CA1093467A - Compose therapeutique contenant de la gomme xanthane ou de la gomme de caroube - Google Patents

Compose therapeutique contenant de la gomme xanthane ou de la gomme de caroube

Info

Publication number: CA1093467A
Authority: CA; Canada
Prior art keywords: gum; locust bean; composition; bean gum; xanthan gum
Prior art date: 1977-01-31
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

CA295,928A

Other languages

English (en)

Inventor

Song-Ling Lin

Maturu K. Pramoda

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Wyeth LLC

Original Assignee

American Home Products Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-01-31

Filing date

1978-01-30

Publication date

1981-01-13

1977-01-31 Priority claimed from US05/764,318 external-priority patent/US4136177A/en

1977-01-31 Priority claimed from US05/764,320 external-priority patent/US4136178A/en

1978-01-30 Application filed by American Home Products Corp filed Critical American Home Products Corp

1981-01-13 Application granted granted Critical

1981-01-13 Publication of CA1093467A publication Critical patent/CA1093467A/fr

Status Expired legal-status Critical Current

Links

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239000000230 xanthan gum Substances 0.000 title claims abstract description 33
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229960001442 gonadorelin Drugs 0.000 description 1
229960004905 gramicidin Drugs 0.000 description 1
ZWCXYZRRTRDGQE-SORVKSEFSA-N gramicidina Chemical compound C1=CC=C2C(C[C@H](NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](CC=3C4=CC=CC=C4NC=3)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](CC=3C4=CC=CC=C4NC=3)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](CC=3C4=CC=CC=C4NC=3)NC(=O)[C@H](C(C)C)NC(=O)[C@H](C(C)C)NC(=O)[C@@H](C(C)C)NC(=O)[C@H](C)NC(=O)[C@H](NC(=O)[C@H](C)NC(=O)CNC(=O)[C@@H](NC=O)C(C)C)CC(C)C)C(=O)NCCO)=CNC2=C1 ZWCXYZRRTRDGQE-SORVKSEFSA-N 0.000 description 1
239000000665 guar gum Substances 0.000 description 1
235000010417 guar gum Nutrition 0.000 description 1
229960002154 guar gum Drugs 0.000 description 1
229960000857 homatropine Drugs 0.000 description 1
229960000890 hydrocortisone Drugs 0.000 description 1
238000002513 implantation Methods 0.000 description 1
238000003780 insertion Methods 0.000 description 1
230000037431 insertion Effects 0.000 description 1
238000007918 intramuscular administration Methods 0.000 description 1
235000015110 jellies Nutrition 0.000 description 1
239000008274 jelly Substances 0.000 description 1
239000000314 lubricant Substances 0.000 description 1
239000002075 main ingredient Substances 0.000 description 1
238000000034 method Methods 0.000 description 1
244000005700 microbiome Species 0.000 description 1
150000002772 monosaccharides Chemical class 0.000 description 1
239000002997 ophthalmic solution Substances 0.000 description 1
239000000734 parasympathomimetic agent Substances 0.000 description 1
230000001499 parasympathomimetic effect Effects 0.000 description 1
229940005542 parasympathomimetics Drugs 0.000 description 1
229960001802 phenylephrine Drugs 0.000 description 1
SONNWYBIRXJNDC-VIFPVBQESA-N phenylephrine Chemical compound CNC[C@H](O)C1=CC=CC(O)=C1 SONNWYBIRXJNDC-VIFPVBQESA-N 0.000 description 1
229960001416 pilocarpine Drugs 0.000 description 1
229920001515 polyalkylene glycol Polymers 0.000 description 1
229920001223 polyethylene glycol Polymers 0.000 description 1
229920001184 polypeptide Polymers 0.000 description 1
239000001267 polyvinylpyrrolidone Substances 0.000 description 1
