CA2902436C - Sel d'omecamtiv mecarbil et procede de preparation de sel - Google Patents

Sel d'omecamtiv mecarbil et procede de preparation de sel

Info

Publication number
CA2902436C
CA2902436C CA2902436A CA2902436A CA2902436C CA 2902436 C CA2902436 C CA 2902436C CA 2902436 A CA2902436 A CA 2902436A CA 2902436 A CA2902436 A CA 2902436A CA 2902436 C CA2902436 C CA 2902436C
Authority
CA
Canada
Prior art keywords
omecamtiv mecarbil
salt
radiation
piperazine
mecarbil dihydrochloride
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CA2902436A
Other languages
English (en)
Other versions
CA2902436A1 (fr
Inventor
Sheng Cui
Henry Morrison
Karthik Nagapudi
Shawn Walker
Charles Bernard
Karl Bennett Hansen
Neil Fred Langille
Alan Martin Allgeier
Steven Mennen
Bradley Paul Morgan
Alex Muci
Jacqueline Woo
Original Assignee
Amgen Inc
Cytokinetics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc, Cytokinetics Inc filed Critical Amgen Inc
Priority claimed from PCT/US2014/027146 external-priority patent/WO2014152270A1/fr
Publication of CA2902436A1 publication Critical patent/CA2902436A1/fr
Application granted granted Critical
Publication of CA2902436C publication Critical patent/CA2902436C/fr
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Abstract

L'invention concerne des formes de sel dichlorhydrate d'omécamtiv mécarbil, des compositions et des formulations pharmaceutiques de celles-ci, et des procédés pour leur préparation et utilisation. L'omécamtiv mécarbil (AMG 423, CK-1827452) ayant la structure :
CA2902436A 2013-03-14 2014-03-14 Sel d'omecamtiv mecarbil et procede de preparation de sel Active CA2902436C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361785763P 2013-03-14 2013-03-14
US61/785,763 2013-03-14
PCT/US2014/027146 WO2014152270A1 (fr) 2013-03-14 2014-03-14 Sel d'omécamtiv mécarbil et procédé de préparation de sel

Publications (2)

Publication Number Publication Date
CA2902436A1 CA2902436A1 (fr) 2014-09-25
CA2902436C true CA2902436C (fr) 2024-09-10

Family

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