BRPI0921019A2 - processo para obtenção de uma composição de rosuvastatina cálcica e produto obtido - Google Patents
processo para obtenção de uma composição de rosuvastatina cálcica e produto obtidoInfo
- Publication number
- BRPI0921019A2 BRPI0921019A2 BRPI0921019A BRPI0921019A BRPI0921019A2 BR PI0921019 A2 BRPI0921019 A2 BR PI0921019A2 BR PI0921019 A BRPI0921019 A BR PI0921019A BR PI0921019 A BRPI0921019 A BR PI0921019A BR PI0921019 A2 BRPI0921019 A2 BR PI0921019A2
- Authority
- BR
- Brazil
- Prior art keywords
- obtaining
- composition
- product obtained
- calcium rosuvastatin
- rosuvastatin
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MX2008014321A MX344885B (es) | 2008-11-10 | 2008-11-10 | Proceso para la obtencion de una composicion de rosuvastatina calcica y producto obtenido. |
| PCT/MX2009/000081 WO2010053343A1 (es) | 2008-11-10 | 2009-07-29 | Proceso para la obtención de una composición de rosuvastatina cálcica y producto obtenido |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0921019A2 true BRPI0921019A2 (pt) | 2015-12-22 |
Family
ID=42153048
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0921019A BRPI0921019A2 (pt) | 2008-11-10 | 2009-07-29 | processo para obtenção de uma composição de rosuvastatina cálcica e produto obtido |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20120269890A1 (pt) |
| EP (1) | EP2347758A4 (pt) |
| JP (1) | JP2012508230A (pt) |
| BR (1) | BRPI0921019A2 (pt) |
| CA (1) | CA2744820C (pt) |
| MX (1) | MX344885B (pt) |
| NZ (1) | NZ593349A (pt) |
| WO (1) | WO2010053343A1 (pt) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20200003219A (ko) | 2011-05-20 | 2020-01-08 | 아스트라제네카 유케이 리미티드 | 로수바스타틴 칼슘의 약학 조성물 |
| CN103874490A (zh) * | 2011-08-15 | 2014-06-18 | 工业研究与发展基金会有限公司 | 咔咯和他汀类药物的组合 |
| JP6161867B2 (ja) * | 2011-11-17 | 2017-07-12 | 株式会社アドバンテスト | 滑沢剤の展延解析装置、方法、プログラム、記録媒体 |
| WO2013083674A1 (de) * | 2011-12-08 | 2013-06-13 | Hexal Ag | Neue pharmazeutische statin-zusammensetzung |
| JP2016098187A (ja) * | 2014-11-19 | 2016-05-30 | ニプロ株式会社 | 口腔内崩壊錠 |
| JP6108635B2 (ja) * | 2015-05-14 | 2017-04-05 | ダイト株式会社 | ロスバスタチン含有口腔内速崩壊錠 |
| JP6167192B2 (ja) * | 2016-01-19 | 2017-07-19 | 株式会社アドバンテスト | 滑沢剤の展延解析装置、方法、プログラム、記録媒体 |
| CN110151725B (zh) * | 2019-06-26 | 2021-06-18 | 海南通用三洋药业有限公司 | 一种稳定的瑞舒伐他汀钙胶囊剂及其制备方法 |
| CN110974793A (zh) * | 2019-12-26 | 2020-04-10 | 鲁南制药集团股份有限公司 | 一种瑞舒伐他汀钙片剂及其制备方法 |
| CN113230223B (zh) * | 2021-05-13 | 2023-04-07 | 宜昌人福药业有限责任公司 | 阿托伐他汀钙薄膜包衣片的制备方法 |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8679534B2 (en) * | 1997-12-12 | 2014-03-25 | Andrx Labs, Llc | HMG-CoA reductase inhibitor extended release formulation |
| US7374779B2 (en) * | 1999-02-26 | 2008-05-20 | Lipocine, Inc. | Pharmaceutical formulations and systems for improved absorption and multistage release of active agents |
| GB0001621D0 (en) * | 2000-01-26 | 2000-03-15 | Astrazeneca Ab | Pharmaceutical compositions |
| AR030414A1 (es) * | 2000-04-03 | 2003-08-20 | Astrazeneca Ab | Combinacion farmaceutica que comprende un beta bloqueante y un inhibidor de hmg-coa reductasa , formulacion farmaceutica, equipo transportable de partes , uso de esta combinacion y de esta formulacion para preparar medicamentos |
| GB0111077D0 (en) * | 2001-05-04 | 2001-06-27 | Biochemie Gmbh | Organic compounds |
