CH443319A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
CH443319A
CH443319A CH1272964A CH1272964A CH443319A CH 443319 A CH443319 A CH 443319A CH 1272964 A CH1272964 A CH 1272964A CH 1272964 A CH1272964 A CH 1272964A CH 443319 A CH443319 A CH 443319A
Authority
CH
Switzerland
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
CH1272964A
Other languages
English (en)
Inventor
Allan Archer Giles
Henryk Sternbach Leo
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH443319A publication Critical patent/CH443319A/de
Priority to CH1013767A priority Critical patent/CH452535A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CH1272964A 1963-10-29 1964-09-30 Verfahren zur Herstellung von Benzodiazepin-Derivaten CH443319A (de)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CH1013767A CH452535A (de) 1963-10-29 1967-09-30 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US319673A US3312688A (en) 1963-10-29 1963-10-29 Process for preparing 2-aminobenzodiazepines

Publications (1)

Publication Number Publication Date
CH443319A true CH443319A (de) 1967-09-15

Family

ID=23243220

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1272964A CH443319A (de) 1963-10-29 1964-09-30 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (14)

Country Link
US (1) US3312688A (de)
BE (1) BE654924A (de)
BR (1) BR6463736D0 (de)
CH (1) CH443319A (de)
DE (2) DE1695217A1 (de)
DK (1) DK114271B (de)
ES (1) ES305413A1 (de)
FR (1) FR1442311A (de)
GB (1) GB1058739A (de)
IL (1) IL22192A (de)
NL (3) NL139527B (de)
NO (1) NO118910B (de)
OA (1) OA00943A (de)
SE (2) SE355580B (de)

Also Published As

Publication number Publication date
SE355580B (de) 1973-04-30
NO118910B (de) 1970-03-02
NL6412484A (de) 1965-05-03
IL22192A (en) 1968-01-25
US3312688A (en) 1967-04-04
ES305413A1 (es) 1965-05-01
BR6463736D0 (pt) 1973-07-17
FR1442311A (fr) 1966-06-17
NL7115681A (de) 1972-02-25
DK114271B (da) 1969-06-16
NL139527B (nl) 1973-08-15
DE1695217A1 (de) 1972-02-17
GB1058739A (en) 1967-02-15
DE1445910A1 (de) 1969-01-23
BE654924A (de) 1965-04-28
NL7115680A (de) 1972-02-25
OA00943A (fr) 1968-03-22
SE329625B (de) 1970-10-19

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