CA2586845A1 - Traitement therapeutique de resorption osseuse acceleree - Google Patents
Traitement therapeutique de resorption osseuse acceleree Download PDFInfo
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- CA2586845A1 CA2586845A1 CA002586845A CA2586845A CA2586845A1 CA 2586845 A1 CA2586845 A1 CA 2586845A1 CA 002586845 A CA002586845 A CA 002586845A CA 2586845 A CA2586845 A CA 2586845A CA 2586845 A1 CA2586845 A1 CA 2586845A1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Physical Education & Sports Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'invention concerne l'utilisation d'un agoniste du récepteur d'adénosine A3 (agoniste de A3AR) pour le traitement de la résorption osseuse accélérée, plus particulièrement de la résorption osseuse induite par une inflammation. Plus spécifiquement, l'invention concerne un procédé et une composition pharmaceutique pour le traitement de cet état pathologique, l'agoniste de A3AR étant formulé en tant que composition pharmaceutique administrée à un sujet souffrant de résorption osseuse accélérée. L'invention concerne également l'utilisation de l'agoniste de A3AR dans la préparation de cette composition pharmaceutique.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US62556404P | 2004-11-08 | 2004-11-08 | |
| US60/625,564 | 2004-11-08 | ||
| PCT/IL2005/001166 WO2006048884A1 (fr) | 2004-11-08 | 2005-11-08 | Traitement therapeutique de resorption osseuse acceleree |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2586845A1 true CA2586845A1 (fr) | 2006-05-11 |
Family
ID=36001028
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002586845A Abandoned CA2586845A1 (fr) | 2004-11-08 | 2005-11-08 | Traitement therapeutique de resorption osseuse acceleree |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1811982A1 (fr) |
| JP (1) | JP2008519029A (fr) |
| KR (1) | KR20070085839A (fr) |
| CN (1) | CN101072554A (fr) |
| AU (1) | AU2005302090A1 (fr) |
| BR (1) | BRPI0517639A (fr) |
| CA (1) | CA2586845A1 (fr) |
| MX (1) | MX2007005525A (fr) |
| WO (1) | WO2006048884A1 (fr) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5339916B2 (ja) * | 2005-11-30 | 2013-11-13 | キャン−ファイト・バイオファーマ・リミテッド | 骨関節炎の治療におけるa3アデノシン受容体アゴニストの使用 |
| US9102698B2 (en) | 2007-03-14 | 2015-08-11 | Can-Fite Biopharma Ltd. | Process for the synthesis of IB-MECA |
| WO2009061516A1 (fr) * | 2007-11-08 | 2009-05-14 | New York University School Of Medicine | Implants médicaux contenant des agonistes du récepteur de l'adénosine et procédés pour inhiber un relâchement d'implant médical |
| JP5849044B2 (ja) * | 2009-05-17 | 2016-01-27 | キャン−ファイト バイオファーマ リミテッド | 眼圧低下のためのa3アデノシン受容体作動薬 |
| UA117095C2 (uk) | 2011-12-22 | 2018-06-25 | Аліос Біофарма, Інк. | Нуклеозидна сполука або її фармацевтично прийнятна сіль |
| US9441007B2 (en) | 2012-03-21 | 2016-09-13 | Alios Biopharma, Inc. | Substituted nucleosides, nucleotides and analogs thereof |
| USRE48171E1 (en) | 2012-03-21 | 2020-08-25 | Janssen Biopharma, Inc. | Substituted nucleosides, nucleotides and analogs thereof |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU5294100A (en) * | 1999-05-27 | 2000-12-18 | University Of Virginia Patent Foundation | Method and compositions for treating the inflammatory response |
| IL133680A0 (en) * | 1999-09-10 | 2001-04-30 | Can Fite Technologies Ltd | Pharmaceutical compositions comprising an adenosine receptor agonist or antagonist |
| US7141553B2 (en) * | 2002-11-19 | 2006-11-28 | Can-Fite Biopharma Ltd. Israel | A3AR agonists for the treatment of inflammatory arthritis |
| GB0305150D0 (en) * | 2003-03-07 | 2003-04-09 | Cambridge Biotechnology Ltd | Use of therapeutic compounds |
| CA2557285A1 (fr) * | 2004-03-05 | 2005-09-15 | Cambridge Biotechnology Limited | Composes therapeutiques |
-
2005
- 2005-11-08 JP JP2007539712A patent/JP2008519029A/ja not_active Withdrawn
- 2005-11-08 WO PCT/IL2005/001166 patent/WO2006048884A1/fr not_active Ceased
- 2005-11-08 CN CNA2005800380014A patent/CN101072554A/zh active Pending
- 2005-11-08 CA CA002586845A patent/CA2586845A1/fr not_active Abandoned
- 2005-11-08 EP EP05799989A patent/EP1811982A1/fr not_active Withdrawn
- 2005-11-08 BR BRPI0517639-5A patent/BRPI0517639A/pt not_active IP Right Cessation
- 2005-11-08 KR KR1020077012806A patent/KR20070085839A/ko not_active Ceased
- 2005-11-08 MX MX2007005525A patent/MX2007005525A/es not_active Application Discontinuation
- 2005-11-08 AU AU2005302090A patent/AU2005302090A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR20070085839A (ko) | 2007-08-27 |
| BRPI0517639A (pt) | 2008-10-14 |
| WO2006048884A1 (fr) | 2006-05-11 |
| CN101072554A (zh) | 2007-11-14 |
| JP2008519029A (ja) | 2008-06-05 |
| AU2005302090A1 (en) | 2006-05-11 |
| MX2007005525A (es) | 2007-07-05 |
| EP1811982A1 (fr) | 2007-08-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued | ||
| FZDE | Discontinued |
Effective date: 20101108 |