CA2192357A1 - Procede de preparation de 2-(1-azabicyclo[2.2.2.]oct-3-yl)-2,4,5,6-tetrahydro-1h-benz[de]isoquiloeine-1-one et de produit intermediaire - Google Patents

Procede de preparation de 2-(1-azabicyclo[2.2.2.]oct-3-yl)-2,4,5,6-tetrahydro-1h-benz[de]isoquiloeine-1-one et de produit intermediaire

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Publication number
CA2192357A1
CA2192357A1 CA002192357A CA2192357A CA2192357A1 CA 2192357 A1 CA2192357 A1 CA 2192357A1 CA 002192357 A CA002192357 A CA 002192357A CA 2192357 A CA2192357 A CA 2192357A CA 2192357 A1 CA2192357 A1 CA 2192357A1
Authority
CA
Canada
Prior art keywords
formula
compound
converting
acid addition
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002192357A
Other languages
English (en)
Other versions
CA2192357C (fr
Inventor
Charles Alois Dvorak
Bruce Andrew Kowalczyk
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/272,715 external-priority patent/US5567818A/en
Application filed by Individual filed Critical Individual
Publication of CA2192357A1 publication Critical patent/CA2192357A1/fr
Application granted granted Critical
Publication of CA2192357C publication Critical patent/CA2192357C/fr
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA002192357A 1994-07-08 1995-07-01 Procede de preparation de 2-(1-azabicyclo[2.2.2.]oct-3-yl)-2,4,5,6-tetrahydro-1h-benz[de]isoquiloeine-1-one et de produit intermediaire Expired - Lifetime CA2192357C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/272,715 US5567818A (en) 1994-07-08 1994-07-08 Processes for preparing 2-(1-azabicyclo[2.2.2]oct-3-yl)-1H-benz[de] isoquinolin-1-one derivatives and intermediates useful therein
US08/272,715 1994-07-08
PCT/EP1995/002556 WO1996001824A1 (fr) 1994-07-08 1995-07-01 Procede de preparation de 2-(1-azabicyclo[2.2.2.]oct-3-yl)-2,4,5,6-tetrahydro-1h-benz[de]isoquiloeine-1-one et de produit intermediaire

Publications (2)

Publication Number Publication Date
CA2192357A1 true CA2192357A1 (fr) 1996-01-25
CA2192357C CA2192357C (fr) 2006-06-27

Family

ID=36644831

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002192357A Expired - Lifetime CA2192357C (fr) 1994-07-08 1995-07-01 Procede de preparation de 2-(1-azabicyclo[2.2.2.]oct-3-yl)-2,4,5,6-tetrahydro-1h-benz[de]isoquiloeine-1-one et de produit intermediaire

Country Status (1)

Country Link
CA (1) CA2192357C (fr)

Also Published As

Publication number Publication date
CA2192357C (fr) 2006-06-27

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