CA2273884A1 - Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleine - Google Patents

Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleine Download PDF

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Publication number
CA2273884A1
CA2273884A1 CA002273884A CA2273884A CA2273884A1 CA 2273884 A1 CA2273884 A1 CA 2273884A1 CA 002273884 A CA002273884 A CA 002273884A CA 2273884 A CA2273884 A CA 2273884A CA 2273884 A1 CA2273884 A1 CA 2273884A1
Authority
CA
Canada
Prior art keywords
library
formula
hydrogen
compounds
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002273884A
Other languages
English (en)
Inventor
Jose Serafin Mendoza
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2273884A1 publication Critical patent/CA2273884A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Cette invention a trait à une nouvelle banque combinatoire diverse de composés de tétrahydroquinoléine ainsi qu'à un dispositif permettant d'accéder facilement à une source d'individualités de cette banque. Le dispositif peut être utilisé dans des nécessaires à épreuves biologiques en tant qu'élément remplaçable de machines automatiques à épreuves biologiques.
CA002273884A 1996-12-18 1997-12-15 Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleine Abandoned CA2273884A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US3366596P 1996-12-18 1996-12-18
US60/033,665 1996-12-18
PCT/US1997/022870 WO1998027093A1 (fr) 1996-12-18 1997-12-15 Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleine

Publications (1)

Publication Number Publication Date
CA2273884A1 true CA2273884A1 (fr) 1998-06-25

Family

ID=21871728

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002273884A Abandoned CA2273884A1 (fr) 1996-12-18 1997-12-15 Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleine

Country Status (5)

Country Link
EP (1) EP0946556A4 (fr)
JP (1) JP2001508050A (fr)
AU (1) AU5797098A (fr)
CA (1) CA2273884A1 (fr)
WO (1) WO1998027093A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7250423B2 (en) * 2001-09-24 2007-07-31 Chao-Jun Li Methods for synthesizing heterocycles and therapeutic use of the heterocycles for cancers
DE10236910A1 (de) * 2002-08-12 2004-03-11 Grünenthal GmbH Substituierte 1,2,3,4-Tetrahydrochinolinderivate
WO2005016255A2 (fr) * 2003-07-16 2005-02-24 Ligand Pharmaceuticals Incorporated Tetrahydroquinolines a substitution, acides phenylacetiques et benzoiques, comme composes modulateurs de recepteur du facteur nucleaire d'hepatocyte 4$g(a) (hnf-4$g(a) )
DE102004031656A1 (de) * 2004-06-30 2006-01-19 Merck Patent Gmbh Tetrahydrochinoline
DE102005027170A1 (de) * 2005-06-13 2006-12-14 Merck Patent Gmbh Substituierte Tetrahydrochinoline
EP2647638A1 (fr) * 2012-04-02 2013-10-09 Almirall, S.A. Composés tricycliques substitués présentant une activité vis-à-vis des récepteurs ep1

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2650226A (en) * 1950-05-24 1953-08-25 Schenley Ind Inc Furo and thieno quinaldines and process for making same
US2650227A (en) * 1950-05-27 1953-08-25 Schenley Ind Inc Derivatives of 2:3-dihydro-4-methylfuro (3:2-c) quinoline and preparation thereof
US2650229A (en) * 1950-05-27 1953-08-25 Schenley Ind Inc Derivatives of 2:3-dihydro-4-methyltfuro(3:2-c) quinoline and preparation thereof
US3631050A (en) * 1968-11-13 1971-12-28 Parke Davis & Co Hexahydro-9b-methylfuro(3 2-c) quinoline compounds
US3632852A (en) * 1969-03-17 1972-01-04 Parke Davis & Co Hexahydrobenzofurofuro(3 2-c) quinoline compounds
KR100310939B1 (ko) * 1992-10-01 2002-06-20 추후제출 태그로암호화한복합조합화학라이브러리

Also Published As

Publication number Publication date
WO1998027093A1 (fr) 1998-06-25
EP0946556A4 (fr) 2001-07-04
AU5797098A (en) 1998-07-15
JP2001508050A (ja) 2001-06-19
EP0946556A1 (fr) 1999-10-06

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Legal Events

Date Code Title Description
FZDE Discontinued