CA2683209A1 - Pyramidinones comme modulateurs de caseine kinase ii (ck2) - Google Patents

Pyramidinones comme modulateurs de caseine kinase ii (ck2) Download PDF

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Publication number
CA2683209A1
CA2683209A1 CA002683209A CA2683209A CA2683209A1 CA 2683209 A1 CA2683209 A1 CA 2683209A1 CA 002683209 A CA002683209 A CA 002683209A CA 2683209 A CA2683209 A CA 2683209A CA 2683209 A1 CA2683209 A1 CA 2683209A1
Authority
CA
Canada
Prior art keywords
alkyl
phenyl
pyrimidin
indazol
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002683209A
Other languages
English (en)
Inventor
Elena S. Koltun
Patrick Kearney
Naing Aay
Arlyn Arcalas
Wai Ki Vicky Chan
Jeffry Kimo Curtis
Hongwang Du
Ping Huang
Brian Kane
Moon Hwan Kim
Michael Pack
Amy L. Tsuhako
Wei Xu
Cristiana A. Zaharia
Peiwen Zhou
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Exelixis Inc
Original Assignee
Exelixis Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Exelixis Inc filed Critical Exelixis Inc
Priority claimed from PCT/US2008/005419 external-priority patent/WO2008143759A1/fr
Publication of CA2683209A1 publication Critical patent/CA2683209A1/fr
Abandoned legal-status Critical Current

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

L'invention concerne un composé ayant la formule I : ou un sel pharmaceutiquement acceptable de celui-ci, dans laquelle X, R, R et R sont tels que définis dans la description ; les compositions pharmaceutiques de celui-ci et des procédés d'utilisation de celui-ci. Les composés de la formule I sont des inhibiteurs des voies de la caséine kinase II (CK2).
CA002683209A 2008-04-24 2008-04-24 Pyramidinones comme modulateurs de caseine kinase ii (ck2) Abandoned CA2683209A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2008/005419 WO2008143759A1 (fr) 2007-04-25 2008-04-24 Pyrimidones en tant que modulateurs de la caséine kinase ii (ck2)

Publications (1)

Publication Number Publication Date
CA2683209A1 true CA2683209A1 (fr) 2009-10-24

Family

ID=41412778

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002683209A Abandoned CA2683209A1 (fr) 2008-04-24 2008-04-24 Pyramidinones comme modulateurs de caseine kinase ii (ck2)

Country Status (1)

Country Link
CA (1) CA2683209A1 (fr)

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Legal Events

Date Code Title Description
EEER Examination request

Effective date: 20130412

FZDE Discontinued

Effective date: 20150716