235000013855 polyvinylpyrrolidone Nutrition 0.000 description 1
239000011591 potassium Substances 0.000 description 1
229910052700 potassium Inorganic materials 0.000 description 1
239000001103 potassium chloride Substances 0.000 description 1
235000011164 potassium chloride Nutrition 0.000 description 1
229960005205 prednisolone Drugs 0.000 description 1
OIGNJSKKLXVSLS-VWUMJDOOSA-N prednisolone Chemical compound O=C1C=C[C@]2(C)[C@H]3[C@@H](O)C[C@](C)([C@@](CC4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 OIGNJSKKLXVSLS-VWUMJDOOSA-N 0.000 description 1
229960004618 prednisone Drugs 0.000 description 1
XOFYZVNMUHMLCC-ZPOLXVRWSA-N prednisone Chemical compound O=C1C=C[C@]2(C)[C@H]3C(=O)C[C@](C)([C@@](CC4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 XOFYZVNMUHMLCC-ZPOLXVRWSA-N 0.000 description 1
239000003755 preservative agent Substances 0.000 description 1
230000008569 process Effects 0.000 description 1
108090000765 processed proteins & peptides Proteins 0.000 description 1
102000004196 processed proteins & peptides Human genes 0.000 description 1
102000004169 proteins and genes Human genes 0.000 description 1
108090000623 proteins and genes Proteins 0.000 description 1
229960002646 scopolamine Drugs 0.000 description 1
STECJAGHUSJQJN-FWXGHANASA-N scopolamine Chemical compound C1([C@@H](CO)C(=O)O[C@H]2C[C@@H]3N([C@H](C2)[C@@H]2[C@H]3O2)C)=CC=CC=C1 STECJAGHUSJQJN-FWXGHANASA-N 0.000 description 1
239000011734 sodium Substances 0.000 description 1
229910052708 sodium Inorganic materials 0.000 description 1
229910000029 sodium carbonate Inorganic materials 0.000 description 1
UMKFIJKKXUZOJY-UHFFFAOYSA-N sodium;(4-aminophenyl)sulfonyl-(6-methoxypyridazin-3-yl)azanide Chemical compound [Na+].N1=NC(OC)=CC=C1[N-]S(=O)(=O)C1=CC=C(N)C=C1 UMKFIJKKXUZOJY-UHFFFAOYSA-N 0.000 description 1
239000007787 solid Substances 0.000 description 1
239000000600 sorbitol Substances 0.000 description 1
239000003381 stabilizer Substances 0.000 description 1
229960002673 sulfacetamide Drugs 0.000 description 1
SKIVFJLNDNKQPD-UHFFFAOYSA-N sulfacetamide Chemical compound CC(=O)NS(=O)(=O)C1=CC=C(N)C=C1 SKIVFJLNDNKQPD-UHFFFAOYSA-N 0.000 description 1
229960000654 sulfafurazole Drugs 0.000 description 1
230000000948 sympatholitic effect Effects 0.000 description 1
229940127230 sympathomimetic drug Drugs 0.000 description 1
229960002180 tetracycline Drugs 0.000 description 1
229930101283 tetracycline Natural products 0.000 description 1
235000019364 tetracycline Nutrition 0.000 description 1
150000003522 tetracyclines Chemical class 0.000 description 1
238000002560 therapeutic procedure Methods 0.000 description 1
JIVZKJJQOZQXQB-UHFFFAOYSA-N tolazoline Chemical compound C=1C=CC=CC=1CC1=NCCN1 JIVZKJJQOZQXQB-UHFFFAOYSA-N 0.000 description 1
229960002312 tolazoline Drugs 0.000 description 1
230000001988 toxicity Effects 0.000 description 1
231100000419 toxicity Toxicity 0.000 description 1
239000000080 wetting agent Substances 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Epidemiology (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Molecular Biology (AREA)
Ophthalmology & Optometry (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

CA295,928A 1977-01-31 1978-01-30 Compose therapeutique contenant de la gomme xanthane ou de la gomme de caroube Expired CA1093467A (fr)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US05/764,318 US4136177A (en)	1977-01-31	1977-01-31	Xanthan gum therapeutic compositions
US764,320		1977-01-31
US05/764,320 US4136178A (en)	1977-01-31	1977-01-31	Locust bean gum therapeutic compositions
US764,318		1977-01-31

