CA2336152A1 - Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire - Google Patents
Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire Download PDFInfo
- Publication number
- CA2336152A1 CA2336152A1 CA002336152A CA2336152A CA2336152A1 CA 2336152 A1 CA2336152 A1 CA 2336152A1 CA 002336152 A CA002336152 A CA 002336152A CA 2336152 A CA2336152 A CA 2336152A CA 2336152 A1 CA2336152 A1 CA 2336152A1
- Authority
- CA
- Canada
- Prior art keywords
- disorders
- vision
- straight
- branched chain
- eye
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/401—Proline; Derivatives thereof, e.g. captopril
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Ophthalmology & Optometry (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
Abstract
L'invention concerne des nouvelles compositions, ainsi que des utilisations d'une urée ou d'un carbamate d'un acide carboxylique N-hétérocyclique, ou d'un isostère de celui-ci, pour traiter un trouble de la vision, améliorer la vision, ou traiter des défauts de mémoire ou améliorer les performances de celle-ci, chez un animal.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13442098A | 1998-08-14 | 1998-08-14 | |
| US09/134,420 | 1998-08-14 | ||
| PCT/US1999/018234 WO2000009125A1 (fr) | 1998-08-14 | 1999-08-12 | Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2336152A1 true CA2336152A1 (fr) | 2000-02-24 |
Family
ID=22463316
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002336152A Abandoned CA2336152A1 (fr) | 1998-08-14 | 1999-08-12 | Urees et carbamates d'acides carboxyliques n-heterocycliques et isosteres destines a des troubles de la vision et de la memoire |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP1107754A1 (fr) |
| JP (1) | JP2002522494A (fr) |
| AU (1) | AU5477899A (fr) |
| CA (1) | CA2336152A1 (fr) |
| MX (1) | MXPA00013031A (fr) |
| WO (1) | WO2000009125A1 (fr) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009020140A1 (fr) * | 2007-08-06 | 2009-02-12 | Dainippon Sumitomo Pharma Co., Ltd. | Dérivé d'adamantylurée |
| EP2822931B1 (fr) | 2012-03-09 | 2017-05-03 | Inception 2, Inc. | Composés de triazolone et leurs utilisations |
| SG11201504622PA (en) | 2012-12-20 | 2015-07-30 | Inception 2 Inc | Triazolone compounds and uses thereof |
| CN105579440A (zh) | 2013-09-06 | 2016-05-11 | 因森普深2公司 | 三唑酮化合物及其应用 |
| WO2023090853A1 (fr) * | 2021-11-19 | 2023-05-25 | 고려대학교 세종산학협력단 | Nouvel antagoniste du récepteur p2x7 à base d'urée ou de carbamate, et composition pharmaceutique pour la prévention ou le traitement d'un trouble dépressif majeur, comprenant celui-ci en tant que principe actif |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0670309A1 (fr) * | 1992-11-20 | 1995-09-06 | Japan Tobacco Inc. | Compose inhibant la prolyle endopeptidase et utilisation pharmaceutique de ce dernier |
-
1999
- 1999-08-12 CA CA002336152A patent/CA2336152A1/fr not_active Abandoned
- 1999-08-12 JP JP2000564628A patent/JP2002522494A/ja active Pending
- 1999-08-12 WO PCT/US1999/018234 patent/WO2000009125A1/fr not_active Ceased
- 1999-08-12 MX MXPA00013031A patent/MXPA00013031A/es unknown
- 1999-08-12 EP EP99941054A patent/EP1107754A1/fr not_active Withdrawn
- 1999-08-12 AU AU54778/99A patent/AU5477899A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2000009125A1 (fr) | 2000-02-24 |
| JP2002522494A (ja) | 2002-07-23 |
| EP1107754A1 (fr) | 2001-06-20 |
| AU5477899A (en) | 2000-03-06 |
| MXPA00013031A (es) | 2002-04-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Dead |