BRPI0920764A2 - composto com estrutura de carbono spiro quiral, método de preparação do mesmo, e composição farmacêutica contendo o mesmo - Google Patents
composto com estrutura de carbono spiro quiral, método de preparação do mesmo, e composição farmacêutica contendo o mesmoInfo
- Publication number
- BRPI0920764A2 BRPI0920764A2 BRPI0920764A BRPI0920764A BRPI0920764A2 BR PI0920764 A2 BRPI0920764 A2 BR PI0920764A2 BR PI0920764 A BRPI0920764 A BR PI0920764A BR PI0920764 A BRPI0920764 A BR PI0920764A BR PI0920764 A2 BRPI0920764 A2 BR PI0920764A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- pharmaceutical composition
- composition containing
- same
- carbon structure
- Prior art date
Links
- -1 carbon structure compound Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000003003 spiro group Chemical group 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/10—Spiro-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Gastroenterology & Hepatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20080107821 | 2008-10-31 | ||
| PCT/KR2009/006357 WO2010050783A2 (ko) | 2008-10-31 | 2009-10-30 | 스파이로키랄 탄소 골격을 갖는 신규한 화합물, 그의 제조방법 및 그를 포함하는 약제학적 조성물 |
| KR1020090104124A KR101149878B1 (ko) | 2008-10-31 | 2009-10-30 | 스파이로키랄 탄소 골격을 갖는 신규한 화합물, 그의 제조방법 및 그를 포함하는 약제학적 조성물 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0920764A2 true BRPI0920764A2 (pt) | 2015-12-22 |
Family
ID=42275585
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0920764A BRPI0920764A2 (pt) | 2008-10-31 | 2009-10-30 | composto com estrutura de carbono spiro quiral, método de preparação do mesmo, e composição farmacêutica contendo o mesmo |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US8703813B2 (pt) |
| EP (1) | EP2363400B1 (pt) |
| JP (1) | JP2012507509A (pt) |
| KR (1) | KR101149878B1 (pt) |
| CN (1) | CN102203099B (pt) |
| AU (1) | AU2009310544A1 (pt) |
| BR (1) | BRPI0920764A2 (pt) |
| CA (1) | CA2742364A1 (pt) |
| ES (1) | ES2423196T3 (pt) |
| RU (1) | RU2492173C2 (pt) |
| WO (1) | WO2010050783A2 (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012033353A2 (ko) * | 2010-09-07 | 2012-03-15 | 서울대학교 산학협력단 | 세스터터핀 화합물 및 이들 물질의 용도 |
| KR101647507B1 (ko) | 2014-10-20 | 2016-08-10 | 건국대학교 글로컬산학협력단 | 정전용량 기반의 혈관삽입형 바이오센서를 이용한 심혈관 질환 진단 데이터 획득 시스템 및 방법 |
| CN104873499B (zh) * | 2015-06-11 | 2017-10-17 | 中国医学科学院医药生物技术研究所 | 一种上调Runx2 转录活性的化合物在防治骨质疏松中的应用 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5328929A (en) * | 1993-07-02 | 1994-07-12 | Arizona Board Of Regents | Isolation and structure of spongistatin 2, spongistatin 3, spongistatin 4 and spongistatin 6 |
| JP3331028B2 (ja) | 1993-11-16 | 2002-10-07 | 第一製薬株式会社 | スピロ化合物及びその製法 |
| JP2003514033A (ja) * | 1999-11-15 | 2003-04-15 | パーカー ヒューズ インスティテュート | 癌治療用のホルボキサゾール誘導体 |
| JP2005035895A (ja) * | 2003-07-15 | 2005-02-10 | Institute Of Physical & Chemical Research | 高カルシウム血症および骨疾患治療剤 |
| US7485631B2 (en) * | 2005-04-21 | 2009-02-03 | The Trustees Of The University Of Pennsylvania | Phorboxazole compounds and methods of their preparation |
| JP4696870B2 (ja) * | 2005-11-21 | 2011-06-08 | Jfeスチール株式会社 | 高強度鋼板及びその製造方法 |
| JP3988833B2 (ja) | 2006-12-01 | 2007-10-10 | 日東電工株式会社 | 新規セスキテルペン系化合物、その製造方法及び組成物 |
-
2009
- 2009-10-30 JP JP2011534397A patent/JP2012507509A/ja not_active Ceased
- 2009-10-30 CN CN200980143890.9A patent/CN102203099B/zh not_active Expired - Fee Related
- 2009-10-30 RU RU2011121877/04A patent/RU2492173C2/ru not_active IP Right Cessation
- 2009-10-30 US US13/126,979 patent/US8703813B2/en active Active
- 2009-10-30 AU AU2009310544A patent/AU2009310544A1/en not_active Abandoned
