CA2817336A1 - Succinate de solifenacine cristallin - Google Patents

Succinate de solifenacine cristallin Download PDF

Info

Publication number
CA2817336A1
CA2817336A1 CA2817336A CA2817336A CA2817336A1 CA 2817336 A1 CA2817336 A1 CA 2817336A1 CA 2817336 A CA2817336 A CA 2817336A CA 2817336 A CA2817336 A CA 2817336A CA 2817336 A1 CA2817336 A1 CA 2817336A1
Authority
CA
Canada
Prior art keywords
solifenacin succinate
crystalline
succinate
axial ratio
particle size
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2817336A
Other languages
English (en)
Inventor
Max Born
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hexal AG
Original Assignee
Hexal AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hexal AG filed Critical Hexal AG
Publication of CA2817336A1 publication Critical patent/CA2817336A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Urology & Nephrology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CA2817336A 2010-11-11 2011-11-11 Succinate de solifenacine cristallin Abandoned CA2817336A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10014527 2010-11-11
EP10014527.5 2010-11-11
PCT/EP2011/069969 WO2012062916A1 (fr) 2010-11-11 2011-11-11 Succinate de solifénacine cristallin

Publications (1)

Publication Number Publication Date
CA2817336A1 true CA2817336A1 (fr) 2012-05-18

Family

ID=43663592

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2817336A Abandoned CA2817336A1 (fr) 2010-11-11 2011-11-11 Succinate de solifenacine cristallin

Country Status (3)

Country Link
EP (1) EP2638039A1 (fr)
CA (1) CA2817336A1 (fr)
WO (1) WO2012062916A1 (fr)

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO2005012I1 (no) 1994-12-28 2005-06-06 Debio Rech Pharma Sa Triptorelin og farmasoytisk akseptable salter derav
US20080287680A1 (en) 2004-02-09 2008-11-20 Astellas Pharma Inc. Solifenacin Succinate-Containing Composition
WO2005087231A1 (fr) 2004-03-16 2005-09-22 Astellas Pharma Inc. Composition contenant de la solifenacine
US20080103171A1 (en) 2004-12-27 2008-05-01 Astellas Pharma Inc. Stable Particular Pharmaceutical Composition of Solifenacin or Salt Thereof
US20080114028A1 (en) 2006-07-24 2008-05-15 Tamas Koltai Process for preparing polymorphic forms of solifenacin succinate
JP2010523539A (ja) 2007-03-30 2010-07-15 メディチェム ソシエダ アノニマ ソリフェナシンの改良された合成法
JP2009538362A (ja) 2007-07-13 2009-11-05 テバ ファーマシューティカル インダストリーズ リミティド ソリフェナシンの調製方法
ITMI20080195A1 (it) 2008-02-08 2009-08-09 Dipharma Francis Srl Procedimento per la preparazione di solifenacin
WO2009139002A2 (fr) 2008-05-12 2009-11-19 Msn Laboratories Limited Procédé perfectionné de fabrication de solifénacine et de ses sels pharmaceutiquement acceptables
PL3067353T3 (pl) * 2008-07-29 2018-04-30 Krka, D.D., Novo Mesto Sposób wytwarzania soli solifenacyny i ich włączenie do farmaceutycznych postaci dawkowania

Also Published As

Publication number Publication date
WO2012062916A1 (fr) 2012-05-18
EP2638039A1 (fr) 2013-09-18

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Effective date: 20161114