CA3085455C - Forme pharmaceutique orale solide comprenant de la linagliptine - Google Patents

Forme pharmaceutique orale solide comprenant de la linagliptine Download PDF

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Publication number
CA3085455C
CA3085455C CA3085455A CA3085455A CA3085455C CA 3085455 C CA3085455 C CA 3085455C CA 3085455 A CA3085455 A CA 3085455A CA 3085455 A CA3085455 A CA 3085455A CA 3085455 C CA3085455 C CA 3085455C
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CA
Canada
Prior art keywords
dosage form
oral dosage
solid oral
weight
linagliptin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
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CA3085455A
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English (en)
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CA3085455A1 (fr
Inventor
Ali Turkyilmaz
Nur Pehlivan Akalin
Merve Ergun Donmez
Original Assignee
Sanovel Ilac Sanayi ve Ticaret AS
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Application filed by Sanovel Ilac Sanayi ve Ticaret AS filed Critical Sanovel Ilac Sanayi ve Ticaret AS
Publication of CA3085455A1 publication Critical patent/CA3085455A1/fr
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Publication of CA3085455C publication Critical patent/CA3085455C/fr
Active legal-status Critical Current
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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La présente invention concerne une forme pharmaceutique orale solide comprenant de la linagliptine et au moins un liant.
CA3085455A 2017-12-15 2018-12-14 Forme pharmaceutique orale solide comprenant de la linagliptine Active CA3085455C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
TR2017/20515 2017-12-15
TR2017/20515A TR201720515A2 (tr) 2017-12-15 2017-12-15 Li̇nagli̇pti̇n i̇çeren bi̇r kati oral dozaj formu
PCT/TR2018/050812 WO2019203755A2 (fr) 2017-12-15 2018-12-14 Forme pharmaceutique orale solide comprenant de la linagliptine

Publications (2)

Publication Number Publication Date
CA3085455A1 CA3085455A1 (fr) 2019-10-24
CA3085455C true CA3085455C (fr) 2022-08-16

Family

ID=67900883

Family Applications (1)

Application Number Title Priority Date Filing Date
CA3085455A Active CA3085455C (fr) 2017-12-15 2018-12-14 Forme pharmaceutique orale solide comprenant de la linagliptine

Country Status (4)

Country Link
EP (1) EP3723761A4 (fr)
CA (1) CA3085455C (fr)
TR (1) TR201720515A2 (fr)
WO (1) WO2019203755A2 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022173406A1 (fr) * 2021-02-15 2022-08-18 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Procédé pour formulations de linagliptine ou d'un sel pharmaceutiquement acceptable de celle-ci
WO2024136773A1 (fr) * 2022-12-21 2024-06-27 Santa Farma Ilac Sanayii A.S. Composition pharmaceutique stable comprenant de la linagliptine
WO2025144125A1 (fr) * 2023-12-27 2025-07-03 Santa Farma Ilac Sanayii A.S. Composition pharmaceutique stable présentant un meilleur profil d'impureté génotoxique

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY32427A (es) * 2009-02-13 2010-09-30 Boheringer Ingelheim Internat Gmbh Composicion farmaceutica, forma farmaceutica, procedimiento para su preparacion, metodos de tratamiento y usos de la misma
WO2013128379A2 (fr) 2012-02-27 2013-09-06 Dr. Reddy's Laboratories Limited Formes polymorphes cristallines de linagliptine
WO2014056942A1 (fr) * 2012-10-09 2014-04-17 Boehringer Ingelheim International Gmbh Utilisation de matière à fabriquer les comprimés dont on ajuste sélectivement l'humidité dans la production de comprimés mécaniquement stables qui contiennent au moins une substance active formant un hydrate et/ou un adjuvant lié à la stabilité mécanique des comprimés, en particulier des comprimés contenant de l'arginine
WO2014080383A1 (fr) * 2012-11-26 2014-05-30 Ranbaxy Laboratories Limited Composition pharmaceutique d'inhibiteurs de la dipeptidyl-peptidase-iv (dpp-iv) en association avec d'autres antidiabétiques
WO2014080384A1 (fr) 2012-11-26 2014-05-30 Ranbaxy Laboratories Limited Composition pharmaceutique de linagliptine
CN106138059A (zh) * 2015-03-27 2016-11-23 天津汉瑞药业有限公司 一种稳定的利格列汀药物组合物
EP3156048A1 (fr) * 2015-10-13 2017-04-19 Galenicum Health S.L. Composition pharmaceutique stable de linagliptine sous forme de comprimé à libération immédiate

Also Published As

Publication number Publication date
CA3085455A1 (fr) 2019-10-24
TR201720515A2 (tr) 2019-07-22
EP3723761A4 (fr) 2021-06-30
WO2019203755A3 (fr) 2020-01-16
WO2019203755A2 (fr) 2019-10-24
EP3723761A2 (fr) 2020-10-21

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EEER Examination request

Effective date: 20200610

EEER Examination request

Effective date: 20200610