CA2244621C - 4-amynopyrrole (3,2-d) pyrimidines comme antagonistes des recepteurs du neuropeptide y - Google Patents

4-amynopyrrole (3,2-d) pyrimidines comme antagonistes des recepteurs du neuropeptide y Download PDF

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Publication number: CA2244621C
Authority: CA; Canada
Prior art keywords: medicine; disease; disorder; condition; abnormal
Prior art date: 1997-08-05
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Fee Related

Application number

CA002244621A

Other languages

English (en)

Other versions

CA2244621A1 (fr

Inventor

Robert Lee Dow

Bonnie Frances Tate

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pfizer Products Inc

Original Assignee

Pfizer Products Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-08-05

Filing date

1998-07-31

Publication date

2003-07-29

1998-07-31 Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc

1999-02-05 Publication of CA2244621A1 publication Critical patent/CA2244621A1/fr

2003-07-29 Application granted granted Critical

2003-07-29 Publication of CA2244621C publication Critical patent/CA2244621C/fr

2018-07-31 Anticipated expiration legal-status Critical

Status Expired - Fee Related legal-status Critical Current

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Medicinal Chemistry (AREA)
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Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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Biomedical Technology (AREA)
Neurology (AREA)
Diabetes (AREA)
Endocrinology (AREA)
Heart & Thoracic Surgery (AREA)
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Pain & Pain Management (AREA)
Psychiatry (AREA)
Urology & Nephrology (AREA)
Epidemiology (AREA)
Hematology (AREA)
Obesity (AREA)
Child & Adolescent Psychology (AREA)
Rheumatology (AREA)
Anesthesiology (AREA)
Hospice & Palliative Care (AREA)
Reproductive Health (AREA)
Vascular Medicine (AREA)
Pulmonology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

CA002244621A 1997-08-05 1998-07-31 4-amynopyrrole (3,2-d) pyrimidines comme antagonistes des recepteurs du neuropeptide y Expired - Fee Related CA2244621C (fr)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US5530797P	1997-08-05	1997-08-05
US60/055,307		1997-08-05

Publications (2)

Publication Number	Publication Date
CA2244621A1 CA2244621A1 (fr)	1999-02-05
CA2244621C true CA2244621C (fr)	2003-07-29

Family

ID=21997003

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002244621A Expired - Fee Related CA2244621C (fr)	1997-08-05	1998-07-31	4-amynopyrrole (3,2-d) pyrimidines comme antagonistes des recepteurs du neuropeptide y

Country Status (16)

Country	Link
US (1)	US6040310A (fr)
EP (1)	EP0896822B1 (fr)
JP (1)	JP2978898B2 (fr)
KR (1)	KR19990023355A (fr)
AT (1)	ATE234098T1 (fr)
AU (1)	AU726676B2 (fr)
CA (1)	CA2244621C (fr)
DE (1)	DE69812010T2 (fr)
DK (1)	DK0896822T3 (fr)
ES (1)	ES2191908T3 (fr)
HU (1)	HUP9801792A3 (fr)
IL (1)	IL125591A0 (fr)
NZ (1)	NZ331233A (fr)
PT (1)	PT896822E (fr)
TW (1)	TW434015B (fr)
ZA (1)	ZA986971B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20040254153A1 (en) *	1999-11-08	2004-12-16	Pfizer Inc	Compounds for the treatment of female sexual dysfunction
US20020091129A1 (en) *	2000-11-20	2002-07-11	Mitradev Boolell	Treatment of premature ejaculation
US20030082647A1 (en) *	2000-12-12	2003-05-01	Reenan Robert A.	Transporter protein
EP1399553A2 (fr)	2000-12-12	2004-03-24	The University of Connecticut	Polynucleotides codant pour des transporteurs cellulaires et procedes de leur utilisation
US8377906B2 (en)	2004-06-04	2013-02-19	Ethicon, Inc.	Compositions and methods for preventing or reducing postoperative ileus and gastric stasis
US8129359B2 (en)	2004-06-04	2012-03-06	Ethicon, Inc.	Composition and method for treating post-surgical pain
WO2006108218A1 (fr) *	2005-04-15	2006-10-19	Regenertech Pty Limited	Utilisation de neuropeptides y (npy) et d'agoniste d'antagonistes de ceux-ci pour regenerer des tissus
CN106188060A (zh) *	2015-04-29	2016-12-07	厦门大学	嘧啶并吡咯类化合物、其制备方法、药用组合物及其应用
US10562902B2 (en)	2015-08-13	2020-02-18	Beijing Hanmi Pharmaceutical Co., Ltd.	IRAK4 inhibitor and use thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE69216509T2 (de) *	1991-08-12	1997-05-28	Takeda Chemical Industries Ltd	Kondensierte Pyrimidinderivate, ihre Herstellung und ihre Verwendung als Antitumormittel
US6562862B1 (en) *	1994-10-20	2003-05-13	Eli Lilly And Company	Methods of inhibiting physiological conditions associated with an excess of neuropeptide Y
AU692977B2 (en) *	1994-11-07	1998-06-18	Pfizer Inc.	Certain substituted benzylamine derivatives; a new class of neuropeptide Y1 specific ligands
US5602024A (en) *	1994-12-02	1997-02-11	Synaptic Pharmaceutical Corporation	DNA encoding a hypothalamic atypical neuropeptide Y/peptide YY receptor (Y5) and uses thereof
EP0729758A3 (fr) *	1995-03-02	1997-10-29	Pfizer	Pyrazolopyrimidines et pyrrolopyrimidines pour traiter les troubles neuronaux et autres maladies
EP0759441A3 (fr) *	1995-06-30	1999-06-30	Eli Lilly And Company	Procédés de traitement des pathologies associées aux peptides neuropeptide Y

