CA1304540C - Dipeptides substitues, procedes pour leur preparation et composes pharmaceutiques en contenant, et leur utilisation pour l'inhibition de l'encephalinase
- Google Patents
Dipeptides substitues, procedes pour leur preparation et composes pharmaceutiques en contenant, et leur utilisation pour l'inhibition de l'encephalinase
Info
Publication number
CA1304540C
CA1304540CCA000405374ACA405374ACA1304540CCA 1304540 CCA1304540 CCA 1304540CCA 000405374 ACA000405374 ACA 000405374ACA 405374 ACA405374 ACA 405374ACA 1304540 CCA1304540 CCA 1304540C
Authority
CA
Canada
Prior art keywords
loweralkyl
aryl
substituted
compound
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Sharp and Dohme LLC
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to EP81110337ApriorityCriticalpatent/EP0054862B1/fr
Priority to CY140681Aprioritypatent/CY1406A/xx
Application filed by Schering CorpfiledCriticalSchering Corp
Priority to AU84947/82Aprioritypatent/AU560004B2/en
Priority to OA57714Aprioritypatent/OA07124A/fr
Priority to CA000405374Aprioritypatent/CA1304540C/fr
Application grantedgrantedCritical
Publication of CA1304540CpublicationCriticalpatent/CA1304540C/fr
Medicines That Contain Protein Lipid Enzymes And Other Medicines
(AREA)
Peptides Or Proteins
(AREA)
CA000405374A1980-12-181982-06-17Dipeptides substitues, procedes pour leur preparation et composes pharmaceutiques en contenant, et leur utilisation pour l'inhibition de l'encephalinase
Expired - LifetimeCA1304540C
(fr)
Substituted dipeptides, processes for their preparation and pharmaceutical compositions containing them and their use in the inhibition of enkephalinase
Dipeptides substitués, procédés pour leur préparation et compositions pharmaceutiques les contenant et leur utilisation pour l'inhibition de l'encéphalinase.
Dipeptides substitues, procedes pour leur preparation et composes pharmaceutiques en contenant, et leur utilisation pour l'inhibition de l'encephalinase
Dipeptides substitues, procedes pour leur preparation et composes pharmaceutiques en contenant, et leur utilisation pour l'inhibition de l'encephalinase
Dipeptides substitues, procedes pour leur preparation et composes pharmaceutiques en contenant, et leur utilisation pour l'inhibition de l'encephalinase
Process for the preparation of cis,endo-2-azabicyclo-square bracket-3.3.0-square bracket octan-3-carboxylic acids and pharmaceutical compositions containing said compounds
Dipeptides substitues, procedes pour leur preparation et composes pharmaceutiques en contenant, et leur utilisation pour l'inhibition de l'encephalinase
Acides n-¬(4,5-dihydroxy-et 4,5,8-trihydroxy-9,10-dihydro-9, 10-dioxo-2-anthracene-yl)carbonyl|amines utiles pour les therapies d'affectations osteoarticulaires
Substituted dipeptides,processes for their preparation and pharmaceutical compositions containing them and their use in the inhibition of enkephalinase