CA2447178C - Composition pharmaceutique a utiliser en therapie de remplacement d'hormones - Google Patents
Composition pharmaceutique a utiliser en therapie de remplacement d'hormones Download PDFInfo
- Publication number
- CA2447178C CA2447178C CA2447178A CA2447178A CA2447178C CA 2447178 C CA2447178 C CA 2447178C CA 2447178 A CA2447178 A CA 2447178A CA 2447178 A CA2447178 A CA 2447178A CA 2447178 C CA2447178 C CA 2447178C
- Authority
- CA
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- Prior art keywords
- estrogenic
- day
- estrogenic component
- use according
- administration
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
Abstract
L'invention concerne, dans un mode de réalisation, un procédé de thérapie de remplacement d'hormones. Ledit procédé consiste à administrer à une personne nécessitant une telle thérapie une dose efficace d'un composant oestrogénique choisi dans le groupe comprenant des substances représentées par la formule suivante (I), dans laquelle R¿1?, R¿2?, R¿3?, R¿4? représentent individuellement un atome d'hydrogène, un groupe hydroxyle ou un groupe alcoxy avec 1-5 atomes de carbone; chacun des R¿5?, R¿6?, R¿7? représente un groupe hydroxyle; et 3 au maximum de R¿1?, R¿2?, R¿3?, R¿4? représentent des atomes d'hydrogène; des précurseurs pouvant libérer une substance suivant la formule susmentionnée lorsqu'elle est utilisée dans ledit procédé, et des mélanges de ceux-ci. Ladite composition ne contient pratiquement pas de progestogène ni d'anti-progestine. Dans un autre mode de réalisation, l'invention concerne un système d'administration de médicaments conçu pour une administration entérale ou parentérale contenant au moins 1 µg du composant oestrogénique et ne contenant ni progestogène, ni anti-progestine.
Applications Claiming Priority (15)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01201896A EP1260225A1 (fr) | 2001-05-18 | 2001-05-18 | Compositions pharmaceutiques pour le traitement hormonal substitutif |
| EP01201896.6 | 2001-05-18 | ||
| EP01201946.9 | 2001-05-23 | ||
| EP01201947.7 | 2001-05-23 | ||
| EP01201947 | 2001-05-23 | ||
| EP01201946 | 2001-05-23 | ||
| EP01201945A EP1293210B1 (fr) | 2001-05-23 | 2001-05-23 | Kit et méthode contraceptive hormonale |
| EP01201945.1 | 2001-05-23 | ||
| EP01203305A EP1287817A1 (fr) | 2001-08-31 | 2001-08-31 | Méthode et dispositif intravaginal pour le traitement des myomes utérins |
| EP01203305.6 | 2001-08-31 | ||
| EP01204377.4 | 2001-11-15 | ||
| EP01204377 | 2001-11-15 | ||
| EP02075695.3 | 2002-02-21 | ||
| EP02075695 | 2002-02-21 | ||
| PCT/NL2002/000317 WO2002094276A1 (fr) | 2001-05-18 | 2002-05-17 | Composition pharmaceutique a utiliser en therapie de remplacement d'hormones |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2447178A1 CA2447178A1 (fr) | 2002-11-28 |
| CA2447178C true CA2447178C (fr) | 2010-06-08 |
Family
ID=27561854
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2447178A Expired - Lifetime CA2447178C (fr) | 2001-05-18 | 2002-05-17 | Composition pharmaceutique a utiliser en therapie de remplacement d'hormones |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8048869B2 (fr) |
| EP (1) | EP1390040B1 (fr) |
| AT (1) | ATE350041T1 (fr) |
| CA (1) | CA2447178C (fr) |
| CY (1) | CY1106457T1 (fr) |
| DE (1) | DE60217324T2 (fr) |
| DK (1) | DK1390040T3 (fr) |
| ES (1) | ES2278924T3 (fr) |
| PT (1) | PT1390040E (fr) |
| WO (1) | WO2002094276A1 (fr) |
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| KR102712911B1 (ko) | 2016-08-05 | 2024-10-04 | 에스테트라, 소시에떼 아 레스폰서빌리떼 리미떼 | 월경통 및 생리통의 관리방법 |
| SG11202009725XA (en) | 2018-04-19 | 2020-11-27 | Estetra Sprl | Compounds and their uses for alleviating menopause-associated symptoms |
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-
2002
- 2002-05-17 AT AT02738951T patent/ATE350041T1/de active
- 2002-05-17 DK DK02738951T patent/DK1390040T3/da active
- 2002-05-17 WO PCT/NL2002/000317 patent/WO2002094276A1/fr not_active Ceased
- 2002-05-17 DE DE60217324T patent/DE60217324T2/de not_active Expired - Lifetime
- 2002-05-17 CA CA2447178A patent/CA2447178C/fr not_active Expired - Lifetime
- 2002-05-17 PT PT02738951T patent/PT1390040E/pt unknown
- 2002-05-17 ES ES02738951T patent/ES2278924T3/es not_active Expired - Lifetime
- 2002-05-17 US US10/478,262 patent/US8048869B2/en not_active Expired - Lifetime
- 2002-05-17 EP EP02738951A patent/EP1390040B1/fr not_active Expired - Lifetime
-
2007
- 2007-03-22 CY CY20071100403T patent/CY1106457T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ATE350041T1 (de) | 2007-01-15 |
| US8048869B2 (en) | 2011-11-01 |
| EP1390040B1 (fr) | 2007-01-03 |
| PT1390040E (pt) | 2007-04-30 |
| US20040198671A1 (en) | 2004-10-07 |
| EP1390040A1 (fr) | 2004-02-25 |
| ES2278924T3 (es) | 2007-08-16 |
| DK1390040T3 (da) | 2007-04-23 |
| CA2447178A1 (fr) | 2002-11-28 |
| CY1106457T1 (el) | 2011-10-12 |
| DE60217324D1 (de) | 2007-02-15 |
| DE60217324T2 (de) | 2007-04-26 |
| WO2002094276A1 (fr) | 2002-11-28 |
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| EEER | Examination request | ||
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Effective date: 20220517 |