
US9040565B2 (en) 2015-05-26
AU2009295813A1 (en) 2010-04-01
NZ591843A (en) 2012-09-28
TW201018684A (en) 2010-05-16
AR073686A1 (es) 2010-11-24
RU2011116129A (ru) 2012-10-27
EP2334652A1 (en) 2011-06-22
JP5342646B2 (ja) 2013-11-13
CA2737384A1 (en) 2010-04-01
IL211148A0 (en) 2011-04-28
ZA201101042B (en) 2011-10-26
US8916599B2 (en) 2014-12-23
MX2011003094A (es) 2011-04-26
MX2011002903A (es) 2011-04-11
NZ591845A (en) 2012-10-26
TW201016696A (en) 2010-05-01
EP2350073B1 (en) 2014-11-12
JP5591808B2 (ja) 2014-09-17
AR073685A1 (es) 2010-11-24
JP5342647B2 (ja) 2013-11-13
US20120122930A1 (en) 2012-05-17
MX2011003152A (es) 2011-04-27
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JP2012503629A (ja) 2012-02-09
RU2011116128A (ru) 2012-10-27

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