CA2975682C - Derives de n-acyl-arylsulfonamide comme inhibiteurs d'aminoacyl-arnt synthetase - Google Patents

Derives de n-acyl-arylsulfonamide comme inhibiteurs d'aminoacyl-arnt synthetase

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Publication number
CA2975682C
CA2975682C CA2975682A CA2975682A CA2975682C CA 2975682 C CA2975682 C CA 2975682C CA 2975682 A CA2975682 A CA 2975682A CA 2975682 A CA2975682 A CA 2975682A CA 2975682 C CA2975682 C CA 2975682C
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CA
Canada
Prior art keywords
prov
independently
halo
infection
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CA2975682A
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English (en)
Other versions
CA2975682A1 (fr
Inventor
Aigars Jirgensons
Einars Loza
Michael CHARLTON
Paul William Finn
Lluis Ribas De Pouplana
Adelaide Saint-Leger
Original Assignee
Oxford Drug Design Ltd
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Publication date
Priority claimed from LVP-15-14A external-priority patent/LV15146B/lv
Priority claimed from LVP-16-06A external-priority patent/LV15257A/lv
Application filed by Oxford Drug Design Ltd filed Critical Oxford Drug Design Ltd
Priority claimed from PCT/LV2016/000001 external-priority patent/WO2016129983A1/fr
Publication of CA2975682A1 publication Critical patent/CA2975682A1/fr
Application granted granted Critical
Publication of CA2975682C publication Critical patent/CA2975682C/fr
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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Abstract

La présente invention concerne de nouveaux N-acyl-diarysulfonamides agissant en tant qu'inhibiteurs d'aminoacyl-ARNt synthétase bactérienne. Ces composés peuvent être utilisés en tant que médicaments ou en tant que composant de médicaments pour le traitement d'infections bactériennes.
CA2975682A 2015-02-13 2016-02-11 Derives de n-acyl-arylsulfonamide comme inhibiteurs d'aminoacyl-arnt synthetase Active CA2975682C (fr)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
LVP-15-14A LV15146B (lv) 2015-02-13 2015-02-13 N-acil-diarilsulfonamīda atvasinājumi kā aminoacil-t-RNS sintetāžu inhibitori
LVP-15-14 2015-02-13
LVP-16-06A LV15257A (lv) 2016-02-10 2016-02-10 Jauni N-acil-arilsulfonamīda atvasinājumi kā aminoacil-tRNS sintetāzes inhibitori
LVP-16-06 2016-02-10
PCT/LV2016/000001 WO2016129983A1 (fr) 2015-02-13 2016-02-11 Nouveaux dérivés de n-acyl-arylsulfonamide utilisés en tant qu'inhibiteurs d'aminoacyl-arnt synthétase

Publications (2)

Publication Number Publication Date
CA2975682A1 CA2975682A1 (fr) 2016-08-18
CA2975682C true CA2975682C (fr) 2025-12-09

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