CA3031079C - Radioligands pour l'imagerie de l'enzyme ido1 - Google Patents

Radioligands pour l'imagerie de l'enzyme ido1

Info

Publication number
CA3031079C
CA3031079C CA3031079A CA3031079A CA3031079C CA 3031079 C CA3031079 C CA 3031079C CA 3031079 A CA3031079 A CA 3031079A CA 3031079 A CA3031079 A CA 3031079A CA 3031079 C CA3031079 C CA 3031079C
Authority
CA
Canada
Prior art keywords
ido1
radiolabeled compound
imaging
tissues
pet
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CA3031079A
Other languages
English (en)
Other versions
CA3031079A1 (fr
Inventor
David J. Donnelly
Erin Lee Cole
Richard Charles Burrell
Wesley A. Turley
Alban J. Allentoff
Michael Arthur Wallace
James Aaron Balog
Audris Huang
Mette Skinbjerg
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Priority claimed from PCT/US2017/042510 external-priority patent/WO2018017529A1/fr
Publication of CA3031079A1 publication Critical patent/CA3031079A1/fr
Application granted granted Critical
Publication of CA3031079C publication Critical patent/CA3031079C/fr
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Abstract

La présente invention concerne des inhibiteurs IDO1 radiomarqués ou leurs sels pharmaceutiquement acceptables qui sont utiles pour l'imagerie quantitative des enzymes IDO chez des mammifères.
CA3031079A 2016-07-19 2017-07-18 Radioligands pour l'imagerie de l'enzyme ido1 Active CA3031079C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662364020P 2016-07-19 2016-07-19
US62/364,020 2016-07-19
PCT/US2017/042510 WO2018017529A1 (fr) 2016-07-19 2017-07-18 Radioligands pour l'imagerie de l'enzyme ido1

Publications (2)

Publication Number Publication Date
CA3031079A1 CA3031079A1 (fr) 2018-01-25
CA3031079C true CA3031079C (fr) 2025-11-18

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