BRPI0923215A2 - método para fabricar um composto. - Google Patents
método para fabricar um composto.Info
- Publication number
- BRPI0923215A2 BRPI0923215A2 BRPI0923215A BRPI0923215A BRPI0923215A2 BR PI0923215 A2 BRPI0923215 A2 BR PI0923215A2 BR PI0923215 A BRPI0923215 A BR PI0923215A BR PI0923215 A BRPI0923215 A BR PI0923215A BR PI0923215 A2 BRPI0923215 A2 BR PI0923215A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- making
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/12—Oxygen or sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US12204408P | 2008-12-12 | 2008-12-12 | |
| PCT/SE2009/051404 WO2010068172A1 (en) | 2008-12-12 | 2009-12-11 | A new process for preparing 4- [4-methyl-5- (cl- 10alkylthio/c5-10aryl-cl-6alkylthio) -4h-1, 2, 4-triazol-3- yl] pyridines. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0923215A2 true BRPI0923215A2 (pt) | 2017-06-06 |
Family
ID=42242955
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0923215A BRPI0923215A2 (pt) | 2008-12-12 | 2009-12-11 | método para fabricar um composto. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20110295016A1 (pt) |
| EP (1) | EP2376474A4 (pt) |
| JP (1) | JP2012511570A (pt) |
| KR (1) | KR20110089868A (pt) |
| CN (1) | CN102245592A (pt) |
| AU (1) | AU2009325178A1 (pt) |
| BR (1) | BRPI0923215A2 (pt) |
| CA (1) | CA2745870A1 (pt) |
| IL (1) | IL213035A0 (pt) |
| MX (1) | MX2011005981A (pt) |
| SG (1) | SG171743A1 (pt) |
| WO (1) | WO2010068172A1 (pt) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3210469A1 (de) | 2016-02-23 | 2017-08-30 | Bayer Cropscience AG | Verwendung von substituierten thio-1,2,4-triazolen zur steigerung der stresstoleranz in pflanzen |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4900743A (en) * | 1987-01-27 | 1990-02-13 | Merrell Dow Pharmaceuticals Inc. | 3-aryl-5-alkylthio-4H-1,2,4-triazoles |
| WO2002078696A1 (en) * | 2001-03-29 | 2002-10-10 | Smithkline Beecham Corporation | Compounds and methods |
| RU2006127575A (ru) * | 2004-02-18 | 2008-03-27 | Астразенека Аб (Se) | Соединение триазола и их применение в качестве антагонистов метаботропного рецептора глутамата |
| WO2005080356A1 (en) * | 2004-02-18 | 2005-09-01 | Astrazeneca Ab | Tetrazole compounds and their use as metabotropic glutamate receptor antagonits |
| SE0402591D0 (sv) * | 2004-10-25 | 2004-10-25 | Astrazeneca Ab | Novel use |
| UY29796A1 (es) * | 2005-09-29 | 2007-04-30 | Astrazeneca Ab | Nuevos compuestos para el tratamiento de trastornos neurológicos, psiquiátricos o del dolor |
-
2009
- 2009-12-11 BR BRPI0923215A patent/BRPI0923215A2/pt not_active IP Right Cessation
- 2009-12-11 WO PCT/SE2009/051404 patent/WO2010068172A1/en not_active Ceased
- 2009-12-11 CA CA2745870A patent/CA2745870A1/en not_active Abandoned
- 2009-12-11 US US13/139,090 patent/US20110295016A1/en not_active Abandoned
- 2009-12-11 KR KR1020117013380A patent/KR20110089868A/ko not_active Withdrawn
- 2009-12-11 MX MX2011005981A patent/MX2011005981A/es not_active Application Discontinuation
- 2009-12-11 JP JP2011540661A patent/JP2012511570A/ja active Pending
- 2009-12-11 AU AU2009325178A patent/AU2009325178A1/en not_active Abandoned
- 2009-12-11 EP EP09832207A patent/EP2376474A4/en not_active Withdrawn
- 2009-12-11 SG SG2011035482A patent/SG171743A1/en unknown
- 2009-12-11 CN CN200980149957XA patent/CN102245592A/zh active Pending
-
2011
- 2011-05-19 IL IL213035A patent/IL213035A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2012511570A (ja) | 2012-05-24 |
| SG171743A1 (en) | 2011-07-28 |
| CN102245592A (zh) | 2011-11-16 |
| WO2010068172A1 (en) | 2010-06-17 |
| CA2745870A1 (en) | 2010-06-17 |
| EP2376474A1 (en) | 2011-10-19 |
| AU2009325178A1 (en) | 2010-06-17 |
| KR20110089868A (ko) | 2011-08-09 |
| MX2011005981A (es) | 2011-06-27 |
| IL213035A0 (en) | 2011-07-31 |
| US20110295016A1 (en) | 2011-12-01 |
| EP2376474A4 (en) | 2012-07-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |