CA2433183A1 - Composes et utilisations associees - Google Patents

Composes et utilisations associees Download PDF

Info

Publication number
CA2433183A1
CA2433183A1 CA002433183A CA2433183A CA2433183A1 CA 2433183 A1 CA2433183 A1 CA 2433183A1 CA 002433183 A CA002433183 A CA 002433183A CA 2433183 A CA2433183 A CA 2433183A CA 2433183 A1 CA2433183 A1 CA 2433183A1
Authority
CA
Canada
Prior art keywords
inositol
deoxy
amino
glucopyranosyl
alpha
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002433183A
Other languages
English (en)
Inventor
Manuel Martin-Lomas
Thomas William Rademacher
Hugo Norbert Caro
Irene Francois
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Rodaris Pharmaceuticals Ltd
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0011594A external-priority patent/GB0011594D0/en
Priority claimed from US09/798,005 external-priority patent/US6953781B2/en
Application filed by Individual filed Critical Individual
Publication of CA2433183A1 publication Critical patent/CA2433183A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Endocrinology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne des composés possédant une propriété antagoniste ou mimétique d'un inositolphosphoglycanne (IPG), ainsi que l'utilisation de ces composés, de même que l'emploi de ceux-ci, par exemple pour traiter un état amélioré par l'administration d'un second messager IPG ou d'un antagoniste IPG de celui-ci. L'invention concerne notamment des composés comportant une liaison 1,6 d'un reste sucre et d'un cyclitol.
CA002433183A 2000-05-12 2001-05-11 Composes et utilisations associees Abandoned CA2433183A1 (fr)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US20359600P 2000-05-12 2000-05-12
US60/203,596 2000-05-12
GB0011594.9 2000-05-12
GB0011594A GB0011594D0 (en) 2000-05-12 2000-05-12 Compounds and their uses
US09/798,005 2001-03-02
US09/798,005 US6953781B2 (en) 2000-05-12 2001-03-02 Compounds and their uses
PCT/GB2001/002088 WO2001085740A2 (fr) 2000-05-12 2001-05-11 Composes et utilisations associees

Publications (1)

Publication Number Publication Date
CA2433183A1 true CA2433183A1 (fr) 2001-11-15

Family

ID=27255717

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002433183A Abandoned CA2433183A1 (fr) 2000-05-12 2001-05-11 Composes et utilisations associees

Country Status (4)

Country Link
EP (1) EP1406913A2 (fr)
AU (1) AU6042601A (fr)
CA (1) CA2433183A1 (fr)
WO (1) WO2001085740A2 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2878850B1 (fr) 2004-12-02 2008-10-31 Cis Bio Internat Sa Derives de l'inositol-1-phosphate
WO2008080064A1 (fr) * 2006-12-21 2008-07-03 Trustees Of Tufts College Glycanes inositol lipophiles synthétiques pour traiter le cancer et des troubles du métabolisme du glucose

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19649350A1 (de) * 1996-11-28 1998-06-04 Hoechst Ag Inositolglykane mit insulinartiger Wirkung

Also Published As

Publication number Publication date
AU6042601A (en) 2001-11-20
EP1406913A2 (fr) 2004-04-14
WO2001085740A2 (fr) 2001-11-15
WO2001085740A3 (fr) 2002-03-28

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Dead