| DE10204336A1 (de) * | 2002-02-01 | 2003-08-14 | Merck Patent Gmbh | Verwendung von Mehrschichtpigmenten im Lebensmittel- und Pharmabereich |
| US20030171407A1 (en) * | 2002-03-07 | 2003-09-11 | Upsher-Smith Laboratories, Inc. | Composition for reducing blood glucose and cholesterol |
| AU2003227691B2 (en) * | 2002-05-03 | 2008-05-15 | Hexal Ag | Stable pharmaceutical formulation for a combination of a statin and an ace inhibitor |
| GB0217306D0 (en) * | 2002-07-25 | 2002-09-04 | Novartis Ag | Compositions comprising organic compounds |
| AR040588A1 (es) * | 2002-07-26 | 2005-04-13 | Schering Corp | Formulacion farmaceutica que comprende un inhibidor de la absorcion del colesterol y un inhibidor de una hmg- co a reductasa |
| EP1599192A4 (en) * | 2003-02-20 | 2009-06-03 | Bpsi Holdings Inc | SHIMMERING FILM COATING SYSTEMS AND SUBSTRATES THAT ARE COATED |
| US7179916B2 (en) * | 2004-07-13 | 2007-02-20 | Teva Pharmaceutical Industries Ltd. | Process for the preparation of rosuvastatin |
| WO2006134604A1 (en) * | 2005-06-15 | 2006-12-21 | Hetero Drugs Limited | Combination composition of cholesterol absorption inhibitor and 3-hydroxy-3-methylglutaryl-coenzyme a (hmg-coa) reductase inhibitor |
| EP1741427A1 (en) * | 2005-07-06 | 2007-01-10 | KRKA, D.D., Novo Mesto | Pharmaceutical composition comprising simvastatin and ezetimibe |
| US20070053892A1 (en) * | 2005-09-07 | 2007-03-08 | Everett Laboratories, Inc. | Methods and kits for co-administration of nutritional supplements |
| TW200744583A (en) * | 2006-03-14 | 2007-12-16 | Ranbaxy Lab Ltd | Statin stabilizing dosage formulations |
| WO2008062476A2 (en) * | 2006-10-31 | 2008-05-29 | Glenmark Pharmaceutical Limited | Pharmaceutical composition comprising rosuvastatin or pharmaceutically accepatble salts thereof |
| JP2010519216A (ja) * | 2007-02-15 | 2010-06-03 | ファイザー・リミテッド | Ccr5拮抗薬のための医薬組成物および方法 |
| CL2008003154A1 (es) * | 2007-10-26 | 2009-10-23 | Eurofarma Laboratorios LTDA | Proceso de obtencion de un extracto estandarizado de aleuterites moluccana; extracto estandarizado de aleurites moluccana; composicion farmaceutica que comprende el extracto; uso del extracto para tratar condiciones de dolor. |
-
2008
- 2008-11-10 MX MX2008014321A patent/MX344885B/es active IP Right Grant
-
2009
- 2009-07-29 CA CA2744820A patent/CA2744820C/en active Active
- 2009-07-29 WO PCT/MX2009/000081 patent/WO2010053343A1/es not_active Ceased
- 2009-07-29 EP EP09825024A patent/EP2347758A4/en not_active Ceased
- 2009-07-29 NZ NZ593349A patent/NZ593349A/xx not_active IP Right Cessation
- 2009-07-29 BR BRPI0921019A patent/BRPI0921019A2/pt not_active IP Right Cessation
- 2009-07-29 JP JP2011535525A patent/JP2012508230A/ja active Pending
- 2009-07-29 US US13/128,329 patent/US20120269890A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2010053343A1 (es) | 2010-05-14 |
| CA2744820A1 (en) | 2010-05-14 |
| EP2347758A4 (en) | 2012-04-25 |
| NZ593349A (en) | 2012-12-21 |
| MX344885B (es) | 2017-01-10 |
| US20120269890A1 (en) | 2012-10-25 |
| MX2008014321A (es) | 2010-06-07 |
| CA2744820C (en) | 2016-03-01 |
| JP2012508230A (ja) | 2012-04-05 |
| EP2347758A1 (en) | 2011-07-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2383 DE 06-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |