CA2477832A1 - Methods of treating diabetes using pde 11a inhibitors - Google Patents

Methods of treating diabetes using pde 11a inhibitors Download PDF

Info

Publication number: CA2477832A1
Authority: CA; Canada
Prior art keywords: inhibitor; diabetes; pde11a; insulin; administering
Prior art date: 2002-03-14
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA002477832A

Other languages

English (en)

French (fr)

Inventor

Haren Vasavada

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bayer Pharmaceuticals Corp

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-03-14

Filing date

2003-03-14

Publication date

2003-09-25

2003-03-14 Application filed by Individual filed Critical Individual

2003-09-25 Publication of CA2477832A1 publication Critical patent/CA2477832A1/en

Status Abandoned legal-status Critical Current

Links

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Health & Medical Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
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General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Epidemiology (AREA)
Urology & Nephrology (AREA)
Reproductive Health (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Gynecology & Obstetrics (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Hospice & Palliative Care (AREA)
Vascular Medicine (AREA)
Psychiatry (AREA)
Hematology (AREA)
Emergency Medicine (AREA)
Pulmonology (AREA)
Pregnancy & Childbirth (AREA)
Obesity (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

CA002477832A 2002-03-14 2003-03-14 Methods of treating diabetes using pde 11a inhibitors Abandoned CA2477832A1 (en)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
US36469702P	2002-03-14	2002-03-14
US60/364,697		2002-03-14
US38903602P	2002-06-13	2002-06-13
US60/389,036		2002-06-13
PCT/US2003/008132 WO2003077949A2 (en)	2002-03-14	2003-03-14	Methods of treating diabetes using pde 11a inhibitors

Publications (1)

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CA2477832A1 true CA2477832A1 (en)	2003-09-25

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CA002477832A Abandoned CA2477832A1 (en)	2002-03-14	2003-03-14	Methods of treating diabetes using pde 11a inhibitors

Country Status (7)

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EP (1)	EP1496940A2 (de)
JP (1)	JP2005527524A (de)
AU (1)	AU2003220342B2 (de)
BR (1)	BR0308415A (de)
CA (1)	CA2477832A1 (de)
MX (1)	MXPA04008195A (de)
WO (1)	WO2003077949A2 (de)

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JP2008502909A (ja) *	2004-06-15	2008-01-31	メタボレックスインコーポレーティッド	糖尿病およびインスリン抵抗性の診断および治療の方法
MEP8509A (en)	2006-09-07	2011-12-20		Combination treatment for diabetes mellitus
KR101560844B1 (ko)	2007-06-04	2015-10-15	벤-구리온 유니버시티 오브 더 네게브 리서치 앤드 디벨럽먼트 어쏘러티	트라이-아릴계 화합물 및 이를 포함하는 조성물
EP3199203B1 (de)	2008-02-29	2020-02-05	Concert Pharmaceuticals Inc.	Substituierte xanthinderivate
US20110053961A1 (en)	2009-02-27	2011-03-03	Concert Pharmaceuticals, Inc.	Substituted xanthine derivatives
JP2012520342A (ja) *	2009-03-16	2012-09-06	ジェンメディカ・セラピューティックス・ソシエダッド・リミターダ	代謝障害を処置するのに有用な抗炎症剤および抗酸化剤のコンジュゲート
WO2013013052A1 (en)	2011-07-19	2013-01-24	Concert Pharmaceuticals, Inc.	Substituted xanthine derivatives
JP2015067538A (ja) *	2013-09-26	2015-04-13	株式会社アイエイアイ	血糖値降下剤
CN106061940A (zh)	2013-11-05	2016-10-26	本古里安大学内盖夫研究发展局	治疗糖尿病和由其引发的并发疾病的化合物
WO2015160913A1 (en)	2014-04-18	2015-10-22	Concert Pharmaceuticals, Inc.	Methods of treating hyperglycemia

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US6414002B1 (en) *	1999-09-22	2002-07-02	Bristol-Myers Squibb Company	Substituted acid derivatives useful as antidiabetic and antiobesity agents and method
EP1297115A2 (de) *	2000-06-26	2003-04-02	Bayer Aktiengesellschaft	Regulation eines menschlichen phosphodiesterase-ähnlichen enzyms
EP1211313A3 (de) *	2000-11-01	2003-04-23	Pfizer Limited	Modulation der PDE11A-AKtivität

2003
- 2003-03-14 MX MXPA04008195A patent/MXPA04008195A/es not_active Application Discontinuation
- 2003-03-14 BR BR0308415-9A patent/BR0308415A/pt not_active IP Right Cessation
- 2003-03-14 AU AU2003220342A patent/AU2003220342B2/en not_active Expired - Fee Related
- 2003-03-14 WO PCT/US2003/008132 patent/WO2003077949A2/en not_active Ceased
- 2003-03-14 CA CA002477832A patent/CA2477832A1/en not_active Abandoned
- 2003-03-14 JP JP2003576002A patent/JP2005527524A/ja not_active Withdrawn
- 2003-03-14 EP EP03716641A patent/EP1496940A2/de not_active Withdrawn

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Publication number	Publication date
WO2003077949A2 (en)	2003-09-25
WO2003077949A3 (en)	2004-03-25
AU2003220342B2 (en)	2007-06-07
AU2003220342A1 (en)	2003-09-29
EP1496940A2 (de)	2005-01-19
BR0308415A (pt)	2005-02-15
MXPA04008195A (es)	2004-11-26
JP2005527524A (ja)	2005-09-15

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US20070032404A1 (en)	2007-02-08	Methods for treating diabetes and related disorders using pde10a inhibitors
Gilligan et al.	2000	Corticotropin releasing factor (CRF) receptor modulators: progress and opportunities for new therapeutic agents
Morelli et al.	1994	Adenosine A2 receptors interact negatively with dopamine D1 and D2 receptors in unilaterally 6-hydroxydopamine-lesioned rats
AU2003220342B2 (en)	2007-06-07	Methods of treating diabetes using PDE 11A inhibitors
Allescher et al.	1996	Regulation of VIP release from rat enteric nerve terminals: evidence for a stimulatory effect of NO
Shpakov et al.	2006	Functional defects in adenylyl cyclase signaling mechanisms of insulin and relaxin in skeletal muscles of rat with streptozotocin type 1 diabetes
US20060074094A1 (en)	2006-04-06	Use of c-Src inhibitors alone or in combination with STI571 for the treatment of leukaemia
WO2002034242A2 (en)	2002-05-02	Method for the treatment of neurological and neuropsychological disorders
US20120157441A1 (en)	2012-06-21	Inhibitors of the mutant form of kit
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JP2008220373A (ja)	2008-09-25	プロテインキナーゼｃイプシロンを欠如する細胞及び動物
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CN1697661A (zh)	2005-11-16	用pde11a抑制剂治疗糖尿病的方法
HK1085392A (en)	2006-08-25	Methods of treating diabetes using pde 11a inhibitors
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