Publications (1)

Publication Number	Publication Date
CA1093467A true CA1093467A (fr)	1981-01-13

Family

ID=27117438

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA295,928A Expired CA1093467A (fr)	1977-01-31	1978-01-30	Compose therapeutique contenant de la gomme xanthane ou de la gomme de caroube

Country Status (2)

Country	Link
CA (1)	CA1093467A (fr)
GB (1)	GB1593954A (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CL2009000985A1 (es) *	2008-04-26	2010-01-15	Alcon Res Ltd	Composicion oftalmica que comprende entre 0,16 y 0,19% p/v de un galactomanano, alrededor de 0,7% p/v de un borato, cis-diol y menos de 5 ppm de concentracion de cationes divalentes; y su uso para lubricar el ojo.
TWI478730B (zh)	2009-12-03	2015-04-01	Alcon Res Ltd	眼科乳劑
TWI913170B (zh)	2018-02-21	2026-01-21	瑞士商愛爾康公司	基於脂質的眼用乳劑

1978
- 1978-01-27 GB GB334978A patent/GB1593954A/en not_active Expired
- 1978-01-30 CA CA295,928A patent/CA1093467A/fr not_active Expired

Also Published As

Publication number	Publication date
GB1593954A (en)	1981-07-22

Legal Events

Date	Code	Title	Description
1998-01-20	MKEX	Expiry

Publication	Publication Date	Title
US4136177A (en)	1979-01-23	Xanthan gum therapeutic compositions
US4136178A (en)	1979-01-23	Locust bean gum therapeutic compositions
DE69522550T2 (de)	2002-05-02	Flüssiges ophthalmologisches abgabesystem mit verzögerter freisetzung
EP0533836B1 (fr)	1996-02-28	Compositions de gelification reversible et modes d'emploi
US4136173A (en)	1979-01-23	Mixed xanthan gum and locust beam gum therapeutic compositions
EP0227494B1 (fr)	1992-03-04	Composition pharmaceutique du type subissant une transition de phase liquide-gel
US6136334A (en)	2000-10-24	Medical uses of in situ formed gels
AU2016344349B2 (en)	2022-05-19	Pharmaceutical formulations that form gel in situ
US11376275B2 (en)	2022-07-05	Ophthalmic compositions with improved dessication protection and retention
EP2586426B1 (fr)	2015-09-23	Suspension de nanoparticules contenant un polymère de type carboxyvinyle
JPH05213757A (ja)	1993-08-24	水性液剤
WO2011018800A2 (fr)	2011-02-17	Nouvelle solution formant un gel in situ pour ladministration de médicaments par voie oculaire
DE60002719T2 (de)	2003-10-09	Ophthalmische zusammensetzungen in form wässriger gele
CA2193149C (fr)	2002-04-23	Systemes cationiques therapeutiques
JP3974431B2 (ja)	2007-09-12	アルギン酸含有組成物
CA1093467A (fr)	1981-01-13	Compose therapeutique contenant de la gomme xanthane ou de la gomme de caroube
JP2634436B2 (ja)	1997-07-23	ラムサンガムを含有する局所用眼科用組成物
EP3229780B1 (fr)	2018-11-28	Compositions ophtalmiques destinées à être utilisées dans le traitement du syndrome de l'oeil sec
EP0888770A1 (fr)	1999-01-07	Compositions pharmaceutiques contenant des polysaccharides cationiques et des médicaments cationiques
KR0159640B1 (ko)	1998-12-01	도파민 수용기 자극제를 포함하는 근시 및 녹내장 치료용 안과 제형
HK1248100B (zh)	2021-10-08	眼用原位凝胶处方
JPH10182498A (ja)	1998-07-07	カチオン治療方式
HK1178802B (en)	2016-04-29	Carboxyvinyl polymer-containing nanoparticle suspensions