- 2009-10-30 KR KR1020090104124A patent/KR101149878B1/ko not_active Expired - Fee Related
- 2009-10-30 BR BRPI0920764A patent/BRPI0920764A2/pt not_active IP Right Cessation
- 2009-10-30 ES ES09823863T patent/ES2423196T3/es active Active
- 2009-10-30 CA CA2742364A patent/CA2742364A1/en not_active Abandoned
- 2009-10-30 EP EP09823863.7A patent/EP2363400B1/en not_active Not-in-force
- 2009-10-30 WO PCT/KR2009/006357 patent/WO2010050783A2/ko not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| EP2363400A4 (en) | 2012-04-18 |
| CA2742364A1 (en) | 2010-05-06 |
| CN102203099A (zh) | 2011-09-28 |
| EP2363400B1 (en) | 2013-06-12 |
| RU2011121877A (ru) | 2012-12-10 |
| AU2009310544A1 (en) | 2010-05-06 |
| KR101149878B1 (ko) | 2012-05-24 |
| JP2012507509A (ja) | 2012-03-29 |
| EP2363400A2 (en) | 2011-09-07 |
| ES2423196T3 (es) | 2013-09-18 |
| RU2492173C2 (ru) | 2013-09-10 |
| US8703813B2 (en) | 2014-04-22 |
| CN102203099B (zh) | 2014-03-12 |
| WO2010050783A3 (ko) | 2010-09-10 |
| KR20100048934A (ko) | 2010-05-11 |
| WO2010050783A2 (ko) | 2010-05-06 |
| US20110218240A1 (en) | 2011-09-08 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK2282994T3 (da) | 3-aminocarbazolforbindelse, farmaceutisk sammensætning indeholdende forbindelsen samt fremstillingsmetode derfor | |
| BRPI0917579A2 (pt) | composto, composição farmacêutica, métodos, e, uso de um composto | |
| BRPI0920263A2 (pt) | composto, uso do composto, composição, e, método | |
| EP2429987A4 (en) | AMIDE COMPOUND, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME | |
| BRPI0821115A2 (pt) | Composto derivado de aminotriazol, medicamento, composição farmacêutica e uso do composto | |
| BRPI0919942A2 (pt) | Composto, composição farmacêutica, e, uso de um composto | |
| BRPI0907562A2 (pt) | composto, composição farmacêutica, e, uso de um composto | |
| BRPI0921375A2 (pt) | composto, composição farmacêutica, e, uso de um composto | |
| BRPI0906962A2 (pt) | Composto, e, composição farmacêutica | |
| BRPI0906556A2 (pt) | Composto, e, composição farmacêutica | |
| BRPI0917001A2 (pt) | composto, composição farmacêutica, e, uso de um composto ou uma composição farmacêutica | |
| BR112012022878A2 (pt) | composto, composição farmacêutica, uso do compostos e método de tratamento | |
| BRPI0918360A2 (pt) | composto, composição farmacêutica e usos de um composto | |
| BRPI0917315A2 (pt) | anticorpo, composicao farmaceutico, e, uso de uma composicao farmaceutica | |
| BRPI0913739A2 (pt) | Composição líquida, método, e, uso de composição | |
| CL2007002377A1 (es) | Compuestos derivados de quinazolina; procedimiento de preparacion; composicion farmaceutica; y su uso como anticancerigeno. | |
| BR112012022879A2 (pt) | composto, composição farmacêutica, uso do composto e método de tratamento | |
| BRPI0921879A2 (pt) | composto, composição farmacêutica , e, uso de um composto | |
| BR112012004335A2 (pt) | composto, composição farmacêutica, e, uso do composto. | |
| BRPI0809661A2 (pt) | Composição farmacêutica estabilizada contendo pregabalina | |
| BRPI0917681A2 (pt) | Composto, e, composição farmacêutica | |
| BRPI0915120A2 (pt) | composto derivado de oxima, uso do referido composto e composição farmacêutica | |
| BRPI1008039A2 (pt) | composto, mistura, composição farmacêutica, e, uso de um coposto, de uma mistura ou de uma composição farmacêutica | |
| BRPI0906937A2 (pt) | composto, composição farmacêutica, e, uso de um composto | |
| BRPI0910179A2 (pt) | composto de amina, composição farmacêutica e uso do composto de amina |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 6A E 7A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |