CA2003308A1 - Trialkylsilyl esters of amino acids and their uses in the synthesis of peptides - Google Patents

Trialkylsilyl esters of amino acids and their uses in the synthesis of peptides

Info

Publication number
CA2003308A1
CA2003308A1 CA002003308A CA2003308A CA2003308A1 CA 2003308 A1 CA2003308 A1 CA 2003308A1 CA 002003308 A CA002003308 A CA 002003308A CA 2003308 A CA2003308 A CA 2003308A CA 2003308 A1 CA2003308 A1 CA 2003308A1
Authority
CA
Canada
Prior art keywords
protected
amino
group
amino acid
alpha
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002003308A
Other languages
English (en)
French (fr)
Inventor
Anthony Atkinson
Michael R. Calder
Ram P. Sharma
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2003308A1 publication Critical patent/CA2003308A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/08—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents
    • C07K1/088—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents containing other elements, e.g. B, Si, As
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
CA002003308A 1988-11-19 1989-11-17 Trialkylsilyl esters of amino acids and their uses in the synthesis of peptides Abandoned CA2003308A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB888827083A GB8827083D0 (en) 1988-11-19 1988-11-19 Trialkylsilyl esters of amino acids & their use in synthesis of peptides
GB8827083.0 1988-11-19

Publications (1)

Publication Number Publication Date
CA2003308A1 true CA2003308A1 (en) 1990-05-19

Family

ID=10647130

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002003308A Abandoned CA2003308A1 (en) 1988-11-19 1989-11-17 Trialkylsilyl esters of amino acids and their uses in the synthesis of peptides

Country Status (10)

Country Link
EP (1) EP0444068A1 (de)
JP (1) JPH04502908A (de)
AU (1) AU4517289A (de)
CA (1) CA2003308A1 (de)
FI (1) FI912411A0 (de)
GB (1) GB8827083D0 (de)
HU (1) HUT58106A (de)
IL (1) IL92338A0 (de)
WO (1) WO1990005738A1 (de)
ZA (1) ZA898774B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9118669D0 (en) * 1991-08-30 1991-10-16 Univ Southampton Preparation of peptides by a soliphase synthesis and intermediates therefor
US7244815B2 (en) 2001-05-23 2007-07-17 The Curators Of The University Of Missouri Attachment and elaboration strategies for inverse peptide synthesis
WO2002094857A1 (en) * 2001-05-23 2002-11-28 The Curators Of The University Of Missouri Inverse solid phase synthesis of peptides
EP2060580A1 (de) * 2007-11-19 2009-05-20 SOLVAY (Société Anonyme) Verfahren zur Herstellung von persilylierten Peptiden
MX2013007006A (es) * 2010-12-22 2013-07-30 Onyx Pharma Inc Acoplamientos eficientes de peptidos y su uso en la sintesis y aislamiento de una sal trisodica de ciclopenta[g]quinazolina.
US9828393B2 (en) * 2013-07-22 2017-11-28 The Regents Of The University Of Colorado, A Body Corporate Silylalkyloxyaryl compounds and methods for treating cancer
CA3078393A1 (en) 2017-10-03 2019-04-11 Nissan Chemical Corporation Method for producing peptide compound
EP3922638A4 (de) 2019-02-04 2022-11-30 Nissan Chemical Corporation Verfahren zur herstellung einer peptidverbindung

Also Published As

Publication number Publication date
IL92338A0 (en) 1990-07-26
HU896580D0 (en) 1991-08-28
WO1990005738A1 (en) 1990-05-31
FI912411A7 (fi) 1991-05-17
EP0444068A1 (de) 1991-09-04
JPH04502908A (ja) 1992-05-28
GB8827083D0 (en) 1988-12-21
HUT58106A (en) 1992-01-28
FI912411A0 (fi) 1991-05-17
ZA898774B (en) 1990-08-29
AU4517289A (en) 1990-06-12

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Legal Events

Date Code Title Description
FZDE Discontinued