1998
- 1998-07-27 DK DK98305963T patent/DK0896822T3/da active
- 1998-07-27 AT AT98305963T patent/ATE234098T1/de not_active IP Right Cessation
- 1998-07-27 ES ES98305963T patent/ES2191908T3/es not_active Expired - Lifetime
- 1998-07-27 PT PT98305963T patent/PT896822E/pt unknown
- 1998-07-27 DE DE69812010T patent/DE69812010T2/de not_active Expired - Fee Related
- 1998-07-27 EP EP98305963A patent/EP0896822B1/fr not_active Expired - Lifetime
- 1998-07-29 US US09/124,025 patent/US6040310A/en not_active Expired - Fee Related
- 1998-07-30 IL IL12559198A patent/IL125591A0/xx unknown
- 1998-07-31 CA CA002244621A patent/CA2244621C/fr not_active Expired - Fee Related
- 1998-07-31 TW TW087112649A patent/TW434015B/zh active
- 1998-08-03 AU AU78694/98A patent/AU726676B2/en not_active Ceased
- 1998-08-03 NZ NZ331233A patent/NZ331233A/xx unknown
- 1998-08-04 KR KR1019980031728A patent/KR19990023355A/ko not_active Ceased
- 1998-08-04 JP JP10220638A patent/JP2978898B2/ja not_active Expired - Fee Related
- 1998-08-04 HU HU9801792A patent/HUP9801792A3/hu unknown
- 1998-08-04 ZA ZA9806971A patent/ZA986971B/xx unknown

Also Published As

Publication number	Publication date
HUP9801792A3 (en)	2001-04-28
CA2244621A1 (fr)	1999-02-05
DE69812010D1 (de)	2003-04-17
EP0896822B1 (fr)	2003-03-12
ATE234098T1 (de)	2003-03-15
JPH11130774A (ja)	1999-05-18
HU9801792D0 (en)	1998-09-28
JP2978898B2 (ja)	1999-11-15
EP0896822A1 (fr)	1999-02-17
PT896822E (pt)	2003-07-31
DE69812010T2 (de)	2004-02-26
AU726676B2 (en)	2000-11-16
KR19990023355A (ko)	1999-03-25
AU7869498A (en)	1999-02-18
IL125591A0 (en)	1999-03-12
NZ331233A (en)	2000-09-29
ZA986971B (en)	2000-02-04
TW434015B (en)	2001-05-16
US6040310A (en)	2000-03-21
DK0896822T3 (da)	2003-06-02
ES2191908T3 (es)	2003-09-16
HUP9801792A2 (hu)	2000-02-28

Legal Events

Date	Code	Title	Description
1998-07-31	EEER	Examination request
2006-07-31	MKLA	Lapsed

Publication	Publication Date	Title
EP1003744B1 (fr)	2005-06-01	4-AMINOPYRROLE(3,2-d)PYRIMIDINES EN TANT QU'ANTAGONISTES DU RECEPTEUR DU NEUROPEPTIDE Y
US5985873A (en)	1999-11-16	Certain substituted benzylamine derivatives a new class of Neuropeptide-Y1 specific ligands
CA2244621C (fr)	2003-07-29	4-amynopyrrole (3,2-d) pyrimidines comme antagonistes des recepteurs du neuropeptide y
EP1027891B1 (fr)	2004-12-29	Antagonistes du neuropeptide Y
US6407120B1 (en)	2002-06-18	Neuropeptide Y antagonists
US6511984B2 (en)	2003-01-28	Neuropeptide Y antagonists
JP3717737B2 (ja)	2005-11-16	神経ペプチドｙアンタゴニスト
CZ439199A3 (cs)	2000-07-12	4-Aminopyrrol(3^-d)pyrimidiny jako antagonisty receptoru neuropeptidu Y
MXPA99012095A (es)	2000-09-04	4-aminopirrol (3,2-d) pirimidinas como antagonistas del receptor del neuropeptido y
US20140094512A1 (en)	2014-04-03	Method of modulating the degree of adipose tissue deposited intramuscularly
MXPA00001707A (en)	2001-06-26	Amide derivatives useful as neuropeptide y (npy) antagonists