CA2336152A1 - Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire - Google Patents

Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire Download PDF

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Publication number
CA2336152A1
CA2336152A1 CA002336152A CA2336152A CA2336152A1 CA 2336152 A1 CA2336152 A1 CA 2336152A1 CA 002336152 A CA002336152 A CA 002336152A CA 2336152 A CA2336152 A CA 2336152A CA 2336152 A1 CA2336152 A1 CA 2336152A1
Authority
CA
Canada
Prior art keywords
disorders
vision
straight
branched chain
eye
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002336152A
Other languages
English (en)
Inventor
Douglas T. Ross
Hansjorg Sauer
Gregory S. Hamilton
Joseph P. Steiner
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GPI Nil Holdings Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2336152A1 publication Critical patent/CA2336152A1/fr
Abandoned legal-status Critical Current

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/401Proline; Derivatives thereof, e.g. captopril
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)

Abstract

L'invention concerne des nouvelles compositions, ainsi que des utilisations d'une urée ou d'un carbamate d'un acide carboxylique N-hétérocyclique, ou d'un isostère de celui-ci, pour traiter un trouble de la vision, améliorer la vision, ou traiter des défauts de mémoire ou améliorer les performances de celle-ci, chez un animal.
CA002336152A 1998-08-14 1999-08-12 Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire Abandoned CA2336152A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US13442098A 1998-08-14 1998-08-14
US09/134,420 1998-08-14
PCT/US1999/018234 WO2000009125A1 (fr) 1998-08-14 1999-08-12 Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire

Publications (1)

Publication Number Publication Date
CA2336152A1 true CA2336152A1 (fr) 2000-02-24

Family

ID=22463316

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002336152A Abandoned CA2336152A1 (fr) 1998-08-14 1999-08-12 Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire

Country Status (6)

Country Link
EP (1) EP1107754A1 (fr)
JP (1) JP2002522494A (fr)
AU (1) AU5477899A (fr)
CA (1) CA2336152A1 (fr)
MX (1) MXPA00013031A (fr)
WO (1) WO2000009125A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009020140A1 (fr) * 2007-08-06 2009-02-12 Dainippon Sumitomo Pharma Co., Ltd. Dérivé d'adamantylurée
EP2822931B1 (fr) 2012-03-09 2017-05-03 Inception 2, Inc. Composés de triazolone et leurs utilisations
SG11201504622PA (en) 2012-12-20 2015-07-30 Inception 2 Inc Triazolone compounds and uses thereof
CN105579440A (zh) 2013-09-06 2016-05-11 因森普深2公司 三唑酮化合物及其应用
WO2023090853A1 (fr) * 2021-11-19 2023-05-25 고려대학교 세종산학협력단 Nouvel antagoniste du récepteur p2x7 à base d'urée ou de carbamate, et composition pharmaceutique pour la prévention ou le traitement d'un trouble dépressif majeur, comprenant celui-ci en tant que principe actif

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0670309A1 (fr) * 1992-11-20 1995-09-06 Japan Tobacco Inc. Compose inhibant la prolyle endopeptidase et utilisation pharmaceutique de ce dernier

Also Published As

Publication number Publication date
WO2000009125A1 (fr) 2000-02-24
JP2002522494A (ja) 2002-07-23
EP1107754A1 (fr) 2001-06-20
AU5477899A (en) 2000-03-06
MXPA00013031A (es) 2002-04-24

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Legal Events

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