CA2817336A1 - Succinate de solifenacine cristallin - Google Patents
Succinate de solifenacine cristallin Download PDFInfo
- Publication number
- CA2817336A1 CA2817336A1 CA2817336A CA2817336A CA2817336A1 CA 2817336 A1 CA2817336 A1 CA 2817336A1 CA 2817336 A CA2817336 A CA 2817336A CA 2817336 A CA2817336 A CA 2817336A CA 2817336 A1 CA2817336 A1 CA 2817336A1
- Authority
- CA
- Canada
- Prior art keywords
- solifenacin succinate
- crystalline
- succinate
- axial ratio
- particle size
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Urology & Nephrology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10014527 | 2010-11-11 | ||
| EP10014527.5 | 2010-11-11 | ||
| PCT/EP2011/069969 WO2012062916A1 (fr) | 2010-11-11 | 2011-11-11 | Succinate de solifénacine cristallin |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2817336A1 true CA2817336A1 (fr) | 2012-05-18 |
Family
ID=43663592
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2817336A Abandoned CA2817336A1 (fr) | 2010-11-11 | 2011-11-11 | Succinate de solifenacine cristallin |
Country Status (3)
| Country | Link |
|---|---|
| EP (1) | EP2638039A1 (fr) |
| CA (1) | CA2817336A1 (fr) |
| WO (1) | WO2012062916A1 (fr) |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO2005012I1 (no) | 1994-12-28 | 2005-06-06 | Debio Rech Pharma Sa | Triptorelin og farmasoytisk akseptable salter derav |
| US20080287680A1 (en) | 2004-02-09 | 2008-11-20 | Astellas Pharma Inc. | Solifenacin Succinate-Containing Composition |
| WO2005087231A1 (fr) | 2004-03-16 | 2005-09-22 | Astellas Pharma Inc. | Composition contenant de la solifenacine |
| US20080103171A1 (en) | 2004-12-27 | 2008-05-01 | Astellas Pharma Inc. | Stable Particular Pharmaceutical Composition of Solifenacin or Salt Thereof |
| US20080114028A1 (en) | 2006-07-24 | 2008-05-15 | Tamas Koltai | Process for preparing polymorphic forms of solifenacin succinate |
| JP2010523539A (ja) | 2007-03-30 | 2010-07-15 | メディチェム ソシエダ アノニマ | ソリフェナシンの改良された合成法 |
| JP2009538362A (ja) | 2007-07-13 | 2009-11-05 | テバ ファーマシューティカル インダストリーズ リミティド | ソリフェナシンの調製方法 |
| ITMI20080195A1 (it) | 2008-02-08 | 2009-08-09 | Dipharma Francis Srl | Procedimento per la preparazione di solifenacin |
| WO2009139002A2 (fr) | 2008-05-12 | 2009-11-19 | Msn Laboratories Limited | Procédé perfectionné de fabrication de solifénacine et de ses sels pharmaceutiquement acceptables |
| PL3067353T3 (pl) * | 2008-07-29 | 2018-04-30 | Krka, D.D., Novo Mesto | Sposób wytwarzania soli solifenacyny i ich włączenie do farmaceutycznych postaci dawkowania |
-
2011
- 2011-11-11 WO PCT/EP2011/069969 patent/WO2012062916A1/fr not_active Ceased
- 2011-11-11 EP EP11782419.3A patent/EP2638039A1/fr not_active Withdrawn
- 2011-11-11 CA CA2817336A patent/CA2817336A1/fr not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2012062916A1 (fr) | 2012-05-18 |
| EP2638039A1 (fr) | 2013-09-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Dead |
Effective date: 20161114 |