CH417576A - Verfahren zur Herstellung von in 6-Stellung halogenierten 1,2a-Methylen- 6-17a-hydroxy-progesteronestern - Google Patents
Verfahren zur Herstellung von in 6-Stellung halogenierten 1,2a-Methylen- 6-17a-hydroxy-progesteronesternInfo
- Publication number
- CH417576A CH417576A CH214862A CH214862A CH417576A CH 417576 A CH417576 A CH 417576A CH 214862 A CH214862 A CH 214862A CH 214862 A CH214862 A CH 214862A CH 417576 A CH417576 A CH 417576A
- Authority
- CH
- Switzerland
- Prior art keywords
- methylene
- hydroxy
- preparation
- progesterone esters
- halogenated
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DESCH29643A DE1158966B (de) | 1961-04-29 | 1961-04-29 | Verfahren zur Herstellung von 6-Chlor-1, 2ª-methylen-í¸-17ª-hydroxyprogesteronestern |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH417576A true CH417576A (de) | 1966-07-31 |
Family
ID=7431494
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH214862A CH417576A (de) | 1961-04-29 | 1962-02-22 | Verfahren zur Herstellung von in 6-Stellung halogenierten 1,2a-Methylen- 6-17a-hydroxy-progesteronestern |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US3234093A (de) |
| BE (1) | BE616989A (de) |
| BR (1) | BR6238435D0 (de) |
| CH (1) | CH417576A (de) |
| DE (1) | DE1158966B (de) |
| GB (1) | GB973908A (de) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1050218A (de) * | 1964-10-13 | |||
| US3401163A (en) * | 1965-10-21 | 1968-09-10 | Squibb & Sons Inc | Preparation of methylene steroids |
| US3423507A (en) * | 1966-02-25 | 1969-01-21 | Schering Corp | Method of treating benign prostratic hypertrophy |
| DE2345377A1 (de) * | 1973-09-06 | 1975-03-20 | Schering Ag | Pharmazeutische zubereitung i |
| GB1570524A (en) * | 1976-03-11 | 1980-07-02 | Unilever Ltd | Cosmetic |
| DE2712861C2 (de) * | 1977-03-21 | 1986-02-27 | Schering AG, 1000 Berlin und 4709 Bergkamen | 17-Acetoxy-6-chlor-15β-hydroxy-1α,2α-methylen-4,6-pregnadien-3,20-dion, Verfahren zu seiner Herstellung und dieses enthaltende Arzneimittel |
| DE3331824A1 (de) * | 1983-09-01 | 1985-03-21 | Schering AG, Berlin und Bergkamen, 1000 Berlin | Verfahren zur herstellung von 17(alpha)-acyloxy-6-chlor-1(alpha),2(alpha)-methylen-3,20-dionen |
| US5439901A (en) * | 1993-07-23 | 1995-08-08 | The Procter & Gamble Company | Cyproterone thiopivalate |
| US5468104A (en) | 1994-08-10 | 1995-11-21 | Fatigue Technology, Inc. | Wall nut assembly |
| US6165504A (en) * | 1998-09-23 | 2000-12-26 | Barr Laboratories, Inc. | Methods for treating hot flashes and improving the quality of life of castrated prostatic cancer patients |
| US6613758B1 (en) | 1999-04-02 | 2003-09-02 | Barr Laboratories, Inc. | Method for treating osteoporosis in castrated prostatic cancer patients |
| EP1359154A1 (de) * | 2002-04-29 | 2003-11-05 | BOEHRINGER INGELHEIM INTERNATIONAL GmbH | Weitere Verfahren zur Herstellung von Cyproteron Azetat |
| US20040024230A1 (en) * | 2002-04-29 | 2004-02-05 | Boehringer Ingelheim International Gmbh | Synthesis of cyproterone acetate |
| US7829552B2 (en) | 2003-11-19 | 2010-11-09 | Metabasis Therapeutics, Inc. | Phosphorus-containing thyromimetics |
| US20060063803A1 (en) * | 2004-09-23 | 2006-03-23 | Pfizer Inc | 4-Amino substituted-2-substituted-1,2,3,4-tetrahydroquinoline compounds |
| US7741317B2 (en) | 2005-10-21 | 2010-06-22 | Bristol-Myers Squibb Company | LXR modulators |
| US7888376B2 (en) | 2005-11-23 | 2011-02-15 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
| US8617597B2 (en) | 2006-07-06 | 2013-12-31 | Bayer Intellectual Property Gmbh | Pharmaceutical composition containing a tetrahydrofolic acid |
| US8404896B2 (en) | 2006-12-01 | 2013-03-26 | Bristol-Myers Squibb Company | N-((3-benzyl)-2,2-(bis-phenyl)-propan-1-amine derivatives as CETP inhibitors for the treatment of atherosclerosis and cardiovascular diseases |
| US20090258040A1 (en) * | 2008-04-09 | 2009-10-15 | Pherin Pharmaceuticals, Inc. | Steroid treatment for hot flashes |
| US20120046364A1 (en) | 2009-02-10 | 2012-02-23 | Metabasis Therapeutics, Inc. | Novel Sulfonic Acid-Containing Thyromimetics, and Methods for Their Use |
| MY176727A (en) | 2012-12-03 | 2020-08-20 | Pfizer | Selective androgen receptor modulators |
-
1961
- 1961-04-29 DE DESCH29643A patent/DE1158966B/de active Pending
-
1962
- 1962-02-22 CH CH214862A patent/CH417576A/de unknown
- 1962-04-11 GB GB14061/62A patent/GB973908A/en not_active Expired
- 1962-04-24 US US189724A patent/US3234093A/en not_active Expired - Lifetime
- 1962-04-25 BR BR138435/62A patent/BR6238435D0/pt unknown
- 1962-04-27 BE BE616989A patent/BE616989A/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE1158966B (de) | 1963-12-12 |
| BR6238435D0 (pt) | 1973-05-24 |
| US3234093A (en) | 1966-02-08 |
| BE616989A (fr) | 1962-10-29 |
| GB973908A (en) | 1964-11-04 |
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